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AR065941A1 - Nuevas formulaciones para la provision de terapeuticas peptidicas antivirales. composicion. - Google Patents

Nuevas formulaciones para la provision de terapeuticas peptidicas antivirales. composicion.

Info

Publication number
AR065941A1
AR065941A1 ARP080101399A ARP080101399A AR065941A1 AR 065941 A1 AR065941 A1 AR 065941A1 AR P080101399 A ARP080101399 A AR P080101399A AR P080101399 A ARP080101399 A AR P080101399A AR 065941 A1 AR065941 A1 AR 065941A1
Authority
AR
Argentina
Prior art keywords
composition
composition according
peptide
antiviral
administration
Prior art date
Application number
ARP080101399A
Other languages
English (en)
Original Assignee
Trimeris Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Trimeris Inc filed Critical Trimeris Inc
Publication of AR065941A1 publication Critical patent/AR065941A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/162Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from virus
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/19Cytokines; Lymphokines; Interferons
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A61K9/0024Solid, semi-solid or solidifying implants, which are implanted or injected in body tissue
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/06Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Virology (AREA)
  • Immunology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Zoology (AREA)
  • Organic Chemistry (AREA)
  • Biomedical Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurosurgery (AREA)
  • Communicable Diseases (AREA)
  • Dermatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Inorganic Chemistry (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Medicinal Preparation (AREA)

Abstract

Composiciones y métodos para su administracion como agentes terapéuticos. En particular, composiciones y su uso para la administracion de terapéuticas peptídicas antivirales. Reivindicacion 1: Una composicion caracterizada porque comprende unsolvente, un material gelante y un molécula bioactiva, en donde tras la administracion a un paciente, dicha composicion formas una matriz y provee una Cmáx de dicha molécula bioactiva de al menos 1 microg/ml dentro de 12 horas de administracionseguida de liberacion sostenidacon niveles plasmáticos de al menos 1 microg/ml durante al menos 7 días. Reivindicacion 2: Una composicion caracterizada porque comprende un solvente, un material gelante y un péptido seleccionado de T20, T1249,T897, T2635, T999 y T1144, o una de sus combinaciones. Reivindicacion 12: La composicion de acuerdo con la reivindicacion 2, caracterizada porque el péptido es T1144. Reivindicacion 14: La composicion de acuerdo con la reivindicacion 2,caracterizada porque dicha composicion también comprende al menos otra molécula bioactiva. Reivindicacion 15: La composicion de acuerdo con la reivindicacion 14, caracterizada porque la otra molécula bioactiva es un agenteantiviral. Reivindicacion 17: La composicion de acuerdo con la reivindicacion 15, caracterizada porque el agente antiviral es una citoquina. Reivindicacion 18: La composicion de acuerdo con la reivindicacion 15, caracterizada porque el agenteviral es inhibidor transcriptasa inversa. Reivindicacion 19: La composicion de acuerdo con la reivindicacion 15, caracterizada porque el agente antiviral es un inhibidor de cubierta de mARN viral. Reivindicacion 32: Un método para la liberacionsostenida de un péptido en un paciente caracterizado porque comprende administrar al paciente una composicion que comprenden un solvente, un material gelante y un péptido seleccionado de T20, T1249, T897, T2635, T999 y T1144, o una de suscombinaciones. Reivindicacion 38: Un método para aliviar un síntoma asociado con una infeccion por HIV, caracterizadol porque comprende administrar a un paciente infectado por HIV una composicion que comprende un solvente, un material gelante y unpéptido seleccionado de T20, T1249, T897, T2635, T999 y T1144, o una de sus combinaciones.
ARP080101399A 2007-04-03 2008-04-03 Nuevas formulaciones para la provision de terapeuticas peptidicas antivirales. composicion. AR065941A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US92170407P 2007-04-03 2007-04-03

Publications (1)

Publication Number Publication Date
AR065941A1 true AR065941A1 (es) 2009-07-15

Family

ID=39831248

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP080101399A AR065941A1 (es) 2007-04-03 2008-04-03 Nuevas formulaciones para la provision de terapeuticas peptidicas antivirales. composicion.

Country Status (11)

Country Link
US (1) US20090068243A1 (es)
EP (1) EP2139526A4 (es)
JP (1) JP2010523564A (es)
KR (1) KR20100016142A (es)
CN (1) CN101678125A (es)
AR (1) AR065941A1 (es)
BR (1) BRPI0809995A2 (es)
CA (1) CA2682848A1 (es)
MX (1) MX2009010689A (es)
TW (1) TW200902043A (es)
WO (1) WO2008124013A1 (es)

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US8852638B2 (en) 2005-09-30 2014-10-07 Durect Corporation Sustained release small molecule drug formulation
EP2907524A1 (en) 2007-05-25 2015-08-19 RB Pharmaceuticals Limited Sustained delivery formulations of risperidone compounds
BRPI0817697A2 (pt) * 2007-09-25 2015-04-07 Trimeris Inc Método de síntese de um peptídeo, conjunto de fragmentos de peptídeo, e, peptídeo
WO2010047826A2 (en) * 2008-10-24 2010-04-29 Trimeris, Inc. Dosing regimens and dosage formulations of an antiviral peptide therapeutic
WO2012074883A1 (en) * 2010-11-24 2012-06-07 Durect Corporation Biodegradable drug delivery composition
EP2782590A4 (en) * 2011-11-23 2016-08-03 Durect Corp BIODEGRADABLE AND MEDIUM-RADIATED STERILIZED MEDICAMENTAL COMPOSITIONS
CN105163719B (zh) 2013-03-11 2019-03-08 度瑞公司 包含高粘度液体载体的可注射控制释放组合物
US20140308352A1 (en) 2013-03-11 2014-10-16 Zogenix Inc. Compositions and methods involving polymer, solvent, and high viscosity liquid carrier material
CA2931547A1 (en) 2013-12-09 2015-06-18 Durect Corporation Pharmaceutically active agent complexes, polymer complexes, and compositions and methods involving the same
CN109320593A (zh) * 2018-11-05 2019-02-12 中国人民解放军军事科学院军事医学研究院 抑制hiv感染的螺旋多肽及其用途
CN112851789B (zh) * 2021-02-04 2022-10-18 大理大学 一种脑靶向hiv进入抑制剂多肽及其应用

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Also Published As

Publication number Publication date
US20090068243A1 (en) 2009-03-12
CN101678125A (zh) 2010-03-24
CA2682848A1 (en) 2008-10-16
MX2009010689A (es) 2009-12-14
TW200902043A (en) 2009-01-16
JP2010523564A (ja) 2010-07-15
EP2139526A4 (en) 2010-07-14
BRPI0809995A2 (pt) 2015-07-21
KR20100016142A (ko) 2010-02-12
WO2008124013A1 (en) 2008-10-16
EP2139526A1 (en) 2010-01-06

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