NO975681D0 - Benzisoxazol- og indazol-derivater som antipsykotiske midler - Google Patents

Benzisoxazol- og indazol-derivater som antipsykotiske midler

Info

Publication number: NO975681D0
Authority: NO; Norway
Prior art keywords: benzisoxazole; antipsychotic agents; indazole derivatives; indazole; derivatives
Prior art date: 1995-06-06

Application number

NO975681A

Other languages

English (en)

Other versions

NO975681L (no

Inventor

Mark G Palermo

Lawrence L Martin

Peter A Nemoto

Original Assignee

Hoechst Marion Roussel Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-06-06

Filing date

1997-12-05

Publication date

1997-12-05

1997-12-05 Application filed by Hoechst Marion Roussel Inc filed Critical Hoechst Marion Roussel Inc

1997-12-05 Publication of NO975681D0 publication Critical patent/NO975681D0/no

1998-02-05 Publication of NO975681L publication Critical patent/NO975681L/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
- C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Psychiatry (AREA)
Pain & Pain Management (AREA)
Hospice & Palliative Care (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

NO975681A 1995-06-06 1997-12-05 Benzisoxazol- og indazol-derivater som antipsykotiske midler NO975681L (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US47040095A	1995-06-06	1995-06-06
PCT/US1996/006851 WO1996039397A1 (en)	1995-06-06	1996-05-14	Benzisoxazole and indazole derivatives as antipsychotic agents

Publications (2)

Publication Number	Publication Date
NO975681D0 true NO975681D0 (no)	1997-12-05
NO975681L NO975681L (no)	1998-02-05

Family

ID=23867483

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO975681A NO975681L (no)	1995-06-06	1997-12-05	Benzisoxazol- og indazol-derivater som antipsykotiske midler

Country Status (20)

Country	Link
US (3)	US5696113A (no)
EP (1)	EP0833820B1 (no)
JP (2)	JP3057763B2 (no)
KR (1)	KR100304179B1 (no)
AR (1)	AR002300A1 (no)
AT (1)	ATE199147T1 (no)
AU (1)	AU697953B2 (no)
CA (1)	CA2218663C (no)
DE (1)	DE69611783T2 (no)
DK (1)	DK0833820T3 (no)
ES (1)	ES2157442T3 (no)
GR (1)	GR3035663T3 (no)
HU (1)	HUP9802492A3 (no)
IL (1)	IL118530A0 (no)
MX (1)	MX9709451A (no)
NO (1)	NO975681L (no)
NZ (1)	NZ307958A (no)
PT (1)	PT833820E (no)
WO (2)	WO1996039397A1 (no)
ZA (1)	ZA964562B (no)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6008348A (en) *	1995-06-06	1999-12-28	Hoechst Marion Roussel, Inc.	Antipsychotic agents, compositions and method of use
TW487572B (en) *	1996-05-20	2002-05-21	Janssen Pharmaceutica Nv	Aqueous suspensions of 9-hydroxyrisperidone fatty acid esters
UA72189C2 (uk)	1997-11-17	2005-02-15	Янссен Фармацевтика Н.В.	Фармацевтична композиція, що містить водну суспензію субмікронних ефірів 9-гідроксирисперидон жирних кислот
US7253165B2 (en) *	1999-09-14	2007-08-07	Aventis Pharmaceuticals Inc.	Benzisoxazolyl-, pyridoisoxazolyl-and benzthienyl-phenoxy derivatives useful as D4 antagonists
US7125903B1 (en)	1999-09-14	2006-10-24	Aventis Pharmaceuticals Inc.	Thienoisoxazolyl-and thienylpyrrazolyl-phenoxy substituted propyl derivatives useful as D4 antagonists
US7091199B1 (en)	1999-09-14	2006-08-15	Aventis Pharmaceuticals Inc.	Thienoisoxazole phenoxy unsubstituted ethyl and propyl derivatives useful as d4 antagonists
GB0117531D0 (en) *	2001-02-16	2001-09-12	Aventis Pharm Prod Inc	Novel heterocyclic amide derivatives and their use as dopamine D3 receptor ligands
KR100627031B1 (ko) *	2004-09-04	2006-09-21	주식회사 케이티프리텔	등산 정보 서비스 제공 방법 및 장치
DE102005038947A1 (de) *	2005-05-18	2006-11-30	Grünenthal GmbH	Substituierte Benzo[d]isoxazol-3-yl-amin-Verbindungen und deren Verwendung in Arzneimitteln
KR100673033B1 (ko) *	2005-06-21	2007-01-22	(주) 엘지텔레콤	레저 전용 휴대 단말기
US7696229B2 (en)	2006-02-17	2010-04-13	Memory Pharmaceuticals Corporation	Compounds having 5-HT6 receptor affinity
JP2012502948A (ja) *	2008-09-23	2012-02-02	エフ．ホフマン−ラロシュアーゲー	ドーパミンｄ３受容体の調節剤として有用なイソオキサゾロ［４，５］ピリジン−３−イル−ピペラジン誘導体
TW201103904A (en) *	2009-06-11	2011-02-01	Hoffmann La Roche	Janus kinase inhibitor compounds and methods
CN110117278B (zh) *	2018-02-07	2022-07-19	石家庄以岭药业股份有限公司	烷氧基苯并五元(六元)杂环胺类化合物及其药物用途

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4411901A (en) *	1981-12-23	1983-10-25	Mead Johnson & Company	Benzisothiazole and benzisoxazole piperazine derivatives
US4670447A (en) *	1983-08-22	1987-06-02	Hoechst-Roussel Pharmaceuticals Inc.	Antipsychotic 3-(piperidinyl)- and 3-(pyrrolidinyl)-1H-indazoles
US4853470A (en) *	1983-08-22	1989-08-01	Hoechst-Roussel Pharmaceuticals, Inc.	3-(piperidinyl)- and 3-(pyrrolidinyl)-1H-indazoles
US4806649A (en) *	1983-08-22	1989-02-21	Hoechst-Roussel Pharmaceuticals, Inc.	3-(piperidinyl)- and 3- (pyrrolidinyl)-1H-indazoles
US4590196A (en) *	1984-08-23	1986-05-20	Bristol-Myers Company	Analgesic 1,2-benzisothiazol-3-ylpiperazine derivatives
MX174210B (es) *	1987-02-17	1994-04-28	Pfizer	Procedimiento para la preparacion de compuestos arilpiperazinil-alquilenfenil-p-heterociclicos
EP0302423A3 (en) *	1987-08-07	1991-01-09	Hoechst-Roussel Pharmaceuticals Incorporated	1-phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments
NZ233525A (en) *	1989-05-15	1991-09-25	Janssen Pharmaceutica Nv	Piperidinyl, pyrrolidinyl and piperazinyl alkylphenol ethers and pharmaceutical compositions
US5364866A (en) *	1989-05-19	1994-11-15	Hoechst-Roussel Pharmaceuticals, Inc.	Heteroarylpiperidines, pyrrolidines and piperazines and their use as antipsychotics and analetics
ATE126512T1 (de) *	1989-05-19	1995-09-15	Hoechst Roussel Pharma	N-(aryloxyalkyl)heteroarylpiperidine und - heteroarylpiperazine, verfahren zu ihrer herstellung und ihre verwendung als medikamente.
US5077405A (en) *	1989-09-11	1991-12-31	Hoechst-Roussel Pharmaceuticals Incorporated	3-(1-Substituted-4-piperazinyl)-1H-indazoles
US4954503A (en) *	1989-09-11	1990-09-04	Hoechst-Roussel Pharmaceuticals, Inc.	3-(1-substituted-4-piperazinyl)-1H-indazoles
FR2671350A1 (fr) *	1991-01-08	1992-07-10	Adir	Nouveaux derives de benzisoxazole et de benzisothiazole, leur procede de preparation, et les compositions pharmaceutiques les renfermant.
FI934223L (fi) *	1991-03-28	1993-09-27	Pfizer	Heterocykliscykliska aminderivat
US5177088A (en) *	1991-04-17	1993-01-05	Hoechst-Roussel Pharmaceuticals Incorporated	Substituted 3-(pyridinylamino)-indoles
US5328920A (en) *	1991-04-17	1994-07-12	Hoechst-Roussel Pharmaceuticals Incorporated	Substituted (pyridinylamino)-indoles
US5206366A (en) *	1992-08-26	1993-04-27	Pfizer Inc.	Process for preparing aryl piperazinyl-heterocyclic compounds
US5494908A (en) *	1992-11-23	1996-02-27	Hoechst-Roussel Pharmaceutical Incorporated	Substituted 3-(aminoalkylamino)-1,2-benzisoxazoles and related compounds

1996
- 1996-05-14 ES ES96915782T patent/ES2157442T3/es not_active Expired - Lifetime
- 1996-05-14 KR KR1019970708743A patent/KR100304179B1/ko not_active Expired - Fee Related
- 1996-05-14 NZ NZ307958A patent/NZ307958A/xx unknown
- 1996-05-14 JP JP9500561A patent/JP3057763B2/ja not_active Expired - Fee Related
- 1996-05-14 MX MX9709451A patent/MX9709451A/es unknown
- 1996-05-14 HU HU9802492A patent/HUP9802492A3/hu unknown
- 1996-05-14 EP EP96915782A patent/EP0833820B1/en not_active Expired - Lifetime
- 1996-05-14 JP JP09500630A patent/JP3122469B2/ja not_active Expired - Fee Related
- 1996-05-14 WO PCT/US1996/006851 patent/WO1996039397A1/en not_active Ceased
- 1996-05-14 DE DE69611783T patent/DE69611783T2/de not_active Expired - Fee Related
- 1996-05-14 AU AU57464/96A patent/AU697953B2/en not_active Ceased
- 1996-05-14 PT PT96915782T patent/PT833820E/pt unknown
- 1996-05-14 DK DK96915782T patent/DK0833820T3/da active
- 1996-05-14 CA CA002218663A patent/CA2218663C/en not_active Expired - Fee Related
- 1996-05-14 WO PCT/US1996/007319 patent/WO1996039405A1/en not_active Ceased
- 1996-05-14 AT AT96915782T patent/ATE199147T1/de not_active IP Right Cessation
- 1996-06-02 IL IL11853096A patent/IL118530A0/xx unknown
- 1996-06-03 ZA ZA964562A patent/ZA964562B/xx unknown
- 1996-06-04 AR ARP960102884A patent/AR002300A1/es unknown
- 1996-06-27 US US08/672,127 patent/US5696113A/en not_active Expired - Fee Related
1997
- 1997-09-02 US US08/921,480 patent/US5852022A/en not_active Expired - Fee Related
- 1997-12-05 NO NO975681A patent/NO975681L/no not_active Application Discontinuation
1998
- 1998-09-11 US US09/150,971 patent/US5965554A/en not_active Expired - Fee Related
2001
- 2001-03-29 GR GR20010400513T patent/GR3035663T3/el not_active IP Right Cessation

Also Published As

Publication number	Publication date
ES2157442T3 (es)	2001-08-16
IL118530A0 (en)	1996-10-16
NZ307958A (en)	1999-02-25
AU5746496A (en)	1996-12-24
US5852022A (en)	1998-12-22
EP0833820A1 (en)	1998-04-08
DK0833820T3 (da)	2001-04-17
JP3057763B2 (ja)	2000-07-04
ATE199147T1 (de)	2001-02-15
MX9709451A (es)	1998-02-28
US5965554A (en)	1999-10-12
JPH11507030A (ja)	1999-06-22
WO1996039405A1 (en)	1996-12-12
AU697953B2 (en)	1998-10-22
CA2218663C (en)	2001-07-31
KR19990022264A (ko)	1999-03-25
CA2218663A1 (en)	1996-12-12
DE69611783T2 (de)	2001-09-20
JPH11506728A (ja)	1999-06-15
KR100304179B1 (ko)	2001-11-22
US5696113A (en)	1997-12-09
GR3035663T3 (en)	2001-06-29
JP3122469B2 (ja)	2001-01-09
WO1996039397A1 (en)	1996-12-12
PT833820E (pt)	2001-07-31
NO975681L (no)	1998-02-05
HUP9802492A2 (hu)	1999-09-28
DE69611783D1 (de)	2001-03-22
HUP9802492A3 (en)	1999-10-28
ZA964562B (en)	1996-12-12
AR002300A1 (es)	1998-03-11
EP0833820B1 (en)	2001-02-14

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FI970864A7 (fi)	1997-04-24	Isoksatsolijohdannaiset
NO963244L (no)	1996-08-02	Orale flytende preparater inneholdende paroxetin-resinat
DE69930518D1 (de)	2006-05-11	Als antikrebsmittel verwendbare alkinyl-substituierte chinolin-2-on-derivate
DK0832061T3 (da)	2001-11-19	Benzamidderivater og anvendelse deraf som vasopressin-antagonister
NO975496L (no)	1998-01-22	Isotiazoloner
KR970707039A (ko)	1997-12-01	알루미노-실리케이트 유도체(alumino-silicate derivatives)
DE59608798D1 (de)	2002-04-04	Endoparasitizide mittel
BR9709051A (pt)	1999-08-03	Derivados de indazol substituidos e compostos relacionados
NO984106D0 (no)	1998-09-07	Azolobenzazepin-derivater som neurologisk aktive midler
DK0991658T3 (da)	2006-05-15	Dolastatin 15-derivater
EP0708091A3 (en)	1996-07-17	Indoloyl-guanidines derivatives
FI971510A7 (fi)	1997-04-11	Atsolijohdannainen
NO984761D0 (no)	1998-10-12	Aminoisokinoliner og aminotienopyridinderivater og deres anvendelse som antiinflammatoriske midler
DK0833820T3 (da)	2001-04-17	Benzisoxazol- og indazolderivater som antipsykotiske midler
DE69520235D1 (de)	2001-04-05	Schweisshemmende mittel
DE69601527D1 (de)	1999-03-25	Pyrrolylbenzimidazol-Derivate
DK0747346T3 (da)	2000-06-05	N-acyl-2-arylcyclopropylmethylaminderivater som melatonerge midler
FI971227L (fi)	1997-05-23	Pyramidinyylipyratsolijohdannaisia
NO975880L (no)	1998-02-13	Formylderivater anvendt som ikke-ioniske kontrastmidler
ATE239018T1 (de)	2003-05-15	Pyrazol-derivate
ATE204255T1 (de)	2001-09-15	Carbostyrilderivate als antithrombotische mittel
ATE192428T1 (de)	2000-05-15	Nitro-benzamides verwendbar als antiarrythmica
DK0848713T3 (da)	2000-12-18	Pyridiniminyl-1,2-benzisoxazoler og -benzisothiazoler som antipsykotiske midler
DE69624122D1 (de)	2002-11-07	Aza-anthracyclinone-derivate
DE59607055D1 (de)	2001-07-19	4-Mercapto-benzoylguanidin-Derivate

Legal Events

Date	Code	Title	Description
2001-01-22	FC2A	Withdrawal, rejection or dismissal of laid open patent application