AU2001278980A1 - Coumarin derivatives useful as tnfalpha inhibitors - Google Patents
Coumarin derivatives useful as tnfalpha inhibitorsInfo
- Publication number
- AU2001278980A1 AU2001278980A1 AU2001278980A AU7898001A AU2001278980A1 AU 2001278980 A1 AU2001278980 A1 AU 2001278980A1 AU 2001278980 A AU2001278980 A AU 2001278980A AU 7898001 A AU7898001 A AU 7898001A AU 2001278980 A1 AU2001278980 A1 AU 2001278980A1
- Authority
- AU
- Australia
- Prior art keywords
- derivatives useful
- coumarin derivatives
- tnfalpha inhibitors
- tnfalpha
- inhibitors
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/365—Lactones
- A61K31/366—Lactones having six-membered rings, e.g. delta-lactones
- A61K31/37—Coumarins, e.g. psoralen
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
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Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US22004800P | 2000-07-21 | 2000-07-21 | |
| US60220048 | 2000-07-21 | ||
| US22544800P | 2000-08-14 | 2000-08-14 | |
| US60225448 | 2000-08-14 | ||
| US30303001P | 2001-07-03 | 2001-07-03 | |
| US60303030 | 2001-07-03 | ||
| PCT/US2001/022950 WO2002008217A2 (en) | 2000-07-21 | 2001-07-19 | COUMARIN DERIVATIVES USEFUL AS TNFα INHIBITORS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2001278980A1 true AU2001278980A1 (en) | 2002-02-05 |
Family
ID=27396753
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2001278980A Abandoned AU2001278980A1 (en) | 2000-07-21 | 2001-07-19 | Coumarin derivatives useful as tnfalpha inhibitors |
Country Status (4)
| Country | Link |
|---|---|
| US (4) | US7026491B2 (en) |
| JP (1) | JP4890723B2 (en) |
| AU (1) | AU2001278980A1 (en) |
| WO (1) | WO2002008217A2 (en) |
Families Citing this family (36)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2003105842A1 (en) * | 2002-06-13 | 2003-12-24 | Novuspharma S.P.A. | Derivatives of chromen-2-one as inhibitors of vegf production in mammalian cells |
| AR059339A1 (en) * | 2006-02-09 | 2008-03-26 | Chugai Pharmaceutical Co Ltd | CUMARINE DERIVATIVES FOR PROLIFERATIVE DISORDERS OF CELLS, PHARMACEUTICAL COMPOSITION AND THERAPEUTIC AGENT CONTAINING THEM |
| EP2172198B1 (en) | 2007-07-20 | 2014-04-16 | Chugai Seiyaku Kabushiki Kaisha | p27 PROTEIN INDUCER |
| JP2009084269A (en) * | 2007-09-05 | 2009-04-23 | Sumitomo Chemical Co Ltd | Coumarin compounds and their uses |
| US20100114768A1 (en) | 2008-10-31 | 2010-05-06 | Wachovia Corporation | Payment vehicle with on and off function |
| US10867298B1 (en) | 2008-10-31 | 2020-12-15 | Wells Fargo Bank, N.A. | Payment vehicle with on and off function |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH522631A (en) | 1961-08-12 | 1972-06-30 | Cassella Farbwerke Mainkur Ag | 7-hydroxy-coumarin derivs |
| US3259635A (en) * | 1962-07-26 | 1966-07-05 | Cassella Farbwerke Mainkur Ag | 7-hydroxy coumarin derivative |
| DE3427985A1 (en) * | 1984-07-28 | 1986-01-30 | Boehringer Mannheim Gmbh, 6800 Mannheim | NEW 2H-L-BENZOPYRAN-2-ON DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND MEDICINAL PRODUCTS CONTAINING THESE COMPOUNDS |
| DE59010069D1 (en) | 1989-11-21 | 1996-02-29 | Bayer Ag | Coumarin derivatives, processes for their preparation, their use and thiazolyl acetic acid derivatives as intermediates |
| GB9109645D0 (en) | 1991-05-03 | 1991-06-26 | Celltech Ltd | Recombinant antibodies |
| WO1996031206A2 (en) * | 1995-04-07 | 1996-10-10 | Warner-Lambert Company | Flavones and coumarins as agents for the treatment of atherosclerosis |
| WO1999015523A1 (en) | 1997-09-24 | 1999-04-01 | Orion Corporation | Bisethers of 1-oxa, aza and thianaphthalen-2-ones as phospholamban inhibitors |
-
2001
- 2001-07-19 JP JP2002514123A patent/JP4890723B2/en not_active Expired - Lifetime
- 2001-07-19 WO PCT/US2001/022950 patent/WO2002008217A2/en not_active Ceased
- 2001-07-19 US US10/333,366 patent/US7026491B2/en not_active Expired - Lifetime
- 2001-07-19 AU AU2001278980A patent/AU2001278980A1/en not_active Abandoned
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2005
- 2005-09-13 US US11/225,940 patent/US7709664B2/en not_active Expired - Lifetime
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2010
- 2010-03-18 US US12/727,053 patent/US7994318B2/en not_active Expired - Fee Related
- 2010-03-18 US US12/726,986 patent/US7872142B2/en not_active Expired - Fee Related
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| WO2002008217A2 (en) | 2002-01-31 |
| US7026491B2 (en) | 2006-04-11 |
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| WO2002008217A3 (en) | 2002-04-18 |
| US20050014705A1 (en) | 2005-01-20 |
| JP4890723B2 (en) | 2012-03-07 |
| US7994318B2 (en) | 2011-08-09 |
| JP2004509855A (en) | 2004-04-02 |
| US7872142B2 (en) | 2011-01-18 |
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