ATE243695T1 - 5-bicycloindolverbindungen - Google Patents
5-bicycloindolverbindungenInfo
- Publication number
- ATE243695T1 ATE243695T1 AT99930958T AT99930958T ATE243695T1 AT E243695 T1 ATE243695 T1 AT E243695T1 AT 99930958 T AT99930958 T AT 99930958T AT 99930958 T AT99930958 T AT 99930958T AT E243695 T1 ATE243695 T1 AT E243695T1
- Authority
- AT
- Austria
- Prior art keywords
- compounds
- bicycloindole
- disclosed
- ht1d receptor
- migrane
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 4
- 101710138068 5-hydroxytryptamine receptor 1D Proteins 0.000 abstract 2
- 239000003814 drug Substances 0.000 abstract 1
- 230000000638 stimulation Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pain & Pain Management (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Indole Compounds (AREA)
- Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US09/116,946 US6329390B1 (en) | 1998-07-17 | 1998-07-17 | 5-Bicycloindole compounds |
| PCT/CA1999/000639 WO2000004019A1 (en) | 1998-07-17 | 1999-07-15 | 5-bicycloindole compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE243695T1 true ATE243695T1 (de) | 2003-07-15 |
Family
ID=22370203
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT99930958T ATE243695T1 (de) | 1998-07-17 | 1999-07-15 | 5-bicycloindolverbindungen |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US6329390B1 (de) |
| EP (1) | EP1098896B1 (de) |
| JP (1) | JP2002520412A (de) |
| AT (1) | ATE243695T1 (de) |
| AU (1) | AU767274B2 (de) |
| CA (1) | CA2343748A1 (de) |
| DE (1) | DE69909097D1 (de) |
| WO (1) | WO2000004019A1 (de) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2666772B1 (de) * | 2002-12-20 | 2017-03-01 | Basf Se | Synthese von Aminen und Zwischenverbindungen für die Synthese davon |
| CN102936240A (zh) * | 2012-10-30 | 2013-02-20 | 浙江省医学科学院 | 一种(r)-5-取代-3-(n-苄氧羰基吡咯烷-2-基羰基)-1h-吲哚的合成方法 |
| WO2025104490A1 (en) * | 2023-11-14 | 2025-05-22 | Mindset Pharma Inc. | Indole derivatives as serotonergic agents useful for the treatment of disorders related thereto |
| WO2025104491A1 (en) * | 2023-11-14 | 2025-05-22 | Mindset Pharma Inc. | Indole derivatives as serotonergic agents useful for the treatment of disorders related thereto |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9407447D0 (en) * | 1994-04-14 | 1994-06-08 | Glaxo Group Ltd | Chemical compounds |
| WO1998023587A1 (en) * | 1996-11-26 | 1998-06-04 | Allelix Biopharmaceuticals Inc. | 5-cyclo indole compounds as 5-ht1d receptor ligands |
-
1998
- 1998-07-17 US US09/116,946 patent/US6329390B1/en not_active Expired - Fee Related
-
1999
- 1999-07-15 JP JP2000560125A patent/JP2002520412A/ja active Pending
- 1999-07-15 AU AU47651/99A patent/AU767274B2/en not_active Ceased
- 1999-07-15 DE DE69909097T patent/DE69909097D1/de not_active Expired - Lifetime
- 1999-07-15 EP EP99930958A patent/EP1098896B1/de not_active Expired - Lifetime
- 1999-07-15 CA CA002343748A patent/CA2343748A1/en not_active Abandoned
- 1999-07-15 AT AT99930958T patent/ATE243695T1/de not_active IP Right Cessation
- 1999-07-15 WO PCT/CA1999/000639 patent/WO2000004019A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| AU4765199A (en) | 2000-02-07 |
| US6329390B1 (en) | 2001-12-11 |
| EP1098896B1 (de) | 2003-06-25 |
| JP2002520412A (ja) | 2002-07-09 |
| EP1098896A1 (de) | 2001-05-16 |
| DE69909097D1 (de) | 2003-07-31 |
| AU767274B2 (en) | 2003-11-06 |
| WO2000004019A1 (en) | 2000-01-27 |
| CA2343748A1 (en) | 2000-01-27 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |