AU2001288658A1 - Screen for glutamate reuptake inhibitors, stimulators, and modulators - Google Patents
Screen for glutamate reuptake inhibitors, stimulators, and modulatorsInfo
- Publication number
- AU2001288658A1 AU2001288658A1 AU2001288658A AU8865801A AU2001288658A1 AU 2001288658 A1 AU2001288658 A1 AU 2001288658A1 AU 2001288658 A AU2001288658 A AU 2001288658A AU 8865801 A AU8865801 A AU 8865801A AU 2001288658 A1 AU2001288658 A1 AU 2001288658A1
- Authority
- AU
- Australia
- Prior art keywords
- receptor
- compound
- glutamate
- compounds
- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- G—PHYSICS
- G01—MEASURING; TESTING
- G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
- G01N33/00—Investigating or analysing materials by specific methods not covered by groups G01N1/00 - G01N31/00
- G01N33/48—Biological material, e.g. blood, urine; Haemocytometers
- G01N33/50—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing
- G01N33/94—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving narcotics or drugs or pharmaceuticals, neurotransmitters or associated receptors
- G01N33/9406—Neurotransmitters
-
- G—PHYSICS
- G01—MEASURING; TESTING
- G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
- G01N2500/00—Screening for compounds of potential therapeutic value
- G01N2500/02—Screening involving studying the effect of compounds C on the interaction between interacting molecules A and B (e.g. A = enzyme and B = substrate for A, or A = receptor and B = ligand for the receptor)
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Molecular Biology (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Urology & Nephrology (AREA)
- Immunology (AREA)
- General Health & Medical Sciences (AREA)
- Hematology (AREA)
- Biomedical Technology (AREA)
- Biotechnology (AREA)
- Physics & Mathematics (AREA)
- Veterinary Medicine (AREA)
- Cell Biology (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Microbiology (AREA)
- Epidemiology (AREA)
- Food Science & Technology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Analytical Chemistry (AREA)
- Biochemistry (AREA)
- General Physics & Mathematics (AREA)
- Pathology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Investigating Or Analysing Biological Materials (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US23015900P | 2000-09-01 | 2000-09-01 | |
| US22995200P | 2000-09-01 | 2000-09-01 | |
| US60230159 | 2000-09-01 | ||
| US60229952 | 2000-09-01 | ||
| PCT/US2001/027323 WO2002018941A2 (fr) | 2000-09-01 | 2001-08-31 | Criblage d'inhibiteurs, de stimulateurs et de modulateurs de recaptage de glutamate |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2001288658A1 true AU2001288658A1 (en) | 2002-03-13 |
Family
ID=26923772
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2001288658A Abandoned AU2001288658A1 (en) | 2000-09-01 | 2001-08-31 | Screen for glutamate reuptake inhibitors, stimulators, and modulators |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US20020115688A1 (fr) |
| EP (1) | EP1314041A2 (fr) |
| AU (1) | AU2001288658A1 (fr) |
| CA (1) | CA2421507A1 (fr) |
| WO (1) | WO2002018941A2 (fr) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2002245137A1 (en) * | 2000-10-30 | 2002-07-24 | Annovis, Inc. | Esters of alkylcarboxy amino acids as prodrugs of modulators of the kainate receptor |
| EP1649009A2 (fr) * | 2003-07-30 | 2006-04-26 | Acucela, Inc. | Culture etendue de cellules retiennes primaires et modeles de stress, ainsi que procedes d'utilisation associes |
| EP2123621A1 (fr) | 2008-05-20 | 2009-11-25 | Bayer Schering Pharma Aktiengesellschaft | Nouveaux acides de glutamine L marqués au {F-18} et dérivés de glutamine L (I), leur utilisation et leur procédé de fabrication |
| JP5529540B2 (ja) * | 2006-11-01 | 2014-06-25 | ピラマル イメージング ソシエテ アノニム | ［ｆ−１８］−ラベルされたｌ−グルタミン酸、［ｆ−１８］−ラベルされたｌ−グルタミン、それらの誘導体、及びそれらの調製のためへのそれらの使用及び方法 |
| EP2123620A1 (fr) * | 2008-05-20 | 2009-11-25 | Bayer Schering Pharma Aktiengesellschaft | Dérivés de l'acide L-glutamique marqué en {F-19} et de L-glutamine (III), leur utilisation et procédé pour les obtenir |
| EP2322171A3 (fr) * | 2009-11-17 | 2011-06-01 | Bayer Schering Pharma Aktiengesellschaft | Dérives de l'acide L-glutamique marqués au fluor |
| US20130149243A1 (en) * | 2009-11-17 | 2013-06-13 | Bayer Intellectual Property Gmbh | Method for production of f-18 labeled glutamic acid derivatives |
| JP2013510894A (ja) * | 2009-11-17 | 2013-03-28 | バイエル・ファルマ・アクチェンゲゼルシャフト | ヨウ素標識のホモグルタミン酸およびグルタミン酸 |
| EP2520556A1 (fr) * | 2011-05-03 | 2012-11-07 | Bayer Pharma Aktiengesellschaft | Acides aminés radiomarqués pour imagerie de diagnostic |
| US9468693B2 (en) * | 2014-01-23 | 2016-10-18 | General Electric Company | Labeled molecular imaging agents and methods of use |
| WO2018132829A1 (fr) * | 2017-01-16 | 2018-07-19 | Drexel University | Nouveaux activateurs de transporteurs de glutamate et procédés les utilisant |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5658782A (en) * | 1993-10-20 | 1997-08-19 | State Of Oregon, Acting By And Through The Oregon State Board Of Higher Education On Behalf Of The Oregon Health Sciences University A Non-Profit Organization | Amino acid transporters and uses |
| CA2216648A1 (fr) * | 1995-02-15 | 1996-08-22 | Bearsden Bio, Inc. | Modulateurs a base d'aminoacides alkylcarboxy du recepteur de kanaite |
-
2001
- 2001-08-31 WO PCT/US2001/027323 patent/WO2002018941A2/fr not_active Ceased
- 2001-08-31 CA CA002421507A patent/CA2421507A1/fr not_active Abandoned
- 2001-08-31 AU AU2001288658A patent/AU2001288658A1/en not_active Abandoned
- 2001-08-31 EP EP01968408A patent/EP1314041A2/fr not_active Withdrawn
- 2001-09-01 US US09/944,954 patent/US20020115688A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| EP1314041A2 (fr) | 2003-05-28 |
| WO2002018941A3 (fr) | 2002-09-26 |
| CA2421507A1 (fr) | 2002-03-07 |
| WO2002018941A2 (fr) | 2002-03-07 |
| US20020115688A1 (en) | 2002-08-22 |
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