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AR112276A1 - 5-FLUORO-4-IMINO-3-METHYL-1-TOSIL-3,4-DIHYDROPYRIMIDIN-2-ONA POLYMORPHES - Google Patents

5-FLUORO-4-IMINO-3-METHYL-1-TOSIL-3,4-DIHYDROPYRIMIDIN-2-ONA POLYMORPHES

Info

Publication number
AR112276A1
AR112276A1 ARP180101983A AR112276A1 AR 112276 A1 AR112276 A1 AR 112276A1 AR P180101983 A ARP180101983 A AR P180101983A AR 112276 A1 AR112276 A1 AR 112276A1
Authority
AR
Argentina
Prior art keywords
tosil
polymorphes
dihydropyrimidin
ona
imino
Prior art date
Application number
Other languages
Spanish (es)
Inventor
Zoltn Nmet
Gal Suez
Michael Grabarnick
Original Assignee
Adama Makhteshim Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adama Makhteshim Ltd filed Critical Adama Makhteshim Ltd
Publication of AR112276A1 publication Critical patent/AR112276A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P3/00—Fungicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Engineering & Computer Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Environmental Sciences (AREA)
  • Plant Pathology (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Microbiology (AREA)
  • Mycology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente materia proporciona una forma cristalina del compuesto que tiene la estructura de fórmula (1), en donde la forma cristalina es un polimorfo, un hidrato o un solvato. Uso como plaguicidas o fungicidas.The present matter provides a crystalline form of the compound having the structure of formula (1), wherein the crystalline form is a polymorph, a hydrate or a solvate. Use as pesticides or fungicides.

ARP180101983 2017-07-17 2018-07-17 5-FLUORO-4-IMINO-3-METHYL-1-TOSIL-3,4-DIHYDROPYRIMIDIN-2-ONA POLYMORPHES AR112276A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201762533509P 2017-07-17 2017-07-17

Publications (1)

Publication Number Publication Date
AR112276A1 true AR112276A1 (en) 2019-10-09

Family

ID=63517924

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP180101983 AR112276A1 (en) 2017-07-17 2018-07-17 5-FLUORO-4-IMINO-3-METHYL-1-TOSIL-3,4-DIHYDROPYRIMIDIN-2-ONA POLYMORPHES

Country Status (11)

Country Link
US (1) US11632954B2 (en)
EP (1) EP3655396A1 (en)
JP (3) JP2020527563A (en)
CN (2) CN118515619A (en)
AR (1) AR112276A1 (en)
AU (1) AU2018320492C1 (en)
CA (1) CA3069619A1 (en)
IL (5) IL271950B2 (en)
MA (1) MA49639A (en)
WO (1) WO2019038583A1 (en)
ZA (1) ZA202000411B (en)

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IL321760A (en) 2019-07-22 2025-08-01 Adama Makhteshim Ltd Fungicidal combinations, mixtures and preparations and their uses
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CA3206570A1 (en) 2021-01-27 2022-08-04 Alexandra ROSENMUND 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1 h)-one for controlling plant diseases
CA3216622A1 (en) 2021-05-04 2022-11-10 Stefano Luca Giaffreda Crystalline forms of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4- dihydropyrimidin-2-one, and mixtures, compositions and methods of use thereof
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AU2023275068A1 (en) 2022-05-26 2024-11-28 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
AR130107A1 (en) 2022-08-03 2024-11-06 Adama Makhteshim Ltd 5-FLUORO-4-IMINO-3-METHYL-1-TOSYL-3,4-DIHYDROPYRIMIDIN-2(1H)-ONE FOR FUNGICIDE-RESISTANT FUNGI
AU2024233301A1 (en) 2023-03-09 2025-09-18 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
WO2024189563A1 (en) 2023-03-14 2024-09-19 Adama Makhteshim Ltd. Liquid compositions containing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1h)-one and derivatives thereof and a uv absorber
AR132381A1 (en) 2023-04-11 2025-06-18 Adama Makhteshim Ltd COMPOUNDS AND PROCESSES RELATED TO FLUMETHYLSULFORIM
AR133680A1 (en) 2023-08-31 2025-10-22 Adama Makhteshim Ltd FUNGICIDAL COMBINATIONS, MIXTURES AND COMPOSITIONS AND THEIR USES
WO2025114931A1 (en) 2023-11-28 2025-06-05 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof

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Also Published As

Publication number Publication date
WO2019038583A1 (en) 2019-02-28
IL323266A (en) 2025-11-01
NZ761039A (en) 2023-09-29
JP2023145572A (en) 2023-10-11
IL323268A (en) 2025-11-01
EP3655396A1 (en) 2020-05-27
AU2018320492C1 (en) 2023-07-13
AU2018320492A1 (en) 2020-02-13
IL271950B1 (en) 2024-02-01
IL271950B2 (en) 2024-06-01
MA49639A (en) 2020-05-27
US20200229437A1 (en) 2020-07-23
US11632954B2 (en) 2023-04-25
IL309708B1 (en) 2025-10-01
IL309708A (en) 2024-02-01
IL323267A (en) 2025-11-01
CN118515619A (en) 2024-08-20
JP2025163080A (en) 2025-10-28
IL271950A (en) 2020-02-27
BR112020000953A2 (en) 2020-07-14
CN111094252B (en) 2024-05-24
CA3069619A1 (en) 2019-02-28
CN111094252A (en) 2020-05-01
JP2020527563A (en) 2020-09-10
AU2018320492B2 (en) 2022-12-01
ZA202000411B (en) 2023-10-25

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