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AR101915A1 - INTERMEDIARIES AND PROCESSES FOR THE PREPARATION OF COMPOUNDS - Google Patents

INTERMEDIARIES AND PROCESSES FOR THE PREPARATION OF COMPOUNDS

Info

Publication number
AR101915A1
AR101915A1 ARP140103154A ARP140103154A AR101915A1 AR 101915 A1 AR101915 A1 AR 101915A1 AR P140103154 A ARP140103154 A AR P140103154A AR P140103154 A ARP140103154 A AR P140103154A AR 101915 A1 AR101915 A1 AR 101915A1
Authority
AR
Argentina
Prior art keywords
compounds
preparation
intermediaries
processes
pyrrolo
Prior art date
Application number
ARP140103154A
Other languages
Spanish (es)
Inventor
Han Chong
Original Assignee
Genentech Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Genentech Inc filed Critical Genentech Inc
Priority to ARP140103154A priority Critical patent/AR101915A1/en
Publication of AR101915A1 publication Critical patent/AR101915A1/en

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  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Intermediarios útiles en la preparación de compuestos que se pueden usar como inhibidores de CHK1, con actividad antineoplásica. Reivindicación 1: 4,5-dibromo-3-nitro-1H-pirrolo[2,3-b]piridina de fórmula (1), e isómeros, tautómeros y sales farmacéuticamente aceptables de estos.Intermediaries useful in the preparation of compounds that can be used as CHK1 inhibitors, with antineoplastic activity. Claim 1: 4,5-dibromo-3-nitro-1H-pyrrolo [2,3-b] pyridine of formula (1), and pharmaceutically acceptable isomers, tautomers and salts thereof.

ARP140103154A 2014-08-22 2014-08-22 INTERMEDIARIES AND PROCESSES FOR THE PREPARATION OF COMPOUNDS AR101915A1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ARP140103154A AR101915A1 (en) 2014-08-22 2014-08-22 INTERMEDIARIES AND PROCESSES FOR THE PREPARATION OF COMPOUNDS

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ARP140103154A AR101915A1 (en) 2014-08-22 2014-08-22 INTERMEDIARIES AND PROCESSES FOR THE PREPARATION OF COMPOUNDS

Publications (1)

Publication Number Publication Date
AR101915A1 true AR101915A1 (en) 2017-01-25

Family

ID=58698650

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP140103154A AR101915A1 (en) 2014-08-22 2014-08-22 INTERMEDIARIES AND PROCESSES FOR THE PREPARATION OF COMPOUNDS

Country Status (1)

Country Link
AR (1) AR101915A1 (en)

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