AR109263A2 - Composición que comprende moxidectina - Google Patents
Composición que comprende moxidectinaInfo
- Publication number
- AR109263A2 AR109263A2 ARP170101975A ARP170101975A AR109263A2 AR 109263 A2 AR109263 A2 AR 109263A2 AR P170101975 A ARP170101975 A AR P170101975A AR P170101975 A ARP170101975 A AR P170101975A AR 109263 A2 AR109263 A2 AR 109263A2
- Authority
- AR
- Argentina
- Prior art keywords
- moxidectine
- composition including
- composition
- demodicosis
- moxidectin
- Prior art date
Links
- YZBLFMPOMVTDJY-LSGXYNIPSA-N Moxidectin Chemical compound O1[C@H](C(\C)=C\C(C)C)[C@@H](C)C(=N/OC)/C[C@@]11O[C@H](C\C=C(C)\C[C@@H](C)\C=C\C=C/2[C@]3([C@H](C(=O)O4)C=C(C)[C@@H](O)[C@H]3OC\2)O)C[C@H]4C1 YZBLFMPOMVTDJY-LSGXYNIPSA-N 0.000 title 1
- 208000020693 Demodicidosis Diseases 0.000 abstract 1
- 239000005906 Imidacloprid Substances 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- YWTYJOPNNQFBPC-UHFFFAOYSA-N imidacloprid Chemical compound [O-][N+](=O)\N=C1/NCCN1CC1=CC=C(Cl)N=C1 YWTYJOPNNQFBPC-UHFFFAOYSA-N 0.000 abstract 1
- 229940056881 imidacloprid Drugs 0.000 abstract 1
- YZBLFMPOMVTDJY-CBYMMZEQSA-N moxidectin Chemical compound O1[C@H](C(\C)=C\C(C)C)[C@@H](C)C(=N/OC)\C[C@@]11O[C@H](C\C=C(C)\C[C@@H](C)\C=C\C=C/2[C@]3([C@H](C(=O)O4)C=C(C)[C@@H](O)[C@H]3OC\2)O)C[C@H]4C1 YZBLFMPOMVTDJY-CBYMMZEQSA-N 0.000 abstract 1
- 229960004816 moxidectin Drugs 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/365—Lactones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Tropical Medicine & Parasitology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Fodder In General (AREA)
- Pyrane Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
Reivindicación 1: Una composición que comprende moxidectina, caracterizada porque se usa en la preparación de un medicamento de aplicación externa para el tratamiento de la demodicosis. Reivindicación 2: Una composición de acuerdo con la reivindicación 1, caracterizada porque además comprende imidacloprid.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102004053964A DE102004053964A1 (de) | 2004-11-09 | 2004-11-09 | Mittel gegen Demodikose |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR109263A2 true AR109263A2 (es) | 2018-11-14 |
Family
ID=35614662
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP050104675A AR051664A1 (es) | 2004-11-09 | 2005-11-08 | Agente contra la demodicosis |
| ARP170101975A AR109263A2 (es) | 2004-11-09 | 2017-07-14 | Composición que comprende moxidectina |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP050104675A AR051664A1 (es) | 2004-11-09 | 2005-11-08 | Agente contra la demodicosis |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US9662309B2 (es) |
| EP (1) | EP1811990B1 (es) |
| AR (2) | AR051664A1 (es) |
| AU (1) | AU2005304103B2 (es) |
| BR (2) | BR122019002159B1 (es) |
| DE (1) | DE102004053964A1 (es) |
| DK (1) | DK1811990T3 (es) |
| ES (1) | ES2711329T3 (es) |
| HU (1) | HUE041365T2 (es) |
| LT (1) | LT1811990T (es) |
| PL (1) | PL1811990T3 (es) |
| PT (1) | PT1811990T (es) |
| SI (1) | SI1811990T1 (es) |
| TR (1) | TR201901390T4 (es) |
| TW (1) | TWI432205B (es) |
| WO (1) | WO2006050816A1 (es) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2947453B1 (fr) * | 2009-07-03 | 2011-08-19 | Akil Sa | Medicament antiparasitaire pour application topique contre les affections dues au demodex |
| CN103641873B (zh) * | 2013-12-17 | 2015-10-28 | 华北制药集团爱诺有限公司 | 一种阿维菌素的制备方法 |
| WO2016022066A1 (en) | 2014-08-04 | 2016-02-11 | Jerry Tan Eye Surgery Pte Ltd | Pharmaceutical compositions for demodex related blepharitis and eyelid crusting |
| PL3236960T3 (pl) * | 2014-12-22 | 2025-07-07 | Intervet International B.V. | Fluralaner do zastosowania w leczeniu demodekozy |
| RU2568869C1 (ru) * | 2015-01-16 | 2015-11-20 | Федеральное государственное бюджетное научное учреждение Всероссийский научно-исследовательский институт фундаментальной и прикладной паразитологии животных и растений им. К.И. Скрябина (ФГБНУ "ВНИИП им. К.И. Скрябина") | Способ лечения демодекоза собак |
| RU2634265C1 (ru) * | 2016-10-18 | 2017-10-24 | Федеральное государственное бюджетное учреждение науки Федеральный исследовательский центр Тюменский научный центр Сибирского отделения Российской академии наук (ТюмНЦ СО РАН) | Способ лечения демодекоза собак |
| KR20250065422A (ko) | 2017-12-15 | 2025-05-12 | 타르서스 파마수티칼스, 아이엔씨. | 안검염을 치료하기 위한 이속사졸린 구충제 제제 및 방법 |
| CN113557015A (zh) * | 2018-12-21 | 2021-10-26 | 礼蓝美国公司 | 杀寄生虫制剂及其用途 |
| WO2020150032A1 (en) * | 2019-01-16 | 2020-07-23 | Boehringer Ingelheim Animal Health USA Inc. | Topical compositions comprising a neonicotinoid and a macrocyclic lactone, methods and uses thereof |
| SI3815677T1 (sl) | 2019-10-30 | 2023-12-29 | Krka, D.D., Novo Mesto | Stabilni veterinarski sestavek, ki obsega moksidektin in imidakloprid |
| WO2023111333A1 (en) * | 2021-12-17 | 2023-06-22 | Bayer Animal Health Gmbh | Topical administration of composition comprising 10% w/v imidacloprid and 1% w/v moxidectin for the treatment of troglostrongylosis in cats |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6426333B1 (en) * | 1996-09-19 | 2002-07-30 | Merial | Spot-on formulations for combating parasites |
| JPS4914624A (es) | 1972-06-08 | 1974-02-08 | ||
| SE434277B (sv) * | 1976-04-19 | 1984-07-16 | Merck & Co Inc | Sett att framstella nya antihelmintiskt verkande foreningar genom odling av streptomyces avermitilis |
| US4199569A (en) * | 1977-10-03 | 1980-04-22 | Merck & Co., Inc. | Selective hydrogenation products of C-076 compounds and derivatives thereof |
| DE3727648A1 (de) * | 1987-08-19 | 1989-03-02 | Bayer Ag | Neue avermectin derivate, verfahren zu ihrer herstellung und ihre verwendung |
| NZ233680A (en) * | 1989-05-17 | 1995-02-24 | Beecham Group Plc | Avermectins and milbemycins and compositions thereof |
| ATE130006T1 (de) | 1989-09-11 | 1995-11-15 | American Cyanamid Co | 13-alkyl-23-imino und 13-halo-23-imino-derivate von ll-f28249-verbindungen und ihre verwendung als endo- und ectoparasitizide, insektizide, akarizide und nematozide mittel. |
| GB9024927D0 (en) * | 1990-11-16 | 1991-01-02 | Beecham Group Plc | Novel treatment |
