AR116305A1 - COMPOUNDS CONTAINING BORON AND THEIR USES - Google Patents
COMPOUNDS CONTAINING BORON AND THEIR USESInfo
- Publication number
- AR116305A1 AR116305A1 ARP190102563A ARP190102563A AR116305A1 AR 116305 A1 AR116305 A1 AR 116305A1 AR P190102563 A ARP190102563 A AR P190102563A AR P190102563 A ARP190102563 A AR P190102563A AR 116305 A1 AR116305 A1 AR 116305A1
- Authority
- AR
- Argentina
- Prior art keywords
- hydrocarbyl
- unsubstituted
- substitutions
- group
- hydrogen
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 4
- 125000001183 hydrocarbyl group Chemical group 0.000 abstract 9
- 238000006467 substitution reaction Methods 0.000 abstract 8
- 239000001257 hydrogen Substances 0.000 abstract 4
- 229910052739 hydrogen Inorganic materials 0.000 abstract 4
- 150000002431 hydrogen Chemical class 0.000 abstract 4
- WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical compound [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 abstract 3
- ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical compound [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 abstract 3
- PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical compound FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 abstract 3
- 125000003118 aryl group Chemical group 0.000 abstract 3
- GDTBXPJZTBHREO-UHFFFAOYSA-N bromine Substances BrBr GDTBXPJZTBHREO-UHFFFAOYSA-N 0.000 abstract 3
- 229910052794 bromium Inorganic materials 0.000 abstract 3
- 229910052801 chlorine Inorganic materials 0.000 abstract 3
- 239000000460 chlorine Substances 0.000 abstract 3
- 229910052731 fluorine Inorganic materials 0.000 abstract 3
- 239000011737 fluorine Substances 0.000 abstract 3
- 125000000623 heterocyclic group Chemical group 0.000 abstract 3
- 241001465754 Metazoa Species 0.000 abstract 2
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 2
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 2
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 2
- 125000001559 cyclopropyl group Chemical group [H]C1([H])C([H])([H])C1([H])* 0.000 abstract 2
- 229910052736 halogen Inorganic materials 0.000 abstract 2
- 150000002367 halogens Chemical group 0.000 abstract 2
- 125000001072 heteroaryl group Chemical group 0.000 abstract 2
- 229910052760 oxygen Inorganic materials 0.000 abstract 2
- 239000001301 oxygen Substances 0.000 abstract 2
- 229910052717 sulfur Inorganic materials 0.000 abstract 2
- 239000011593 sulfur Substances 0.000 abstract 2
- 241000239223 Arachnida Species 0.000 abstract 1
- ZOXJGFHDIHLPTG-UHFFFAOYSA-N Boron Chemical compound [B] ZOXJGFHDIHLPTG-UHFFFAOYSA-N 0.000 abstract 1
- 241000238631 Hexapoda Species 0.000 abstract 1
- 101100477978 Hypocrea jecorina (strain QM6a) sor6 gene Proteins 0.000 abstract 1
- 239000013543 active substance Substances 0.000 abstract 1
- 239000012872 agrochemical composition Substances 0.000 abstract 1
- 230000000845 anti-microbial effect Effects 0.000 abstract 1
- 230000002141 anti-parasite Effects 0.000 abstract 1
- 229910052796 boron Inorganic materials 0.000 abstract 1
- 235000013399 edible fruits Nutrition 0.000 abstract 1
- 230000002708 enhancing effect Effects 0.000 abstract 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 abstract 1
- 230000001747 exhibiting effect Effects 0.000 abstract 1
- 125000001188 haloalkyl group Chemical group 0.000 abstract 1
- 238000003898 horticulture Methods 0.000 abstract 1
- 230000000749 insecticidal effect Effects 0.000 abstract 1
- 239000000463 material Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
