NO306022B1 - Process for obtaining 3- {2- [4- (6-fluoro-benzo [d] isoxazol-3-yl) piperidin-1-yl] ethyl} -2-methyl-6,7,8,9-tetrahydro -4H-pyrido [1,2-a] pyrimidin-4-one - Google Patents

Process for obtaining 3- {2- [4- (6-fluoro-benzo [d] isoxazol-3-yl) piperidin-1-yl] ethyl} -2-methyl-6,7,8,9-tetrahydro -4H-pyrido [1,2-a] pyrimidin-4-one

Info

Publication number: NO306022B1
Authority: NO; Norway
Prior art keywords: isoxazol; pyrido; pyrimidin; piperidin; benzo
Prior art date: 1994-02-11

Application number

NO950501A

Other languages

Norwegian (no)

Other versions

NO950501L (en

NO950501D0 (en

Inventor

Pere Dalmases Barjoan

Francisco Marquillas Olondriz

Joan Huguet Clotet

Ana Bosch Rovira

Juan Carlos Del Castillo Nieto

Jose Maria Caldero Ges

Original Assignee

Vita Invest Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1994-02-11

Filing date

1995-02-09

Publication date

1999-09-06

1995-02-09 Application filed by Vita Invest Sa filed Critical Vita Invest Sa

1995-02-09 Publication of NO950501D0 publication Critical patent/NO950501D0/en

1995-08-14 Publication of NO950501L publication Critical patent/NO950501L/en

1999-09-06 Publication of NO306022B1 publication Critical patent/NO306022B1/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

NO950501A 1994-02-11 1995-02-09 Process for obtaining 3- {2- [4- (6-fluoro-benzo [d] isoxazol-3-yl) piperidin-1-yl] ethyl} -2-methyl-6,7,8,9-tetrahydro -4H-pyrido [1,2-a] pyrimidin-4-one NO306022B1 (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
ES09400252A ES2074966B1 (en)	1994-02-11	1994-02-11	PROCEDURE FOR OBTAINING 3- (2- (4- (6-FLUORO-BENZO (D) ISOXAZOL-3-IL) PIPERIDIN-1-IL) -ETIL) -2-METHYL-6,7,8,9- TETRAHIDRO-4H-PIRIDO- (1,2-A) PIRIMIDIN-4-ONA.

Publications (3)

Publication Number	Publication Date
NO950501D0 NO950501D0 (en)	1995-02-09
NO950501L NO950501L (en)	1995-08-14
NO306022B1 true NO306022B1 (en)	1999-09-06

Family

ID=8285178

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO950501A NO306022B1 (en)	1994-02-11	1995-02-09	Process for obtaining 3- {2- [4- (6-fluoro-benzo [d] isoxazol-3-yl) piperidin-1-yl] ethyl} -2-methyl-6,7,8,9-tetrahydro -4H-pyrido [1,2-a] pyrimidin-4-one

Country Status (14)