| DE19613972A1 (de) * | 1996-04-09 | 1997-10-16 | Bayer Ag | Injektionsformulierungen von Avermectinen und Milbemycinen auf Basis von Rizinusöl |
| DE19654079A1 (de) * | 1996-12-23 | 1998-06-25 | Bayer Ag | Endo-ekto-parasitizide Mittel |
| US5952372A (en) * | 1998-09-17 | 1999-09-14 | Mcdaniel; William Robert | Method for treating rosacea using oral or topical ivermectin |
| GB9825402D0 (en) * | 1998-11-19 | 1999-01-13 | Pfizer Ltd | Antiparasitic formulations |
| PE20011289A1 (es) * | 2000-04-07 | 2001-12-21 | Upjohn Co | Composiciones antihelminticas que comprenden lactonas macrociclicas y espirodioxepinoindoles |
| DE10117676A1 (de) * | 2001-04-09 | 2002-10-10 | Bayer Ag | Dermal applizierbare flüssige Formulierungen zur Bekämpfung von parasitierenden Insekten an Tieren |
| DK1610613T3 (en) * | 2003-04-04 | 2017-02-27 | Merial Inc | TOPICAL ANTHELMINTIC VETERINARY FORMULATIONS |
| US7514464B2 (en) * | 2003-12-18 | 2009-04-07 | Pfizer Limited | Substituted arylpyrazoles |
-
2004
- 2004-11-09 DE DE102004053964A patent/DE102004053964A1/de not_active Withdrawn
-
2005
- 2005-10-27 US US11/718,914 patent/US9662309B2/en not_active Expired - Lifetime
- 2005-10-27 PL PL05802055T patent/PL1811990T3/pl unknown
- 2005-10-27 TR TR2019/01390T patent/TR201901390T4/tr unknown
- 2005-10-27 WO PCT/EP2005/011484 patent/WO2006050816A1/de not_active Ceased
- 2005-10-27 AU AU2005304103A patent/AU2005304103B2/en not_active Expired
- 2005-10-27 BR BR122019002159-7A patent/BR122019002159B1/pt active IP Right Grant
- 2005-10-27 DK DK05802055.3T patent/DK1811990T3/en active
- 2005-10-27 HU HUE05802055A patent/HUE041365T2/hu unknown
- 2005-10-27 LT LTEP05802055.3T patent/LT1811990T/lt unknown
- 2005-10-27 ES ES05802055T patent/ES2711329T3/es not_active Expired - Lifetime
- 2005-10-27 EP EP05802055.3A patent/EP1811990B1/de not_active Expired - Lifetime
- 2005-10-27 PT PT05802055T patent/PT1811990T/pt unknown
- 2005-10-27 SI SI200532243T patent/SI1811990T1/sl unknown
- 2005-10-27 BR BRPI0517966-1A patent/BRPI0517966B1/pt active IP Right Grant
- 2005-11-08 TW TW094139036A patent/TWI432205B/zh active
- 2005-11-08 AR ARP050104675A patent/AR051664A1/es unknown
-
2017
- 2017-07-14 AR ARP170101975A patent/AR109263A2/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| US20080039519A1 (en) | 2008-02-14 |
| TW200626162A (en) | 2006-08-01 |
| TR201901390T4 (tr) | 2019-02-21 |
| AU2005304103A1 (en) | 2006-05-18 |
| US9662309B2 (en) | 2017-05-30 |
| HUE041365T2 (hu) | 2019-05-28 |
| LT1811990T (lt) | 2019-02-25 |
| BRPI0517966A (pt) | 2008-10-28 |
| BR122019002159B1 (pt) | 2021-08-17 |
| EP1811990B1 (de) | 2018-11-21 |
| AU2005304103B2 (en) | 2012-02-02 |
| PT1811990T (pt) | 2019-02-19 |
| SI1811990T1 (sl) | 2019-03-29 |
| TWI432205B (zh) | 2014-04-01 |
| AR051664A1 (es) | 2007-01-31 |
| BRPI0517966B1 (pt) | 2023-09-26 |
| ES2711329T3 (es) | 2019-05-03 |
| DK1811990T3 (en) | 2019-03-11 |
| PL1811990T3 (pl) | 2019-05-31 |
| EP1811990A1 (de) | 2007-08-01 |
| DE102004053964A1 (de) | 2006-05-11 |
| WO2006050816A1 (de) | 2006-05-18 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC | Refusal |