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AU2001286237A1 - Oral preparations with favorable disintegration characteristics - Google Patents

Oral preparations with favorable disintegration characteristics

Info

Publication number
AU2001286237A1
AU2001286237A1 AU2001286237A AU8623701A AU2001286237A1 AU 2001286237 A1 AU2001286237 A1 AU 2001286237A1 AU 2001286237 A AU2001286237 A AU 2001286237A AU 8623701 A AU8623701 A AU 8623701A AU 2001286237 A1 AU2001286237 A1 AU 2001286237A1
Authority
AU
Australia
Prior art keywords
water
carmellose
sodium
disintegrant
granule
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2001286237A
Other languages
English (en)
Inventor
Kazuyuki Fujihara
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sumitomo Pharma Co Ltd
Original Assignee
Sumitomo Pharmaceuticals Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=18771855&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU2001286237(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sumitomo Pharmaceuticals Co Ltd filed Critical Sumitomo Pharmaceuticals Co Ltd
Publication of AU2001286237A1 publication Critical patent/AU2001286237A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1617Organic compounds, e.g. phospholipids, fats
    • A61K9/1623Sugars or sugar alcohols, e.g. lactose; Derivatives thereof; Homeopathic globules
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1652Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Zoology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Inorganic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Cosmetics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2001286237A 2000-09-22 2001-09-14 Oral preparations with favorable disintegration characteristics Abandoned AU2001286237A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2000-288234 2000-09-22
JP2000288234 2000-09-22
PCT/JP2001/007983 WO2002024166A1 (fr) 2000-09-22 2001-09-14 Preparations orales dotees de bonnes caracteristiques de desagregation

Publications (1)

Publication Number Publication Date
AU2001286237A1 true AU2001286237A1 (en) 2002-04-02

Family

ID=18771855

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2001286237A Abandoned AU2001286237A1 (en) 2000-09-22 2001-09-14 Oral preparations with favorable disintegration characteristics

Country Status (11)

Country Link
US (1) US7727553B2 (fr)
EP (2) EP1974724A3 (fr)
JP (1) JP4868695B2 (fr)
AT (1) ATE431136T1 (fr)
AU (1) AU2001286237A1 (fr)
CA (2) CA2424001C (fr)
DE (1) DE60138722D1 (fr)
DK (1) DK1327440T5 (fr)
ES (1) ES2325764T3 (fr)
TW (2) TWI289062B (fr)
WO (1) WO2002024166A1 (fr)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2003257589A1 (en) * 2002-08-22 2004-03-11 Sumitomo Pharmaceuticals Company, Limited Remedy for integration dysfunction syndrome
SE0203778D0 (sv) * 2002-12-09 2002-12-09 Astrazeneca Ab A new oral immediated release dosage form
AU2004249621B2 (en) * 2003-06-23 2009-08-06 Dainippon Sumitomo Pharma Co., Ltd. Therapeutic agent for senile dementia
WO2005080976A1 (fr) 2004-02-20 2005-09-01 Dainippon Sumitomo Pharma Co., Ltd. Procédé de recherche par criblage in vivo d'un agent thérapeutique pour un dysfonctionnement de la mémoire/de l'apprentissage par schizophrénie
CN101180046B (zh) 2005-05-18 2011-12-28 大日本住友制药株式会社 含有屈昔多巴的稳定片剂
CN101184489B (zh) 2005-05-26 2011-01-19 大日本住友制药株式会社 药物组合物
KR101328857B1 (ko) * 2005-06-13 2013-11-13 다이닛본 스미토모 세이야꾸 가부시끼가이샤 가용화 제제
JP5366233B2 (ja) * 2005-08-10 2013-12-11 塩野義製薬株式会社 口腔内崩壊錠剤
CN101282717B (zh) * 2005-08-10 2012-07-04 盐野义制药株式会社 苦味抑制制剂
US20090123543A1 (en) * 2006-01-02 2009-05-14 Rubicon Research Private Limited Pharmaceutical compositions
PE20081891A1 (es) * 2007-03-22 2008-12-27 Opko Health Inc Formulaciones de comprimidos que contienen sales de 8-[{1-(3,5-bis-(trifluorometil)fenil)-etoxi}-metil]-8-fenil-1,7-diaza-spiro[4.5]decan-2-ona y comprimidos elaborados a partir de estas
CA2704209C (fr) 2007-10-31 2017-02-28 Mcneil-Ppc, Inc. Forme de dosage a desintegration orale
CA2714524A1 (fr) 2008-02-11 2009-08-20 Makiko Yanagida Comprime presentant des proprietes d'elution ameliorees
JP5583012B2 (ja) 2008-06-13 2014-09-03 大日本住友製薬株式会社 口腔内速崩壊錠及びその製造方法
CN102238941A (zh) * 2008-09-17 2011-11-09 迈兰实验室公司 颗粒、制备它们的方法和包含它们的药物产品
US20110318411A1 (en) 2010-06-24 2011-12-29 Luber Joseph R Multi-layered orally disintegrating tablet and the manufacture thereof
US8343533B2 (en) 2009-09-24 2013-01-01 Mcneil-Ppc, Inc. Manufacture of lozenge product with radiofrequency
US8258139B2 (en) 2010-11-08 2012-09-04 Dainippon Sumitomo Pharma Co., Ltd. Method of treatment for mental disorders
WO2012107890A2 (fr) * 2011-02-10 2012-08-16 Ranbaxy Laboratories Limited Formes cristallines de chlorhydrate de lurasidone
US9433620B2 (en) * 2011-05-13 2016-09-06 Cadila Healthcare Limited Pharmaceutical compositions of lurasidone
CN104321013B (zh) 2012-03-21 2017-08-15 皇家飞利浦有限公司 用于基于ecg信号来提供睡眠质量的视觉表示的方法和装置
US9445971B2 (en) 2012-05-01 2016-09-20 Johnson & Johnson Consumer Inc. Method of manufacturing solid dosage form
US9511028B2 (en) 2012-05-01 2016-12-06 Johnson & Johnson Consumer Inc. Orally disintegrating tablet
US9233491B2 (en) 2012-05-01 2016-01-12 Johnson & Johnson Consumer Inc. Machine for production of solid dosage forms
JP6007169B2 (ja) * 2012-11-30 2016-10-12 大原薬品工業株式会社 アリピプラゾール無水物を含有する固形製剤の製造方法
WO2014090386A1 (fr) 2012-12-11 2014-06-19 Alfred E. Tiefenbacher (Gmbh & Co. Kg) Comprimé à désintégration orale contenant de l'asénapine
JP2014129238A (ja) * 2012-12-28 2014-07-10 Lion Corp エトドラク含有固形製剤
JP6037824B2 (ja) * 2012-12-28 2016-12-07 ライオン株式会社 エトドラク含有固形製剤
EP3091966B1 (fr) 2014-01-10 2019-07-31 Johnson & Johnson Consumer Inc. Procédé pour fabriquer un comprimé par radiofréquence et particules revêtues à perte
WO2016012898A1 (fr) 2014-07-25 2016-01-28 Lupin Limited Composition pharmaceutique orale de lurasidone
WO2016139683A2 (fr) * 2015-03-05 2016-09-09 Jubilant Generics Limited Compositions pharmaceutiques de lurasidone et son procédé de préparation
US10966928B2 (en) 2016-03-25 2021-04-06 Universiteit Gent Oral dosage form
ES2883352T3 (es) 2016-03-25 2021-12-07 Univ Gent Forma de dosificación oral
US11413295B2 (en) 2016-03-31 2022-08-16 Intercept Pharmaceuticals, Inc. Oral preparation of obeticholic acid
JPWO2018043613A1 (ja) * 2016-08-31 2019-06-24 大日本住友製薬株式会社 水性懸濁型製剤
WO2018130943A1 (fr) 2017-01-11 2018-07-19 Piramal Enterprises Limited Composition pharmaceutique orale de lurasidone et sa préparation
US10493026B2 (en) 2017-03-20 2019-12-03 Johnson & Johnson Consumer Inc. Process for making tablet using radiofrequency and lossy coated particles
AT17300U3 (de) * 2020-12-03 2022-02-15 G L Pharma Gmbh Feste orale pharmazeutische Zusammensetzung
WO2023078366A1 (fr) * 2021-11-04 2023-05-11 上海博志研新药物技术有限公司 Composition de film orale soluble de chlorhydrate de lurasidone, procédé de préparation et utilisation associés

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JP2800953B2 (ja) 1990-07-06 1998-09-21 住友製薬株式会社 新規なイミド誘導体
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US5972383A (en) * 1994-03-02 1999-10-26 Eli Lilly And Company Solid orally administerable raloxifene hydrochloride pharmaceutical formulation
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US5994348A (en) 1995-06-07 1999-11-30 Sanofi Pharmaceutical compositions containing irbesartan
US5958453A (en) * 1996-10-31 1999-09-28 Takeda Chemical Industries, Ltd. Solid pharmaceutical preparation with improved buccal disintegrability and/or dissolubility
TW482675B (en) 1997-01-31 2002-04-11 Green Cross Corp Compositions for oral administration containing pyridazinone compounds technical field of the invention
NZ505123A (en) 1997-12-19 2003-07-25 Smithkline Beecham Corp Process for manufacturing bite-dispersion tablets by compressing medicaments and other ingredients into granulates then compressing the granulates and other ingredients into tablets, and the tablets thereof
US6465009B1 (en) * 1998-03-18 2002-10-15 Yamanouchi Pharmaceutical Co., Ltd. Water soluble polymer-based rapidly dissolving tablets and production processes thereof
JP4438121B2 (ja) * 1998-04-27 2010-03-24 大正製薬株式会社 口腔内速崩錠及びその製造方法
KR100267576B1 (ko) * 1998-07-25 2000-11-01 허계성 활성성분을 분리함유한 츄잉 연질정제 및 그의 제조방법
JP2000086503A (ja) 1998-09-07 2000-03-28 Pola Chem Ind Inc 錠剤医薬組成物
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Also Published As

Publication number Publication date
DE60138722D1 (de) 2009-06-25
CA2824077A1 (fr) 2002-03-28
TWI289062B (en) 2007-11-01
DK1327440T5 (da) 2009-09-07
US7727553B2 (en) 2010-06-01
ATE431136T1 (de) 2009-05-15
ES2325764T3 (es) 2009-09-16
EP1327440A1 (fr) 2003-07-16
JPWO2002024166A1 (ja) 2004-01-29
CA2424001A1 (fr) 2003-03-20
EP1327440B1 (fr) 2009-05-13
CA2824077C (fr) 2016-01-26
TW200524642A (en) 2005-08-01
EP1327440A4 (fr) 2006-02-01
CA2424001C (fr) 2013-10-22
EP1974724A2 (fr) 2008-10-01
DK1327440T3 (da) 2009-06-08
JP4868695B2 (ja) 2012-02-01
US20040028741A1 (en) 2004-02-12
WO2002024166A1 (fr) 2002-03-28
EP1974724A3 (fr) 2008-11-12
TWI289063B (en) 2007-11-01

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