NO20091057L - Oral form of birth control - Google Patents
Oral form of birth controlInfo
- Publication number
- NO20091057L NO20091057L NO20091057A NO20091057A NO20091057L NO 20091057 L NO20091057 L NO 20091057L NO 20091057 A NO20091057 A NO 20091057A NO 20091057 A NO20091057 A NO 20091057A NO 20091057 L NO20091057 L NO 20091057L
- Authority
- NO
- Norway
- Prior art keywords
- birth control
- dienogest
- oral form
- less
- daily dose
- Prior art date
Links
- BFPYWIDHMRZLRN-SLHNCBLASA-N Ethinyl estradiol Chemical compound OC1=CC=C2[C@H]3CC[C@](C)([C@](CC4)(O)C#C)[C@@H]4[C@@H]3CCC2=C1 BFPYWIDHMRZLRN-SLHNCBLASA-N 0.000 abstract 3
- 239000004480 active ingredient Substances 0.000 abstract 2
- AZFLJNIPTRTECV-FUMNGEBKSA-N dienogest Chemical compound C1CC(=O)C=C2CC[C@@H]([C@H]3[C@@](C)([C@](CC3)(O)CC#N)CC3)C3=C21 AZFLJNIPTRTECV-FUMNGEBKSA-N 0.000 abstract 2
- 229960003309 dienogest Drugs 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 1
- 239000003937 drug carrier Substances 0.000 abstract 1
- 229960002568 ethinylestradiol Drugs 0.000 abstract 1
- 230000003179 granulation Effects 0.000 abstract 1
- 238000005469 granulation Methods 0.000 abstract 1
- 239000002245 particle Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
- A61K31/569—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone substituted in position 17 alpha, e.g. ethisterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/567—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Reproductive Health (AREA)
- Engineering & Computer Science (AREA)
- Endocrinology (AREA)
- Epidemiology (AREA)
- Gynecology & Obstetrics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Steroid Compounds (AREA)
Abstract
Oral legemiddelform for prevensjon omfatter som en aktiv forbindelse, 17a-cyanometyl-17-ß-hydroksyøstra-4,9-dien-3-on (dienogest) i en daglig dose lik eller mindre enn 2,0 mg og som annen aktiv komponent 17a-etynyløstradiol (etynyløstradiol) i en daglig dose på mindre enn 0,03 mg, sammen med én eller flere farmasøytisk akseptable bærere. Den aktive bestanddel dienogest er til stede i krystallinsk form med en midlere partikkelstørrelse på fra 25 til 70 µm. Den aktive bestanddel etynyløstradiol er innført i mikronisert form eller som etanolisk løsning under granuleringen.Oral form of birth control comprises, as an active compound, 17α-cyanomethyl-17-β-hydroxyester-4,9-dien-3-one (dienogest) in a daily dose equal to or less than 2.0 mg and as another active component 17a -ethynyl estradiol (ethynyl estradiol) at a daily dose of less than 0.03 mg, together with one or more pharmaceutically acceptable carriers. The active ingredient dienogest is present in crystalline form with an average particle size of from 25 to 70 µm. The active ingredient ethynyl oestradiol is introduced in micronized form or as ethanolic solution during the granulation.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP06016694A EP1886694B1 (en) | 2006-08-10 | 2006-08-10 | Peroral formulation of dienogest and ethinylestradiol for contraception |
| PCT/EP2007/003662 WO2008017331A2 (en) | 2006-08-10 | 2007-04-26 | Peroral drug form comprising dienogest and ethinyl estradiol for contraception |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO20091057L true NO20091057L (en) | 2009-03-09 |
Family
ID=37561777
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20091057A NO20091057L (en) | 2006-08-10 | 2009-03-09 | Oral form of birth control |
Country Status (18)
| Country | Link |
|---|---|
| EP (1) | EP1886694B1 (en) |
| AR (1) | AR062323A1 (en) |
| AT (1) | ATE432714T1 (en) |
| CL (1) | CL2007002323A1 (en) |
| CY (1) | CY1110348T1 (en) |
| DE (1) | DE502006003892D1 (en) |
| DK (1) | DK1886694T3 (en) |
| DO (1) | DOP2007000122A (en) |
| ES (1) | ES2327665T3 (en) |
| HR (1) | HRP20090438T1 (en) |
| NO (1) | NO20091057L (en) |
| PE (1) | PE20080541A1 (en) |
| PL (1) | PL1886694T3 (en) |
| PT (1) | PT1886694E (en) |
| SI (1) | SI1886694T1 (en) |
| TW (1) | TW200817012A (en) |
| UY (1) | UY30530A1 (en) |
| WO (1) | WO2008017331A2 (en) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE102010003711B4 (en) | 2010-04-08 | 2015-04-09 | Jesalis Pharma Gmbh | Process for the preparation of crystalline active substance particles |
| CN115487198B (en) * | 2022-09-20 | 2024-01-02 | 华中药业股份有限公司 | Levonorgestrel preparation with fast dissolution rate and preparation method thereof |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1216713A1 (en) * | 2000-12-20 | 2002-06-26 | Schering Aktiengesellschaft | Compositions of estrogen-cyclodextrin complexes |
| DE10218107A1 (en) * | 2002-04-23 | 2003-11-20 | Jenapharm Gmbh | Process for the production of crystals of steroids, crystals available thereafter and their use in pharmaceutical formulations |
-
2006
- 2006-08-10 DE DE502006003892T patent/DE502006003892D1/en active Active
- 2006-08-10 ES ES06016694T patent/ES2327665T3/en active Active
- 2006-08-10 EP EP06016694A patent/EP1886694B1/en active Active
- 2006-08-10 DK DK06016694T patent/DK1886694T3/en active
- 2006-08-10 PL PL06016694T patent/PL1886694T3/en unknown
- 2006-08-10 SI SI200630376T patent/SI1886694T1/en unknown
- 2006-08-10 AT AT06016694T patent/ATE432714T1/en active
- 2006-08-10 PT PT06016694T patent/PT1886694E/en unknown
-
2007
- 2007-04-26 WO PCT/EP2007/003662 patent/WO2008017331A2/en not_active Ceased
- 2007-07-16 TW TW096125903A patent/TW200817012A/en unknown
- 2007-08-07 UY UY30530A patent/UY30530A1/en unknown
- 2007-08-09 CL CL200702323A patent/CL2007002323A1/en unknown
- 2007-08-09 DO DO2007000122A patent/DOP2007000122A/en unknown
- 2007-08-09 PE PE2007001064A patent/PE20080541A1/en not_active Application Discontinuation
- 2007-08-10 AR ARP070103547A patent/AR062323A1/en not_active Application Discontinuation
-
2009
- 2009-03-09 NO NO20091057A patent/NO20091057L/en not_active Application Discontinuation
- 2009-08-13 HR HR20090438T patent/HRP20090438T1/en unknown
- 2009-09-03 CY CY20091100928T patent/CY1110348T1/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ES2327665T3 (en) | 2009-11-02 |
| PT1886694E (en) | 2009-08-17 |
| WO2008017331A2 (en) | 2008-02-14 |
| CL2007002323A1 (en) | 2008-02-15 |
| EP1886694B1 (en) | 2009-06-03 |
| UY30530A1 (en) | 2008-03-31 |
| WO2008017331A3 (en) | 2009-01-08 |
| PL1886694T3 (en) | 2009-11-30 |
| CY1110348T1 (en) | 2015-04-29 |
| SI1886694T1 (en) | 2009-10-31 |
| ATE432714T1 (en) | 2009-06-15 |
| EP1886694A1 (en) | 2008-02-13 |
| DOP2007000122A (en) | 2008-02-15 |
| TW200817012A (en) | 2008-04-16 |
| DE502006003892D1 (en) | 2009-07-16 |
| DK1886694T3 (en) | 2009-09-28 |
| AR062323A1 (en) | 2008-10-29 |
| PE20080541A1 (en) | 2008-07-10 |
| HRP20090438T1 (en) | 2009-09-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |