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AR113688A1 - Proceso para la preparación de compuestos de piridiminio ópticamente activo - Google Patents

Proceso para la preparación de compuestos de piridiminio ópticamente activo

Info

Publication number
AR113688A1
AR113688A1 ARP180101083A ARP180101083A AR113688A1 AR 113688 A1 AR113688 A1 AR 113688A1 AR P180101083 A ARP180101083 A AR P180101083A AR P180101083 A ARP180101083 A AR P180101083A AR 113688 A1 AR113688 A1 AR 113688A1
Authority
AR
Argentina
Prior art keywords
compounds
optically active
pyridiminium
preparation
unsubstituted
Prior art date
Application number
ARP180101083A
Other languages
English (en)
Original Assignee
Basf Se
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Se filed Critical Basf Se
Publication of AR113688A1 publication Critical patent/AR113688A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F15/00—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
    • C07F15/0006—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table compounds of the platinum group
    • C07F15/0033—Iridium compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F15/00—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
    • C07F15/0006—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table compounds of the platinum group
    • C07F15/0046—Ruthenium compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F15/00—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
    • C07F15/0006—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table compounds of the platinum group
    • C07F15/0073—Rhodium compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Thiazole And Isothizaole Compounds (AREA)

Abstract

Un proceso para preparar un compuesto de pirimidinio ópticamente activo de la fórmula (1) y sus intermediarios, en donde: C* es un átomo de carbono asimétrico de configuración S o R; R¹ es C₁₋₄-alquilo, C₃₋₆-cicloalquilo, C₂₋₄-alquenilo o -CH₂-fenilo, en donde los grupos son no sustituidos o sustituidos con halógeno o C₁₋₄-alquilo; R² es un anillo carbocíclico o heterocíclico saturado, parcialmente insaturado o aromático de 5 ó 6 miembros, en donde el anillo es no sustituido o sustituido con R²ᵃ; Het se selecciona de los compuestos de fórmula (2), (3) y (4).
ARP180101083A 2017-04-27 2018-04-26 Proceso para la preparación de compuestos de piridiminio ópticamente activo AR113688A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP17168354 2017-04-27

Publications (1)

Publication Number Publication Date
AR113688A1 true AR113688A1 (es) 2020-06-03

Family

ID=58638745

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP180101083A AR113688A1 (es) 2017-04-27 2018-04-26 Proceso para la preparación de compuestos de piridiminio ópticamente activo

Country Status (13)

Country Link
US (1) US11124528B2 (es)
EP (1) EP3615543B1 (es)
JP (1) JP7263250B2 (es)
KR (1) KR102591738B1 (es)
CN (1) CN110546153B (es)
AR (1) AR113688A1 (es)
AU (1) AU2018260180B2 (es)
CA (1) CA3058083A1 (es)
IL (1) IL270134B (es)
MX (1) MX394953B (es)
MY (1) MY199348A (es)
PH (1) PH12019502286A1 (es)
WO (1) WO2018197541A1 (es)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2019011785A (es) * 2017-03-31 2019-11-18 Basf Se Proceso para preparar compuestos de 2,3-dihidrotiazolo[3,2-a]pirim idin-4-io quirales.
EP3619217B1 (en) 2017-05-03 2021-07-07 Basf Se Process for preparing chiral 2,3-dihydrothiazolo[3,2-a]pyrimidin-4-ium compounds
BR112019025191B1 (pt) 2017-06-19 2023-11-28 Basf Se Compostos de pirimidínio substituídos, composição, método para proteger culturas, semente revestida, uso dos compostos e uso de um composto
EP3704086B1 (en) 2017-11-02 2024-02-21 Basf Se Process for preparing 4-chlorobenzyl propargyl ether
CN110041365B (zh) * 2018-12-05 2020-12-22 华东师范大学 吡咯啉类手性双膦配体及其制备方法和应用
US11187127B2 (en) 2019-06-28 2021-11-30 Deere & Company Exhaust gas treatment system and method with four-way catalyzed filter element
AU2020360778A1 (en) * 2019-10-04 2022-04-14 Basf Se Preparation of 2-chloro-1-(2-chlorothiazol-5-yl)ethanone
WO2021130143A1 (en) * 2019-12-23 2021-07-01 Basf Se Enzyme enhanced root uptake of agrochemical active compound
EP3974417A1 (en) 2020-09-29 2022-03-30 Basf Se Preparation of 2-chloro-1-(2-chlorothiazol-5-yl)ethanone
EP4032893A1 (en) 2021-01-22 2022-07-27 Basf Se Method for preparing an enantiomerically enriched form of 3-(2-chlorothiazol-5-yl)-8-methyl-7-oxo-6-phenyl-2,3-dihydrothiazolo[3,2-a]pyrimidin-4-ium-5-olate
EP4032886A1 (en) * 2021-01-22 2022-07-27 Basf Se Method for preparing an enantiomerically enriched form of 2-[2-(2-chlorothiazol-5-yl)-2-hydroxy-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one
EP4032878A1 (en) 2021-01-22 2022-07-27 Basf Se Method for preparing 2-[2-(2-chlorothiazol-5-yl)-2-oxo-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one
EP4032894A1 (en) * 2021-01-22 2022-07-27 Basf Se Method for preparing an enantiomerically enriched form of 3-(2-chlorothiazol-5-yl)-8-methyl-7-oxo-6-phenyl-2,3-dihydrothiazolo[3,2-a]pyrimidin-4-ium-5-olate
EP4063362A1 (en) 2021-03-25 2022-09-28 Basf Se Method for preparing enantiomerically enriched 2-[2-(2-chlorothiazol-5-yl)-2-hydroxy-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one by hydrogenation of the 2-oxo derivative in the presence of a chiral transition metal catalyst
WO2025223938A1 (en) 2024-04-26 2025-10-30 Basf Se Method for preparing an enantiomerically enriched form of 2-[2-(2-chlorothiazol-5-yl)-2- hydroxy-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one
WO2025252510A1 (en) 2024-06-04 2025-12-11 Basf Se Method for preparing an enantiomerically enriched form of 2-[2-(2-chlorothiazol-5-yl)-2-hydroxy-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9019095D0 (en) * 1990-09-01 1990-10-17 Beecham Group Plc Novel compounds
UA107804C2 (en) * 2009-08-05 2015-02-25 Du Pont Mixtures of pesticides mezoionnyh
MX2012001646A (es) * 2009-08-05 2012-03-21 Du Pont Pesticidas mesoionicos.
WO2013076092A1 (en) * 2011-11-21 2013-05-30 Basf Se Process for preparing n-substituted 1h-pyrazole-5-carboxylate compounds and derivatives thereof
MX366855B (es) 2013-03-01 2019-07-26 Amgen Inc Compuestos perfluorados de 5,6-dihidro-4h-1,3-oxazin-2-amina como inhibidores de beta-secretasa y metodos de uso.
AR096022A1 (es) * 2013-04-11 2015-12-02 Basf Se Compuestos de pirimidinio sustituido, útiles para combatir plagas de animales
BR112017005140A2 (pt) * 2014-10-06 2018-01-23 Basf Se compostos, mistura, composição, métodos para a proteção de culturas e para o combate ou controle de praga de invertebrados, método não terapêutico para o tratamento de animais infestados ou infectados por parasitas e semente
EP3619217B1 (en) * 2017-05-03 2021-07-07 Basf Se Process for preparing chiral 2,3-dihydrothiazolo[3,2-a]pyrimidin-4-ium compounds

Also Published As

Publication number Publication date
AU2018260180A1 (en) 2019-10-31
MX2019012815A (es) 2020-01-14
US20200055872A1 (en) 2020-02-20
JP7263250B2 (ja) 2023-04-24
EP3615543A1 (en) 2020-03-04
KR20190141711A (ko) 2019-12-24
CN110546153B (zh) 2022-09-06
CA3058083A1 (en) 2018-11-01
US11124528B2 (en) 2021-09-21
MX394953B (es) 2025-03-24
MY199348A (en) 2023-10-24
EP3615543B1 (en) 2021-10-20
JP2020517684A (ja) 2020-06-18
AU2018260180B2 (en) 2021-12-09
KR102591738B1 (ko) 2023-10-19
IL270134B (en) 2022-05-01
BR112019021122A2 (pt) 2020-05-12
CN110546153A (zh) 2019-12-06
WO2018197541A1 (en) 2018-11-01
PH12019502286A1 (en) 2020-09-14

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