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AP2012006419A0 - Aminoquinoline derivatives - Google Patents

Aminoquinoline derivatives

Info

Publication number
AP2012006419A0
AP2012006419A0 AP2012006419A AP2012006419A AP2012006419A0 AP 2012006419 A0 AP2012006419 A0 AP 2012006419A0 AP 2012006419 A AP2012006419 A AP 2012006419A AP 2012006419 A AP2012006419 A AP 2012006419A AP 2012006419 A0 AP2012006419 A0 AP 2012006419A0
Authority
AP
ARIPO
Prior art keywords
aminoquinoline derivatives
aminoquinoline
derivatives
Prior art date
Application number
AP2012006419A
Other languages
English (en)
Inventor
Roger Tung
Original Assignee
Concert Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Concert Pharmaceuticals Inc filed Critical Concert Pharmaceuticals Inc
Publication of AP2012006419A0 publication Critical patent/AP2012006419A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38Nitrogen atoms
    • C07D215/40Nitrogen atoms attached in position 8
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/06Antimalarials
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/08Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis for Pneumocystis carinii

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AP2012006419A 2010-01-19 2011-01-19 Aminoquinoline derivatives AP2012006419A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US29626410P 2010-01-19 2010-01-19
PCT/US2011/021715 WO2011091035A1 (fr) 2010-01-19 2011-01-19 Dérivés d'aminoquinoléine

Publications (1)

Publication Number Publication Date
AP2012006419A0 true AP2012006419A0 (en) 2012-08-31

Family

ID=44307182

Family Applications (1)

Application Number Title Priority Date Filing Date
AP2012006419A AP2012006419A0 (en) 2010-01-19 2011-01-19 Aminoquinoline derivatives

Country Status (4)

Country Link
US (1) US20130053333A1 (fr)
AP (1) AP2012006419A0 (fr)
PH (1) PH12012501476A1 (fr)
WO (1) WO2011091035A1 (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2016109795A1 (fr) 2014-12-31 2016-07-07 Concert Pharmaceuticals, Inc. Funapide et difluorofunapide deutérés
US10683305B2 (en) 2015-04-27 2020-06-16 Concert Pharmaceuticals, Inc. Deuterated OTX-015
CN105348186B (zh) * 2015-10-15 2018-05-22 青岛海洋生物医药研究院股份有限公司 氘代双芳基脲类化合物及其制备方法和在制备抗肿瘤的药物中的应用
CN109438345A (zh) * 2018-11-14 2019-03-08 康化(上海)新药研发有限公司 一种二氘代伯氨喹的合成方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6342507B1 (en) * 1997-09-05 2002-01-29 Isotechnika, Inc. Deuterated rapamycin compounds, method and uses thereof

Also Published As

Publication number Publication date
WO2011091035A1 (fr) 2011-07-28
PH12012501476A1 (en) 2012-10-22
US20130053333A1 (en) 2013-02-28

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