AR004700A1 - 1alfa, 26 dihidroxi-d-homo-vitamina d3, una composicion farmaceutica que la comprende, un procedimiento para su preparacion y el uso de los mismos en laelaboracion de un medicamento - Google Patents
1alfa, 26 dihidroxi-d-homo-vitamina d3, una composicion farmaceutica que la comprende, un procedimiento para su preparacion y el uso de los mismos en laelaboracion de un medicamentoInfo
- Publication number
- AR004700A1 AR004700A1 ARP960104943A ARP960104943A AR004700A1 AR 004700 A1 AR004700 A1 AR 004700A1 AR P960104943 A ARP960104943 A AR P960104943A AR P960104943 A ARP960104943 A AR P960104943A AR 004700 A1 AR004700 A1 AR 004700A1
- Authority
- AR
- Argentina
- Prior art keywords
- homo
- vitamin
- procedure
- preparation
- pharmaceutical composition
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 229940126601 medicinal product Drugs 0.000 title 1
- 108010034984 D3 compound Proteins 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 239000011647 vitamin D3 Substances 0.000 abstract 1
- 229940021056 vitamin d3 Drugs 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C401/00—Irradiation products of cholesterol or its derivatives; Vitamin D derivatives, 9,10-seco cyclopenta[a]phenanthrene or analogues obtained by chemical preparation without irradiation
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Physical Education & Sports Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Engineering & Computer Science (AREA)
- Rheumatology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Un compuesto de 1alfa, 26-dihidroxi-D-homo-vitamina D3 de fórmula (I). Se refiere además a una composición farmacéutica que lo comprende, a unprocedimiento para su preparación y el uso del mismo en la elaboración de un medicamento.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP95117037 | 1995-10-30 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR004700A1 true AR004700A1 (es) | 1999-03-10 |
Family
ID=8219763
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP960104943A AR004700A1 (es) | 1995-10-30 | 1996-10-28 | 1alfa, 26 dihidroxi-d-homo-vitamina d3, una composicion farmaceutica que la comprende, un procedimiento para su preparacion y el uso de los mismos en laelaboracion de un medicamento |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US5905074A (es) |
| EP (1) | EP0771789B1 (es) |
| JP (1) | JP3059108B2 (es) |
| CN (1) | CN1157818A (es) |
| AR (1) | AR004700A1 (es) |
| AT (1) | ATE189812T1 (es) |
| BR (1) | BR9605354A (es) |
| CA (1) | CA2188634A1 (es) |
| DE (1) | DE69606680T2 (es) |
| DK (1) | DK0771789T3 (es) |
| ES (1) | ES2144183T3 (es) |
| GR (1) | GR3033254T3 (es) |
| MX (1) | MX9605206A (es) |
| PT (1) | PT771789E (es) |
| TR (1) | TR199600849A2 (es) |
Families Citing this family (30)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5763429A (en) * | 1993-09-10 | 1998-06-09 | Bone Care International, Inc. | Method of treating prostatic diseases using active vitamin D analogues |
| US6242434B1 (en) * | 1997-08-08 | 2001-06-05 | Bone Care International, Inc. | 24-hydroxyvitamin D, analogs and uses thereof |
| US20020183288A1 (en) * | 1995-04-03 | 2002-12-05 | Bone Care International, Inc. | Method for treating and preventing hyperparathyroidism |
