OA10934A - Substituted indazole derivatives ad their use as phosphodiesterase (pde) type iv and tumor necrosis factor (tnf) inhibitors - Google Patents
Substituted indazole derivatives ad their use as phosphodiesterase (pde) type iv and tumor necrosis factor (tnf) inhibitors Download PDFInfo
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- OA10934A OA10934A OA9800235A OA9800235A OA10934A OA 10934 A OA10934 A OA 10934A OA 9800235 A OA9800235 A OA 9800235A OA 9800235 A OA9800235 A OA 9800235A OA 10934 A OA10934 A OA 10934A
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- alkyl
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- compound
- daim
- cyano
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- 108060008682 Tumor Necrosis Factor Proteins 0.000 title claims abstract description 21
- 102000003390 tumor necrosis factor Human genes 0.000 title claims abstract description 21
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
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- A—HUMAN NECESSITIES
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- A61P35/00—Antineoplastic agents
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- A61P37/00—Drugs for immunological or allergic disorders
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
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- Medicinal Chemistry (AREA)
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- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pain & Pain Management (AREA)
- Communicable Diseases (AREA)
- Obesity (AREA)
- Immunology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Rheumatology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Oncology (AREA)
- Dermatology (AREA)
- Pulmonology (AREA)
- Physical Education & Sports Medicine (AREA)
- Urology & Nephrology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US2038596P | 1996-06-25 | 1996-06-25 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| OA10934A true OA10934A (en) | 2002-02-18 |
Family
ID=21798354
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| OA9800235A OA10934A (en) | 1996-06-25 | 1998-12-11 | Substituted indazole derivatives ad their use as phosphodiesterase (pde) type iv and tumor necrosis factor (tnf) inhibitors |
Country Status (42)
| Country | Link |
|---|---|
| US (1) | US6040329A (fr) |
| EP (1) | EP0912558B1 (fr) |
| JP (1) | JP3152940B2 (fr) |
| KR (1) | KR20000022516A (fr) |
| CN (1) | CN1080260C (fr) |
| AP (1) | AP1025A (fr) |
| AR (1) | AR007456A1 (fr) |
| AT (1) | ATE244713T1 (fr) |
| AU (1) | AU716376B2 (fr) |
| BG (1) | BG64052B1 (fr) |
| BR (1) | BR9712782A (fr) |
| CA (1) | CA2258285C (fr) |
| CO (1) | CO4900056A1 (fr) |
| CZ (1) | CZ423398A3 (fr) |
| DE (1) | DE69723447T2 (fr) |
| DK (1) | DK0912558T3 (fr) |
| DZ (1) | DZ2254A1 (fr) |
| EA (1) | EA002274B1 (fr) |
| ES (1) | ES2201299T3 (fr) |
| GT (1) | GT199700075A (fr) |
| HN (1) | HN1997000079A (fr) |
| HR (1) | HRP970350B1 (fr) |
| HU (1) | HUP9903009A3 (fr) |
| ID (1) | ID18579A (fr) |
| IL (1) | IL127036A (fr) |
| IS (1) | IS4910A (fr) |
| MA (1) | MA24225A1 (fr) |
| MY (1) | MY116915A (fr) |
| NO (1) | NO986103L (fr) |
| NZ (1) | NZ332752A (fr) |
| OA (1) | OA10934A (fr) |
| PA (1) | PA8432301A1 (fr) |
| PL (1) | PL330974A1 (fr) |
| PT (1) | PT912558E (fr) |
| SI (1) | SI0912558T1 (fr) |
| SK (1) | SK176598A3 (fr) |
| TN (1) | TNSN97108A1 (fr) |
| TR (1) | TR199802685T2 (fr) |
| TW (1) | TW434237B (fr) |
| WO (1) | WO1997049702A1 (fr) |
| YU (1) | YU60198A (fr) |
| ZA (1) | ZA975581B (fr) |
Families Citing this family (39)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
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1997
- 1997-06-02 HU HU9903009A patent/HUP9903009A3/hu unknown
- 1997-06-02 TR TR1998/02685T patent/TR199802685T2/xx unknown
- 1997-06-02 CZ CZ984233A patent/CZ423398A3/cs unknown
- 1997-06-02 EP EP97921992A patent/EP0912558B1/fr not_active Expired - Lifetime
- 1997-06-02 DK DK97921992T patent/DK0912558T3/da active
- 1997-06-02 JP JP50258998A patent/JP3152940B2/ja not_active Expired - Fee Related
- 1997-06-02 KR KR1019980710961A patent/KR20000022516A/ko not_active Abandoned
- 1997-06-02 BR BR9712782-5A patent/BR9712782A/pt not_active Application Discontinuation
- 1997-06-02 DE DE69723447T patent/DE69723447T2/de not_active Expired - Fee Related
- 1997-06-02 AT AT97921992T patent/ATE244713T1/de not_active IP Right Cessation
- 1997-06-02 WO PCT/IB1997/000630 patent/WO1997049702A1/fr not_active Ceased
- 1997-06-02 PT PT97921992T patent/PT912558E/pt unknown
- 1997-06-02 SK SK1765-98A patent/SK176598A3/sk unknown
- 1997-06-02 AU AU27857/97A patent/AU716376B2/en not_active Ceased
- 1997-06-02 PL PL97330974A patent/PL330974A1/xx unknown
- 1997-06-02 CN CN97195846A patent/CN1080260C/zh not_active Expired - Fee Related
- 1997-06-02 ES ES97921992T patent/ES2201299T3/es not_active Expired - Lifetime
- 1997-06-02 CA CA002258285A patent/CA2258285C/fr not_active Expired - Fee Related
- 1997-06-02 SI SI9730553T patent/SI0912558T1/xx unknown
- 1997-06-02 IL IL12703697A patent/IL127036A/en not_active IP Right Cessation
- 1997-06-02 EA EA199801047A patent/EA002274B1/ru not_active IP Right Cessation
- 1997-06-05 HN HN1997000079A patent/HN1997000079A/es unknown
- 1997-06-05 US US08/869,358 patent/US6040329A/en not_active Expired - Fee Related
- 1997-06-10 PA PA19978432301A patent/PA8432301A1/es unknown
- 1997-06-12 GT GT199700075A patent/GT199700075A/es unknown
- 1997-06-19 AP APAP/P/1997/001020A patent/AP1025A/en active
- 1997-06-20 TW TW086108723A patent/TW434237B/zh not_active IP Right Cessation
- 1997-06-23 AR ARP970102755A patent/AR007456A1/es unknown
- 1997-06-23 MY MYPI97002820A patent/MY116915A/en unknown
- 1997-06-24 ID IDP972170A patent/ID18579A/id unknown
- 1997-06-24 DZ DZ970104A patent/DZ2254A1/fr active
- 1997-06-24 ZA ZA975581A patent/ZA975581B/xx unknown
- 1997-06-24 TN TNTNSN97108A patent/TNSN97108A1/fr unknown
- 1997-06-25 MA MA24679A patent/MA24225A1/fr unknown
- 1997-06-25 HR HR970350A patent/HRP970350B1/xx not_active Application Discontinuation
- 1997-06-25 CO CO97035540A patent/CO4900056A1/es unknown
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1998
- 1998-11-27 IS IS4910A patent/IS4910A/is unknown
- 1998-12-11 OA OA9800235A patent/OA10934A/en unknown
- 1998-12-23 NZ NZ332752A patent/NZ332752A/en unknown
- 1998-12-23 NO NO986103A patent/NO986103L/no not_active Application Discontinuation
- 1998-12-24 YU YU60198A patent/YU60198A/sh unknown
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1999
- 1999-01-07 BG BG103056A patent/BG64052B1/bg unknown
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