AR076929A1 - Composicion farmaceutica para modular las funciones mediadas por claudina. uso de un derivado de acido graso - Google Patents
Composicion farmaceutica para modular las funciones mediadas por claudina. uso de un derivado de acido grasoInfo
- Publication number
- AR076929A1 AR076929A1 ARP100101835A ARP100101835A AR076929A1 AR 076929 A1 AR076929 A1 AR 076929A1 AR P100101835 A ARP100101835 A AR P100101835A AR P100101835 A ARP100101835 A AR P100101835A AR 076929 A1 AR076929 A1 AR 076929A1
- Authority
- AR
- Argentina
- Prior art keywords
- fatty acid
- acid derivative
- pharmaceutical composition
- claudine
- claudin
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
- A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/557—Eicosanoids, e.g. leukotrienes or prostaglandins
- A61K31/5575—Eicosanoids, e.g. leukotrienes or prostaglandins having a cyclopentane, e.g. prostaglandin E2, prostaglandin F2-alpha
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/557—Eicosanoids, e.g. leukotrienes or prostaglandins
- A61K31/558—Eicosanoids, e.g. leukotrienes or prostaglandins having heterocyclic rings containing oxygen as the only ring hetero atom, e.g. thromboxanes
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Uso de un derivado de ácido graso para la produccion de una composicion farmacéutica para modular una funcion mediada por claudina en un sujeto mamífero. Uso del mismo derivado de ácido graso que el anterior para la produccion de una composicion farmacéutica para tratar una enfermedad dermatologica y aquélla para la modulacion de una expresion de una claudina en un sujeto mamífero. Reivindicacion 15: El uso de acuerdo con la reivindicacion 1, caracterizado porque dicho derivado de ácido graso es ácido (-) -7-[(2R, 4aR, 7aR) -2- (1, 1-difluoropentil)-2-hidroxi-6- oxooctahidrociclopenta [b] piran-5-il] heptanoico o su derivado funcional. Reivindicacion 16: El uso de acuerdo con la reivindicacion 1, caracterizado porque dicha enfermedad dermatologica es una ulcera cutánea o una escara. Reivindicacion 19: El uso de acuerdo con la reivindicacion 17, caracterizado porque dicha funcion mediada por claudina es una funcion de barrera epidérmica.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US18146309P | 2009-05-27 | 2009-05-27 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR076929A1 true AR076929A1 (es) | 2011-07-20 |
Family
ID=42352317
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP100101835A AR076929A1 (es) | 2009-05-27 | 2010-05-27 | Composicion farmaceutica para modular las funciones mediadas por claudina. uso de un derivado de acido graso |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US20100305203A1 (es) |
| EP (1) | EP2435049A1 (es) |
| JP (1) | JP2012528077A (es) |
| KR (1) | KR20120031954A (es) |
| CN (1) | CN102448463A (es) |
| AR (1) | AR076929A1 (es) |
| AU (1) | AU2010253720A1 (es) |
| BR (1) | BRPI1011658A2 (es) |
| CA (1) | CA2761250A1 (es) |
| IL (1) | IL216218A0 (es) |
| MX (1) | MX2011012595A (es) |
| NZ (1) | NZ596555A (es) |
| RU (1) | RU2011153196A (es) |
| TW (1) | TW201102070A (es) |
| WO (1) | WO2010137731A1 (es) |
| ZA (1) | ZA201109532B (es) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2014159679A1 (en) | 2013-03-12 | 2014-10-02 | The United States Of America, As Represented By The Secretary, Department Of Health & Human Services | Methods for using lubiprostone to absorb fluid from the subretinal space |
| EP4440561A4 (en) * | 2021-12-03 | 2025-12-10 | Univ Chicago | CLAUDIN INHIBITORS AND THEIR METHODS OF USE |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5166174A (en) * | 1987-01-28 | 1992-11-24 | K.K. Ueno Seiyaku Oyo Kenkyujo | Prostaglandins E and anti-ulcers containing same |
| JPH01265021A (ja) * | 1987-10-29 | 1989-10-23 | Hercon Lab Corp | 薬理学的活性物質を含有する組成物を動物組織に制御放出および供給するための物品 |
| CA2030344C (en) * | 1989-11-22 | 2000-04-18 | Ryuji Ueno | Treatment of pulmonary dysfunction with 15-keto-prostaglandin compounds |
| JPH04300833A (ja) * | 1991-03-29 | 1992-10-23 | Green Cross Corp:The | プロスタグランジンe1 含有脂肪乳剤充填噴霧剤 |
| JP2802912B2 (ja) * | 1995-08-16 | 1998-09-24 | 小野薬品工業株式会社 | プロスタグランジンe1エステル、それらを含有するリポソーム製剤、およびそれらを含有する医薬 |
| TW367324B (en) * | 1995-08-16 | 1999-08-21 | Ono Pharmaceutical Co | Prostaglandin derivatives |
| JPH09124593A (ja) * | 1995-08-25 | 1997-05-13 | Ono Pharmaceut Co Ltd | プロスタグランジンe1エステル、それらを含有するリポソーム製剤、およびそれらを含有する医薬 |
| KR100227541B1 (ko) * | 1995-08-25 | 1999-11-01 | 우에노 도시오 | 프로스타글란딘 유도체 |
| US20060100181A1 (en) * | 2002-05-03 | 2006-05-11 | Jost-Price Edward R | Combinations for the treatment of inflammatory skin disorders |
| US7737182B2 (en) * | 2002-08-09 | 2010-06-15 | Taisho Pharmaceutical Co., Ltd. | Pharmaceuticals for xerosis |
| JP2005139194A (ja) * | 2002-08-09 | 2005-06-02 | Taisho Pharmaceut Co Ltd | 止痒剤 |
| PT2465537T (pt) * | 2002-10-10 | 2016-08-03 | Ono Pharmaceutical Co | Microsferas compreendendo ono-1301 |
| NZ561414A (en) * | 2005-03-04 | 2010-10-29 | Sucampo Ag | Method and composition for treating peripheral vascular diseases |
| CN101180096B (zh) * | 2005-03-21 | 2015-04-22 | 苏坎波公司 | 用于治疗粘膜疾病的方法和组合物 |
| US20060281818A1 (en) * | 2005-03-21 | 2006-12-14 | Sucampo Ag, North Carolina State University | Method for treating mucosal disorders |
| US8871752B2 (en) * | 2008-02-19 | 2014-10-28 | Sucampo Ag | Method for modulating stem cell growth |
| CN101318948B (zh) * | 2008-04-01 | 2011-04-27 | 上海天伟生物制药有限公司 | 鲁比前列酮晶体、其制备方法及用途 |
-
2010
- 2010-05-26 MX MX2011012595A patent/MX2011012595A/es not_active Application Discontinuation
- 2010-05-26 CA CA2761250A patent/CA2761250A1/en not_active Abandoned
- 2010-05-26 CN CN2010800230554A patent/CN102448463A/zh active Pending
- 2010-05-26 KR KR1020117030946A patent/KR20120031954A/ko not_active Withdrawn
- 2010-05-26 EP EP10722792A patent/EP2435049A1/en not_active Withdrawn
- 2010-05-26 AU AU2010253720A patent/AU2010253720A1/en not_active Abandoned
- 2010-05-26 JP JP2011550343A patent/JP2012528077A/ja active Pending
- 2010-05-26 RU RU2011153196/15A patent/RU2011153196A/ru not_active Application Discontinuation
- 2010-05-26 NZ NZ596555A patent/NZ596555A/en not_active IP Right Cessation
- 2010-05-26 WO PCT/JP2010/059300 patent/WO2010137731A1/en not_active Ceased
- 2010-05-26 BR BRPI1011658A patent/BRPI1011658A2/pt not_active IP Right Cessation
- 2010-05-26 US US12/787,947 patent/US20100305203A1/en not_active Abandoned
- 2010-05-27 TW TW099116952A patent/TW201102070A/zh unknown
- 2010-05-27 AR ARP100101835A patent/AR076929A1/es unknown
-
2011
- 2011-11-08 IL IL216218A patent/IL216218A0/en unknown
- 2011-12-23 ZA ZA2011/09532A patent/ZA201109532B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN102448463A (zh) | 2012-05-09 |
| NZ596555A (en) | 2014-01-31 |
| TW201102070A (en) | 2011-01-16 |
| AU2010253720A1 (en) | 2011-12-08 |
| US20100305203A1 (en) | 2010-12-02 |
| WO2010137731A1 (en) | 2010-12-02 |
| KR20120031954A (ko) | 2012-04-04 |
| MX2011012595A (es) | 2011-12-16 |
| JP2012528077A (ja) | 2012-11-12 |
| ZA201109532B (en) | 2012-09-26 |
| IL216218A0 (en) | 2012-01-31 |
| BRPI1011658A2 (pt) | 2018-03-06 |
| EP2435049A1 (en) | 2012-04-04 |
| CA2761250A1 (en) | 2010-12-02 |
| RU2011153196A (ru) | 2013-07-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |