ATE527264T1 - Kondensierte heterozyklische verbindungen als hemmer von proteinkinasen - Google Patents
Kondensierte heterozyklische verbindungen als hemmer von proteinkinasenInfo
- Publication number
- ATE527264T1 ATE527264T1 AT08780617T AT08780617T ATE527264T1 AT E527264 T1 ATE527264 T1 AT E527264T1 AT 08780617 T AT08780617 T AT 08780617T AT 08780617 T AT08780617 T AT 08780617T AT E527264 T1 ATE527264 T1 AT E527264T1
- Authority
- AT
- Austria
- Prior art keywords
- inhibitors
- heterocyclic compounds
- protein kinases
- condensed heterocyclic
- compounds
- Prior art date
Links
- 102000001253 Protein Kinase Human genes 0.000 title 1
- 150000002391 heterocyclic compounds Chemical class 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
- 108060006633 protein kinase Proteins 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 102000003989 Aurora kinases Human genes 0.000 abstract 1
- 108090000433 Aurora kinases Proteins 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US91684607P | 2007-05-09 | 2007-05-09 | |
| US91683807P | 2007-05-09 | 2007-05-09 | |
| PCT/US2008/063197 WO2008141145A1 (en) | 2007-05-09 | 2008-05-09 | Condensed heterocyclic compounds as inhibitors of protein kinases |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE527264T1 true ATE527264T1 (de) | 2011-10-15 |
Family
ID=39650562
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT08780617T ATE527264T1 (de) | 2007-05-09 | 2008-05-09 | Kondensierte heterozyklische verbindungen als hemmer von proteinkinasen |
Country Status (8)
| Country | Link |
|---|---|
| EP (1) | EP2150553B1 (de) |
| JP (1) | JP5412424B2 (de) |
| CN (1) | CN101730700A (de) |
| AT (1) | ATE527264T1 (de) |
| CA (1) | CA2685351A1 (de) |
| ES (1) | ES2372559T3 (de) |
| MX (1) | MX2009012079A (de) |
| WO (1) | WO2008141145A1 (de) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8624027B2 (en) | 2005-05-12 | 2014-01-07 | Abbvie Inc. | Combination therapy for treating cancer and diagnostic assays for use therein |
| US8124759B2 (en) | 2007-05-09 | 2012-02-28 | Abbott Laboratories | Inhibitors of protein kinases |
| CN102532042A (zh) * | 2010-12-30 | 2012-07-04 | 上海医药工业研究院 | 一种芳基脲类化合物、其中间体及其应用 |
| KR20150061651A (ko) * | 2012-09-26 | 2015-06-04 | 더 리젠츠 오브 더 유니버시티 오브 캘리포니아 | Ire1의 조절 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BRPI0415395A (pt) * | 2003-10-15 | 2006-12-12 | Osi Pharm Inc | composto, métodos para inibir a atividade da proteìna quinase e para tratar um paciente que tenha uma condição que seja mediada pela atividade da proteìna quinase, e, composição |
| AR048518A1 (es) * | 2004-04-02 | 2006-05-03 | Osi Pharm Inc | Inhibidores heterobiciclicos de proteina quinasas sustituidos con anillos 6,6 -biciclicos |
| US7776865B2 (en) * | 2005-10-06 | 2010-08-17 | Schering Corporation | Substituted pyrazolo[1,5-a]pyrimidines as protein kinase inhibitors |
| CA2630271C (en) * | 2005-11-17 | 2014-04-08 | Osi Pharmaceuticals, Inc. | Fused bicyclic mtor inhibitors |
| AR057960A1 (es) * | 2005-12-02 | 2007-12-26 | Osi Pharm Inc | Inhibidores de proteina quinasa biciclicos |
| WO2007087395A2 (en) * | 2006-01-25 | 2007-08-02 | Osi Pharmaceuticals, Inc. | UNSATURATED mTOR INHIBITORS |
| EP1996193A2 (de) * | 2006-03-13 | 2008-12-03 | OSI Pharmaceuticals, Inc. | Kombinierte behandlung mit einem egfr-kinase-hemmber und einem wirkstoff, der tumorzellen für die wirkung von egfr-kinase-hemmern sensibilisiert |
-
2008
- 2008-05-09 ES ES08780617T patent/ES2372559T3/es active Active
- 2008-05-09 CA CA002685351A patent/CA2685351A1/en not_active Abandoned
- 2008-05-09 AT AT08780617T patent/ATE527264T1/de not_active IP Right Cessation
- 2008-05-09 WO PCT/US2008/063197 patent/WO2008141145A1/en not_active Ceased
- 2008-05-09 MX MX2009012079A patent/MX2009012079A/es active IP Right Grant
- 2008-05-09 CN CN200880023583A patent/CN101730700A/zh active Pending
- 2008-05-09 EP EP08780617A patent/EP2150553B1/de active Active
- 2008-05-09 JP JP2010507687A patent/JP5412424B2/ja not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| CA2685351A1 (en) | 2008-11-20 |
| MX2009012079A (es) | 2009-11-19 |
| JP5412424B2 (ja) | 2014-02-12 |
| JP2010526833A (ja) | 2010-08-05 |
| EP2150553B1 (de) | 2011-10-05 |
| EP2150553A1 (de) | 2010-02-10 |
| ES2372559T3 (es) | 2012-01-23 |
| CN101730700A (zh) | 2010-06-09 |
| WO2008141145A1 (en) | 2008-11-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |