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NZ717669A - Process of producing cycloalkylcarboxamido-indole compounds - Google Patents

Process of producing cycloalkylcarboxamido-indole compounds

Info

Publication number
NZ717669A
NZ717669A NZ717669A NZ71766911A NZ717669A NZ 717669 A NZ717669 A NZ 717669A NZ 717669 A NZ717669 A NZ 717669A NZ 71766911 A NZ71766911 A NZ 71766911A NZ 717669 A NZ717669 A NZ 717669A
Authority
NZ
New Zealand
Prior art keywords
indole compounds
cycloalkylcarboxamido
intermediates
producing
protecting group
Prior art date
Application number
NZ717669A
Inventor
Elaine Chungmin Lee
Robert Michael Hughes
Peter Jamison Rose
Gerald J Tanoury
Daniel T Belmont
Cristian Harrison
David Andrew Siesel
Benjamin Joseph Littler
Young Chun Jung
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vertex Pharma filed Critical Vertex Pharma
Priority to NZ734535A priority Critical patent/NZ734535A/en
Publication of NZ717669A publication Critical patent/NZ717669A/en

Links

Classifications

    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Indole Compounds (AREA)

Abstract

intermediates for the preparation of Tezacaftor(VX-661) and its analogues. The intermediates are protecting group (P) bearing indole derivatives of formula III. the protecting group may be one of acetyl, benzoyl, benzyl, methoxyethoxymethyl, dimethoxytrityl, methoxymethyl, methoxytrityl, p-methoxybenzyl, pivaloyl, tetrahydropyranyl, trityl, or trimethylsilyl.
NZ717669A 2010-04-22 2011-04-21 Process of producing cycloalkylcarboxamido-indole compounds NZ717669A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
NZ734535A NZ734535A (en) 2010-04-22 2011-04-21 Process of producing cycloalkylcarboxamido-indole compounds

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US33387010P 2010-05-12 2010-05-12
NZ62900011 2011-04-21

Publications (1)

Publication Number Publication Date
NZ717669A true NZ717669A (en) 2017-09-29

Family

ID=59955235

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ717669A NZ717669A (en) 2010-04-22 2011-04-21 Process of producing cycloalkylcarboxamido-indole compounds

Country Status (1)

Country Link
NZ (1) NZ717669A (en)

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