- IJGRMHOSHXDMSA-UHFFFAOYSA-N nitrogen Substances N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 abstract 1
- 244000045947 parasite Species 0.000 abstract 1
- 230000000361 pesticidal effect Effects 0.000 abstract 1
- 230000001737 promoting effect Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 235000013311 vegetables Nutrition 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N55/00—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
- A01N55/08—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur containing boron
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Agronomy & Crop Science (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
La presente contempla compuestos que contienen boro y sus usos como agentes activos que presentan actividad plaguicida tal como actividad antimicrobiana, insecticida, aracnicida y/o antiparasitaria. Una composición agroquímica que contiene dicho compuesto y sus usos también está contemplada en la salud animal, la agricultura, o la horticultura. También está contemplado un método para promover el rendimiento de las plantas y/o para reducir, mejorar o controlar microbios, insectos, arácnidos y/o parásitos sobre o dentro de un animal, una planta, una parte de una planta, el material para la propagación de las plantas y/o frutas o verduras cosechadas. Reivindicación 1: Un compuesto de la fórmula (1), en donde: X¹ se selecciona del grupo que consiste en: hidrógeno, flúor, cloro, bromo, CN, hidrocarbilo C₁₋₃ no sustituido, hidrocarbilo C₁₋₃ que tiene 1 - 7 sustituciones de halógeno y ciclopropilo; X¹ se selecciona del grupo que consiste en: hidrógeno, flúor, cloro, bromo, CN, hidrocarbilo C₁₋₃ no sustituido, hidrocarbilo C₁₋₃ que tiene 1 - 7 sustituciones de halógeno y ciclopropilo; Z¹ es oxígeno o azufre; Y¹ se selecciona del grupo que consiste en oxígeno, azufre y NH; R¹ se selecciona del grupo que consiste en: hidrógeno, hidrocarbilo C₁₋₈ no sustituido, hidrocarbilo C₁₋₈ que tiene 1 - 17 sustituciones de R¹ᵃ, ciclohidrocarbilo C₃₋₆ no sustituido, ciclohidrocarbilo C₃₋₆ que tiene 1 - 11 sustituciones de R¹ᵃ, arilo no sustituido, arilo que tiene 1 - 5 sustituciones de R¹ᵃ, bencilo no sustituido, bencilo que tiene 1 - 7 sustituciones de R¹ᵃ, heteroarilo no sustituido, heteroarilo sustituido con una o más sustituciones de R¹ᵃ, heterociclilo no sustituido y heterociclilo sustituido con una o más sustituciones de R¹ᵃ; cada R¹ᵃ se selecciona independientemente del grupo que consiste en hidrocarbilo C₁₋₈, NH₂, OH, NO₂, CN, haloalquilo C₁₋₂, OR⁶, SR⁶, SOR⁶, SO₂R⁶, NHC(O)OR⁶, NR⁶R⁷, C(O)OR, arilo no sustituido, ciclohidrocarbilo C₃₋₆, flúor, cloro, bromo, yodo, heteroarilo y heterociclilo; R⁶ y R⁷ se seleccionan independientemente del grupo que consiste en hidrocarbilo C₁₋₆ e hidrocarbilo sustituido, o R⁶ y R⁷ se pueden tomar junto con el nitrógeno al cual están unidos para formar un anillo de no más de 8 miembros; y cada uno de R⁸ y R⁹ se selecciona independientemente del grupo que consiste en: hidrógeno, metilo, etilo; o R⁸ y R⁹ se pueden tomar juntos para formar un anillo de 3 - 6 miembros; o una sal, estereoisómero, enantiómero, o tautómero de él.The present contemplates boron-containing compounds and their uses as active agents exhibiting pesticidal activity such as antimicrobial, insecticidal, arachnicidal and/or antiparasitic activity. An agrochemical composition containing said compound and its uses are also contemplated in animal health, agriculture, or horticulture. Also contemplated