| US6566353B2 (en) * | 1996-12-30 | 2003-05-20 | Bone Care International, Inc. | Method of treating malignancy associated hypercalcemia using active vitamin D analogues |
| US20020128240A1 (en) * | 1996-12-30 | 2002-09-12 | Bone Care International, Inc. | Treatment of hyperproliferative diseases using active vitamin D analogues |
| US5965734A (en) * | 1997-01-31 | 1999-10-12 | Celgene Corporation | Processes and intermediates for preparing 2-substituted piperidine stereoisomers |
| US20030129194A1 (en) * | 1997-02-13 | 2003-07-10 | Bone Care International, Inc. | Targeted therapeutic delivery of vitamin D compounds |
| CA2296145A1 (en) * | 1997-07-17 | 1999-01-28 | F. Hoffmann-La Roche Ag | Dihomo-seco-cholestanes with two unsaturated bonds in the side chain |
| US6087350A (en) * | 1997-08-29 | 2000-07-11 | University Of Pittsburgh Of The Commonwealth System Of Higher Education | Use of pretreatment chemicals to enhance efficacy of cytotoxic agents |
| US5919986A (en) * | 1997-10-17 | 1999-07-06 | Hoffmann-La Roche Inc. | D-homo vitamin D3 derivatives |
| EP2340840B1 (en) * | 1998-03-27 | 2012-08-29 | Oregon Health Sciences University | Pulse dose Vitamin D drug for the treatment of hyperproliferative skin diseases |
| ATE462689T1 (de) * | 1999-08-27 | 2010-04-15 | Hiroaki Takayama | Vitamin-d-derivate mit substituenten an der 2- alpha-position |
| US6358939B1 (en) | 1999-12-21 | 2002-03-19 | Northern Lights Pharmaceuticals, Llc | Use of biologically active vitamin D compounds for the prevention and treatment of inflammatory bowel disease |
| US6989377B2 (en) | 1999-12-21 | 2006-01-24 | Wisconsin Alumni Research Foundation | Treating vitamin D responsive diseases |
| IL153378A0 (en) * | 2000-07-18 | 2003-07-06 | Bone Care Internat Inc | STABILIZED 1alpha-HYDROXY VITAMIN D |
| US20030191093A1 (en) * | 2001-12-03 | 2003-10-09 | Novacea, Inc. | Pharmaceutical compositions comprising active vitamin D compounds |
| CA2503801A1 (en) * | 2001-12-26 | 2003-07-10 | Chugai Seiyaku Kabushiki Kaisha | 2-substituted vitamin d derivatives |
| US7148211B2 (en) * | 2002-09-18 | 2006-12-12 | Genzyme Corporation | Formulation for lipophilic agents |
| US20050026877A1 (en) * | 2002-12-03 | 2005-02-03 | Novacea, Inc. | Pharmaceutical compositions comprising active vitamin D compounds |
| CA2514614C (en) * | 2003-01-30 | 2011-09-13 | Teijin Pharma Limited | Vitamin d3 lactone derivatives |
| US20050020546A1 (en) * | 2003-06-11 | 2005-01-27 | Novacea, Inc. | Pharmaceutical compositions comprising active vitamin D compounds |
| US20060189586A1 (en) * | 2003-06-11 | 2006-08-24 | Cleland Jeffrey L | Pharmaceutical compositions comprising active vitamin D compounds |
| US20060003950A1 (en) * | 2004-06-30 | 2006-01-05 | Bone Care International, Inc. | Method of treating prostatic diseases using a combination of vitamin D analogues and other agents |
| US7094775B2 (en) * | 2004-06-30 | 2006-08-22 | Bone Care International, Llc | Method of treating breast cancer using a combination of vitamin D analogues and other agents |
| MX2007006545A (es) * | 2004-11-22 | 2007-09-21 | Wisconsin Alumni Res Found | 2a-metil-19-nor-1a-hidroxi-homopregnacalciferol y sus usos. |
| JP4719284B2 (ja) | 2008-10-10 | 2011-07-06 | トヨタ自動車株式会社 | 表面検査装置 |
| CA2981549A1 (en) | 2009-01-27 | 2010-08-05 | Berg Llc | Vitamin d3 and analogs thereof for alleviating side effects associated with chemotherapy |
| AU2010282731C1 (en) | 2009-08-14 | 2016-04-21 | Berg Llc | Vitamin D3 and analogs thereof for treating alopecia |
| CA2913543C (en) | 2013-05-29 | 2024-01-09 | Berg Llc | Preventing or mitigating chemotherapy induced alopecia using vitamin d |
| CN105348163B (zh) * | 2014-08-18 | 2017-06-16 | 武汉启瑞药业有限公司 | 维生素d类似物及其制备方法和医药用途 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3697559A (en) * | 1971-02-25 | 1972-10-10 | Wisconsin Alumni Res Found | 1,25-dihydroxycholecalciferol |
| US4410515A (en) * | 1981-04-01 | 1983-10-18 | Massachusetts General Hospital | Vitamin D glycosides and a method of use |
| US4595776A (en) * | 1983-03-21 | 1986-06-17 | Hoffmann-La Roche Inc. | Synthesis of 1α,25-dihydroxyergocalciferol |
| US4521410A (en) * | 1984-05-03 | 1985-06-04 | The General Hospital Corporation | Vitamin D glycosyl orthoesters |
| AU666563B2 (en) * | 1992-08-07 | 1996-02-15 | Wisconsin Alumni Research Foundation | Preparation of 19-nor-vitamin D compounds |
| DK0707566T3 (da) * | 1993-07-09 | 2000-09-04 | Theramex | Hidtil ukendte strukturelle analoger til vitamin D |
| FR2709126B1 (fr) * | 1993-08-18 | 1995-09-29 | Adir | Nouveaux dérivés de naphtalène, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent. |
-
1996
- 1996-10-18 ES ES96116735T patent/ES2144183T3/es not_active Expired - Lifetime
- 1996-10-18 AT AT96116735T patent/ATE189812T1/de not_active IP Right Cessation
- 1996-10-18 DK DK96116735T patent/DK0771789T3/da active
- 1996-10-18 DE DE69606680T patent/DE69606680T2/de not_active Expired - Fee Related
- 1996-10-18 PT PT96116735T patent/PT771789E/pt unknown
- 1996-10-18 EP EP96116735A patent/EP0771789B1/en not_active Expired - Lifetime
- 1996-10-23 CA CA002188634A patent/CA2188634A1/en not_active Abandoned
- 1996-10-24 TR TR96/00849A patent/TR199600849A2/xx unknown
- 1996-10-25 JP JP8283924A patent/JP3059108B2/ja not_active Expired - Lifetime
- 1996-10-28 CN CN96122882A patent/CN1157818A/zh active Pending
- 1996-10-28 AR ARP960104943A patent/AR004700A1/es unknown
- 1996-10-29 MX MX9605206A patent/MX9605206A/es not_active IP Right Cessation
- 1996-10-30 BR BR9605354A patent/BR9605354A/pt unknown
-
1997
- 1997-12-18 US US08/993,851 patent/US5905074A/en not_active Expired - Fee Related
-
2000
- 2000-04-17 GR GR20000400937T patent/GR3033254T3/el not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| EP0771789B1 (en) | 2000-02-16 |
| JPH09165369A (ja) | 1997-06-24 |
| MX198725B (es) | 2000-09-22 |
| DE69606680T2 (de) | 2000-08-17 |
| CA2188634A1 (en) | 1997-05-01 |
| ES2144183T3 (es) | 2000-06-01 |
| MX9605206A (es) | 1997-04-30 |
| GR3033254T3 (en) | 2000-09-29 |
| BR9605354A (pt) | 1998-07-28 |
| CN1157818A (zh) | 1997-08-27 |
| DK0771789T3 (da) | 2000-06-13 |
| US5905074A (en) | 1999-05-18 |
| TR199600849A2 (tr) | 1997-05-21 |
| DE69606680D1 (de) | 2000-03-23 |
| ATE189812T1 (de) | 2000-03-15 |
| PT771789E (pt) | 2000-05-31 |
| JP3059108B2 (ja) | 2000-07-04 |
| EP0771789A1 (en) | 1997-05-07 |
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