Country	Link
KR (1)	KR100221108B1 (en)
AT (1)	AT405401B (en)
CZ (1)	CZ286398B6 (en)
EG (1)	EG20877A (en)
ES (1)	ES2074966B1 (en)
FI (1)	FI110000B (en)
GR (1)	GR1002344B (en)
HU (1)	HU222110B1 (en)
IS (1)	IS1766B (en)
NO (1)	NO306022B1 (en)
PL (1)	PL181420B1 (en)
PT (1)	PT101654B (en)
RU (1)	RU2123004C1 (en)
SK (1)	SK281752B6 (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES2101646B1 (en) *	1995-04-12	1998-04-01	Ferrer Int	NEW COMPOUND DERIVED FROM CHROMENE.
ES2144355B1 (en) *	1997-12-30	2001-01-01	Ferrer Int	COMPOUNDS DERIVED FROM THE CHROME.
CZ295402B6 (en) *	2000-05-05	2005-08-17	Rpg Life Sciences Limited	Process for the preparation of anti-psychotic 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2,-a]pyrimidin-4-one
CA2419314C (en)	2000-08-14	2006-07-11	Teva Pharmaceutical Industries Ltd.	Preparation of risperidone
ES2197801B1 (en) *	2002-03-05	2005-03-16	Ferrer Internacional,S.A	PROCEDURE FOR OBTAINING THE 3- (2- (4- (6-FLUORO-BENZO (D) ISOXAZOL-3-IL) PIPERIDIN-1-IL) -ETIL) -2-METHYL-6,7,8,9- TETRAHIDRO-4H-PIRIDO- (1,2-A) PIRIMIDIN-4-ONA.
KR20040034996A (en)	2002-10-18	2004-04-29	한미약품 주식회사	Improved method for the preparation of risperidone
CN100390146C (en)	2002-11-13	2008-05-28	斯索恩有限公司	Process for preparing risperidone and intermediates therefor
RU2310653C1 (en) *	2006-07-17	2007-11-20	Государственное образовательное учреждение высшего профессионального образования "Кубанский государственный технологический университет" (ГОУВПО "КубГТУ")	METHOD FOR PREPARING DERIVATIVES OF 2-METHYL-5-(5-METHYL-2-FURYL)-4,10-DIHYDRO-3H-PYRIDAZINO[1,6-b]ISOQUINOLINE-10-ONE (VARIANTS)
US8314110B2 (en) *	2007-04-19	2012-11-20	Youxin Li	Compounds for treating mental disorders, and preparation and uses thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AT327199B (en) *	1971-10-14	1976-01-26	Sumitomo Chemical Co	PROCESS FOR PRODUCING NEW NITROCHINAZOLINONES
US4352811A (en) *	1981-11-12	1982-10-05	Hoechst-Roussel Pharmaceuticals Inc.	3-(1-Substituted-4-piperidyl)-1,2-benzisoxazoles
US4485107A (en) *	1982-11-01	1984-11-27	Janssen Pharmaceutica N.V.	[[Bis(aryl)methylene]-1-piperidinyl]alkyl-pyrimidinones
US4804663A (en) *	1985-03-27	1989-02-14	Janssen Pharmaceutica N.V.	3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles
US4980365A (en) *	1987-07-13	1990-12-25	Hoechst-Roussel Pharmaceuticals Inc.	N-substituted-5,6-dimethoxy-1,2-benzisoxazole-3-propanamine and related compounds as analgesic and hypotensive agents

1994
- 1994-02-11 ES ES09400252A patent/ES2074966B1/en not_active Expired - Fee Related
1995
- 1995-02-01 GR GR950100035A patent/GR1002344B/en not_active IP Right Cessation
- 1995-02-07 SK SK156-95A patent/SK281752B6/en not_active IP Right Cessation
- 1995-02-08 CZ CZ1995329A patent/CZ286398B6/en not_active IP Right Cessation
- 1995-02-08 IS IS4259A patent/IS1766B/en unknown
- 1995-02-09 NO NO950501A patent/NO306022B1/en not_active IP Right Cessation
- 1995-02-09 PT PT101654A patent/PT101654B/en active IP Right Grant
- 1995-02-09 EG EG11595A patent/EG20877A/en active
- 1995-02-10 AT AT0024995A patent/AT405401B/en not_active IP Right Cessation
- 1995-02-10 RU RU95101859/04A patent/RU2123004C1/en not_active IP Right Cessation
- 1995-02-10 FI FI950579A patent/FI110000B/en not_active IP Right Cessation
- 1995-02-10 PL PL95307200A patent/PL181420B1/en not_active IP Right Cessation
- 1995-02-10 HU HU9500418A patent/HU222110B1/en not_active IP Right Cessation
- 1995-02-11 KR KR1019950002516A patent/KR100221108B1/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
KR950032196A (en)	1995-12-20
HUT70169A (en)	1995-09-28
PL307200A1 (en)	1995-08-21
RU95101859A (en)	1997-03-20
RU2123004C1 (en)	1998-12-10
CZ286398B6 (en)	2000-04-12
NO950501L (en)	1995-08-14
FI950579L (en)	1995-08-12
FI110000B (en)	2002-11-15
CZ32995A3 (en)	1995-09-13
SK15695A3 (en)	1995-10-11
GR1002344B (en)	1996-05-24
IS4259A (en)	1995-08-12
IS1766B (en)	2001-03-15
SK281752B6 (en)	2001-07-10
PL181420B1 (en)	2001-07-31
ES2074966B1 (en)	1996-06-16
AT405401B (en)	1999-08-25
NO950501D0 (en)	1995-02-09
KR100221108B1 (en)	1999-09-15
ATA24995A (en)	1998-12-15
PT101654A (en)	1995-09-12
HU222110B1 (en)	2003-04-28
ES2074966A1 (en)	1995-09-16
HU9500418D0 (en)	1995-03-28
FI950579A0 (en)	1995-02-10
PT101654B (en)	2002-01-30
EG20877A (en)	2000-05-31

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Legal Events

Date	Code	Title	Description
2011-09-26	MM1K	Lapsed by not paying the annual fees