is a method for promoting plant performance and/or for reducing, enhancing or controlling microbes, insects, arachnids and/or parasites on or in an animal, plant, plant part, material for propagation of plants and/or harvested fruits or vegetables. Claim 1: A compound of formula (1), wherein: X¹ is selected from the group consisting of: hydrogen, fluorine, chlorine, bromine, CN, unsubstituted C₁₋₃ hydrocarbyl, C₁₋₃ hydrocarbyl having 1-7 halogen and cyclopropyl substitutions; X¹ is selected from the group consisting of: hydrogen, fluorine, chlorine, bromine, CN, C₁₋₃ unsubstituted hydrocarbyl, C₁₋₃ hydrocarbyl having 1-7 halogen and cyclopropyl substitutions; Z¹ is oxygen or sulfur; Y¹ is selected from the group consisting of oxygen, sulfur, and NH; R¹ is selected from the group consisting of: hydrogen, unsubstituted C₁₋₈ hydrocarbyl, C₁₋₈ hydrocarbyl having 1-17 R¹ᵃ substitutions, unsubstituted C₃₋₆ cyclohydrocarbyl, C₃₋₆ cyclohydrocarbyl having 1-11 R¹ᵃ substitutions , unsubstituted aryl, aryl having 1 - 5 R¹ᵃ substitutions, unsubstituted benzyl, benzyl having 1 - 7 R¹ᵃ substitutions, unsubstituted heteroaryl, heteroaryl substituted with one or more R¹ᵃ substitutions, unsubstituted heterocyclyl, and heterocyclyl substituted with one or more R¹ᵃ substitutions; each R¹ᵃ is independently selected from the group consisting of C₁₋₈ hydrocarbyl, NH₂, OH, NO₂, CN, C₁₋₂ haloalkyl, OR⁶, SR⁶, SOR⁶, SO₂R⁶, NHC(O)OR⁶, NR⁶R⁷, C(O)OR, unsubstituted aryl, C₃₋₆ cyclohydrocarbyl, fluorine, chlorine, bromine, iodine, heteroaryl and heterocyclyl; R⁶ and R⁷ are independently selected from the group consisting of C₁₋₆ hydrocarbyl and substituted hydrocarbyl, or R⁶ and R⁷ may be taken together with the nitrogen to which they are attached to form a ring of not more than 8 members; and each of R⁸ and R⁹ is independently selected from the group consisting of: hydrogen, methyl, ethyl; or R⁸ and R⁹ can be taken together to form a 3-6 membered ring; or a salt, stereoisomer, enantiomer, or tautomer thereof.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862728632P | 2018-09-07 | 2018-09-07 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR116305A1 true AR116305A1 (en) | 2021-04-21 |
Family
ID=69722876
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP190102563A AR116305A1 (en) | 2018-09-07 | 2019-09-09 | COMPOUNDS CONTAINING BORON AND THEIR USES |
Country Status (2)
| Country | Link |
|---|---|
| AR (1) | AR116305A1 (en) |
| WO (1) | WO2020051575A1 (en) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN115385836B (en) * | 2022-08-17 | 2023-11-07 | 南通大学 | A kind of synthesis method of aminoselenate compounds |
| WO2024040009A2 (en) * | 2022-08-17 | 2024-02-22 | Primetime Life Sciences, Llc | Inhibitors of methionine aminopeptidase-2 and methods of preparation and uses thereof |
| WO2025122491A1 (en) * | 2023-12-04 | 2025-06-12 | Aviko Radiopharmaceuticals, Llc | Fused bicyclic aryl compounds for boron neutron capture therapy |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JO3396B1 (en) * | 2007-06-20 | 2019-10-20 | Anacor Pharmaceuticals Inc | Boron-containing small molecules |
| WO2019152641A1 (en) * | 2018-02-01 | 2019-08-08 | Boragen, Inc. | Benzoxaborole compositions having a growth enhancing effect |
-
2019
- 2019-09-09 AR ARP190102563A patent/AR116305A1/en unknown
- 2019-09-09 WO PCT/US2019/050162 patent/WO2020051575A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO2020051575A1 (en) | 2020-03-12 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |