AR014119A1 - Utilizacion de cetolidas para la fabricacion de composiciones farmaceuticas destinadas a prevenir complicaciones tromboticas arteriales asociadas a laaterosclerosis - Google Patents
Utilizacion de cetolidas para la fabricacion de composiciones farmaceuticas destinadas a prevenir complicaciones tromboticas arteriales asociadas a laaterosclerosisInfo
- Publication number
- AR014119A1 AR014119A1 ARP980105823A ARP980105823A AR014119A1 AR 014119 A1 AR014119 A1 AR 014119A1 AR P980105823 A ARP980105823 A AR P980105823A AR P980105823 A ARP980105823 A AR P980105823A AR 014119 A1 AR014119 A1 AR 014119A1
- Authority
- AR
- Argentina
- Prior art keywords
- pharmaceutical compositions
- complications associated
- compositions intended
- laterosclerosis
- cetolids
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 230000001732 thrombotic effect Effects 0.000 title abstract 2
- 238000004519 manufacturing process Methods 0.000 title 1
- 201000001320 Atherosclerosis Diseases 0.000 abstract 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 125000001072 heteroaryl group Chemical class 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 239000003835 ketolide antibiotic agent Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Molecular Biology (AREA)
- Epidemiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Cardiology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Abstract
Se describe la utilizacion de cetolidas para la preparacion de composiciones farmacéuticas destinadas a prevenir las complicacionestromboticas arteriales asociadas a la aterosclerosis. Las cetolidas responden a la formula (I) en la cualR representa un radical (CH2)mOn(X)YAr en la cual mrepresenta el numero 0 o 1, n representa el numero 0 o 1, X representa un radical (NH)a, CH2 o SO2, representando al numero 0 o 1, Y representa unradical (CH2)b-(CH=CH)c-(CH2)d con c= 0 o 1, b+ c + d < o = que 8, Z representa un átomo de hidrogeno o de halogeno, y Ar representa un radicalarilo o heteroarilo eventualmente sustituido.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9714358A FR2771008B1 (fr) | 1997-11-17 | 1997-11-17 | Utilisation des ketolides pour la preparation de compositions pharmaceutiques destinees a prevenir les complications thrombotiques arterielles liees a l'atherosclerose |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR014119A1 true AR014119A1 (es) | 2001-02-07 |
Family
ID=9513423
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP980105823A AR014119A1 (es) | 1997-11-17 | 1998-11-17 | Utilizacion de cetolidas para la fabricacion de composiciones farmaceuticas destinadas a prevenir complicaciones tromboticas arteriales asociadas a laaterosclerosis |
Country Status (35)
| Country | Link |
|---|---|
| US (1) | US20080139489A1 (es) |
| EP (1) | EP1030673B1 (es) |
| JP (1) | JP4550273B2 (es) |
| KR (1) | KR20010032130A (es) |
| CN (1) | CN1286633A (es) |
| AP (1) | AP1196A (es) |
| AR (1) | AR014119A1 (es) |
| AT (1) | ATE271875T1 (es) |
| AU (1) | AU744419B2 (es) |
| BG (1) | BG104427A (es) |
| BR (1) | BR9814199A (es) |
| CA (1) | CA2312021C (es) |
| DE (1) | DE69825308T2 (es) |
| DZ (1) | DZ2654A1 (es) |
| EA (1) | EA003322B1 (es) |
| EE (1) | EE04095B1 (es) |
| ES (1) | ES2224446T3 (es) |
| FR (1) | FR2771008B1 (es) |
| GE (1) | GEP20032968B (es) |
| HR (1) | HRP20000314A2 (es) |
| HU (1) | HUP0004507A3 (es) |
| ID (1) | ID24940A (es) |
| IL (1) | IL136149A0 (es) |
| MA (1) | MA26566A1 (es) |
| NO (1) | NO20002435L (es) |
| NZ (1) | NZ504305A (es) |
| OA (1) | OA11411A (es) |
| PL (1) | PL340373A1 (es) |
| SK (1) | SK7042000A3 (es) |
| TN (1) | TNSN98206A1 (es) |
| TR (1) | TR200001384T2 (es) |
| TW (1) | TW472061B (es) |
| WO (1) | WO1999025365A1 (es) |
| YU (1) | YU29600A (es) |
| ZA (1) | ZA9810357B (es) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2777282B1 (fr) * | 1998-04-08 | 2001-04-20 | Hoechst Marion Roussel Inc | Nouveaux derives de la 2-fluoro 3-de((2,6-dideoxy 3-c-methyl 3-0-methyl-alpha-l-ribohexopyranosyl) oxyl) 6-o-methyl 3-oxo erythromycine, leur procede de preparation et leur application a la synthese de principes actifs de medicaments |
| TR200102129T2 (tr) | 1998-12-10 | 2002-01-21 | Pfizer Products Inc. | Karbamat ve karbazat ketolid antibiyotikleri. |
| KR20020002380A (ko) * | 1999-01-27 | 2002-01-09 | 실버스타인 아써 에이. | 케톨라이드 항생물질 |
| EP1114826A3 (en) * | 1999-12-29 | 2001-10-31 | Pfizer Products Inc. | Novel antibacterial and prokinetic macrolides |
| CA2405132A1 (en) | 2000-04-04 | 2001-10-11 | Smithkline Beecham Plc | 2-hydroxy-mutilin carbamate derivatives for antibacterial use |
| JP2004323414A (ja) * | 2003-04-24 | 2004-11-18 | Japan Science & Technology Agency | １４員環マクロライド化合物を利用した、血管平滑筋の増殖に起因する疾患治療剤 |
| GB0402578D0 (en) * | 2004-02-05 | 2004-03-10 | Cambridge Theranostics Ltd | Methods of treatment of atherosclerosis |
| US9815863B2 (en) * | 2010-09-10 | 2017-11-14 | Cempra Pharmaceuticals, Inc. | Hydrogen bond forming fluoro ketolides for treating diseases |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2249892A (en) * | 1991-06-14 | 1993-01-12 | Board Of Regents Of The University Of Washington, The | Diagnosis and treatment of arterial chlamydial granuloma |
| FR2718450B1 (fr) * | 1994-04-08 | 1997-01-10 | Roussel Uclaf | Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments. |
| FR2719587B1 (fr) * | 1994-05-03 | 1996-07-12 | Roussel Uclaf | Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments. |
| FR2742757B1 (fr) * | 1995-12-22 | 1998-01-30 | Roussel Uclaf | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
| US6271255B1 (en) * | 1996-07-05 | 2001-08-07 | Biotica Technology Limited | Erythromycins and process for their preparation |
| GB9621771D0 (en) * | 1996-10-18 | 1996-12-11 | St George S Enterprises Ltd | Method of treatment of heart disease |
| FR2757168B1 (fr) * | 1996-12-12 | 1999-06-11 | Hoechst Marion Roussel Inc | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
| EP0895999A1 (en) * | 1997-08-06 | 1999-02-10 | Pfizer Products Inc. | C-4" substituted macrolide antibiotics |
-
1997
- 1997-11-17 FR FR9714358A patent/FR2771008B1/fr not_active Expired - Fee Related
-
1998
- 1998-11-12 ZA ZA9810357A patent/ZA9810357B/xx unknown
- 1998-11-13 TW TW087118866A patent/TW472061B/zh not_active IP Right Cessation
- 1998-11-16 CN CN98813159A patent/CN1286633A/zh active Pending
- 1998-11-16 EA EA200000531A patent/EA003322B1/ru not_active IP Right Cessation
- 1998-11-16 ES ES98955662T patent/ES2224446T3/es not_active Expired - Lifetime
- 1998-11-16 HR HR20000314A patent/HRP20000314A2/hr not_active Application Discontinuation
- 1998-11-16 IL IL13614998A patent/IL136149A0/xx unknown
- 1998-11-16 SK SK704-2000A patent/SK7042000A3/sk unknown
- 1998-11-16 BR BR9814199-6A patent/BR9814199A/pt not_active Application Discontinuation
- 1998-11-16 DE DE69825308T patent/DE69825308T2/de not_active Expired - Lifetime
- 1998-11-16 DZ DZ980264A patent/DZ2654A1/xx active
- 1998-11-16 ID IDW20000930A patent/ID24940A/id unknown
- 1998-11-16 YU YU29600A patent/YU29600A/sh unknown
- 1998-11-16 AT AT98955662T patent/ATE271875T1/de not_active IP Right Cessation
- 1998-11-16 JP JP2000520798A patent/JP4550273B2/ja not_active Expired - Fee Related
- 1998-11-16 AP APAP/P/2000/001825A patent/AP1196A/en active
- 1998-11-16 EE EEP200000244A patent/EE04095B1/xx not_active IP Right Cessation
- 1998-11-16 KR KR1020007005317A patent/KR20010032130A/ko not_active Ceased
- 1998-11-16 HU HU0004507A patent/HUP0004507A3/hu unknown
- 1998-11-16 EP EP98955662A patent/EP1030673B1/fr not_active Expired - Lifetime
- 1998-11-16 TR TR2000/01384T patent/TR200001384T2/xx unknown
- 1998-11-16 MA MA25348A patent/MA26566A1/fr unknown
- 1998-11-16 TN TNTNSN98206A patent/TNSN98206A1/fr unknown
- 1998-11-16 NZ NZ504305A patent/NZ504305A/xx unknown
- 1998-11-16 WO PCT/FR1998/002436 patent/WO1999025365A1/fr not_active Ceased
- 1998-11-16 CA CA002312021A patent/CA2312021C/fr not_active Expired - Fee Related
- 1998-11-16 AU AU12425/99A patent/AU744419B2/en not_active Ceased
- 1998-11-16 GE GEAP19985410A patent/GEP20032968B/en unknown
- 1998-11-16 PL PL98340373A patent/PL340373A1/xx unknown
- 1998-11-17 AR ARP980105823A patent/AR014119A1/es not_active Application Discontinuation
-
2000
- 2000-05-11 NO NO20002435A patent/NO20002435L/no unknown
- 2000-05-11 BG BG104427A patent/BG104427A/xx unknown
- 2000-05-17 OA OA1200000144A patent/OA11411A/fr unknown
-
2007
- 2007-09-28 US US11/863,329 patent/US20080139489A1/en not_active Abandoned
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |