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NO20084533L - Pyrimidin-derivat som PI3K-inhibitor og bruk av dette - Google Patents

Pyrimidin-derivat som PI3K-inhibitor og bruk av dette

Info

Publication number
NO20084533L
NO20084533L NO20084533A NO20084533A NO20084533L NO 20084533 L NO20084533 L NO 20084533L NO 20084533 A NO20084533 A NO 20084533A NO 20084533 A NO20084533 A NO 20084533A NO 20084533 L NO20084533 L NO 20084533L
Authority
NO
Norway
Prior art keywords
pi3k inhibitor
pyrimidine derivative
pyrimidine
derivative
pi3k
Prior art date
Application number
NO20084533A
Other languages
English (en)
Other versions
NO342978B1 (no
Inventor
Nobuo Shimma
Jun Ohwada
Hirosato Ebiike
Hatsuo Kawada
Kenji Morikami
Mitsuaki Nakamura
Miyuki Yoshida
Nobuya Ishii
Masami Hasegawa
Shun Yamamoto
Kohei Koyama
Original Assignee
Chugai Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39032956&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20084533(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Chugai Pharmaceutical Co Ltd filed Critical Chugai Pharmaceutical Co Ltd
Publication of NO20084533L publication Critical patent/NO20084533L/no
Publication of NO342978B1 publication Critical patent/NO342978B1/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
NO20084533A 2006-08-08 2008-10-28 Pyrimidin-derivat som PI3K-inhibitor og bruk av dette NO342978B1 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2006216108 2006-08-08
JP2007118631 2007-04-27
PCT/JP2007/065396 WO2008018426A1 (en) 2006-08-08 2007-08-07 Pyrimidine derivative as pi3k inhibitor and use thereof

Publications (2)

Publication Number Publication Date
NO20084533L true NO20084533L (no) 2009-01-09
NO342978B1 NO342978B1 (no) 2018-09-17

Family

ID=39032956

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20084533A NO342978B1 (no) 2006-08-08 2008-10-28 Pyrimidin-derivat som PI3K-inhibitor og bruk av dette

Country Status (26)

Country Link
US (1) US8022205B2 (no)
EP (1) EP2050749B1 (no)
JP (1) JP4450857B2 (no)
KR (1) KR101435692B1 (no)
AR (1) AR062292A1 (no)
AU (1) AU2007282535B9 (no)
BR (1) BRPI0714908B8 (no)
CA (1) CA2659604C (no)
CL (1) CL2007002316A1 (no)
CY (1) CY1119882T1 (no)
DK (1) DK2050749T3 (no)
ES (1) ES2657635T3 (no)
HU (1) HUE035116T2 (no)
IL (1) IL196601A (no)
LT (1) LT2050749T (no)
MX (1) MX2009001451A (no)
MY (1) MY145385A (no)
NO (1) NO342978B1 (no)
NZ (1) NZ575274A (no)
PE (1) PE20080527A1 (no)
PL (1) PL2050749T3 (no)
PT (1) PT2050749T (no)
RU (1) RU2448109C2 (no)
SI (1) SI2050749T1 (no)
TW (1) TWI394758B (no)
WO (1) WO2008018426A1 (no)

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US8822513B2 (en) 2010-03-01 2014-09-02 Gtx, Inc. Compounds for treatment of cancer
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Also Published As

Publication number Publication date
CL2007002316A1 (es) 2008-02-01
EP2050749B1 (en) 2017-11-22
CA2659604A1 (en) 2008-02-14
EP2050749A4 (en) 2011-03-30
SI2050749T1 (en) 2018-04-30
IL196601A (en) 2015-03-31
NO342978B1 (no) 2018-09-17
IL196601A0 (en) 2009-11-18
PT2050749T (pt) 2018-01-02
AU2007282535B9 (en) 2013-06-20
KR20090047462A (ko) 2009-05-12
WO2008018426A1 (en) 2008-02-14
DK2050749T3 (en) 2018-01-08
NZ575274A (en) 2010-11-26
TWI394758B (zh) 2013-05-01
CY1119882T1 (el) 2018-06-27
HUE035116T2 (hu) 2018-05-02
US20100069629A1 (en) 2010-03-18
AR062292A1 (es) 2008-10-29
KR101435692B1 (ko) 2014-09-01
PL2050749T3 (pl) 2018-03-30
AU2007282535A1 (en) 2008-02-14
RU2009108328A (ru) 2010-09-20
MX2009001451A (es) 2009-02-18
RU2448109C2 (ru) 2012-04-20
US8022205B2 (en) 2011-09-20
EP2050749A1 (en) 2009-04-22
TW200817411A (en) 2008-04-16
BRPI0714908A2 (pt) 2013-05-28
LT2050749T (lt) 2018-01-10
CA2659604C (en) 2015-04-28
JPWO2008018426A1 (ja) 2009-12-24
ES2657635T3 (es) 2018-03-06
PE20080527A1 (es) 2008-07-09
JP4450857B2 (ja) 2010-04-14
MY145385A (en) 2012-01-31
BRPI0714908B8 (pt) 2021-05-25
BRPI0714908B1 (pt) 2020-10-13
AU2007282535B2 (en) 2013-05-30

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