NO20083562L - Cannabinoidreseptormodulatorer - Google Patents
CannabinoidreseptormodulatorerInfo
- Publication number
- NO20083562L NO20083562L NO20083562A NO20083562A NO20083562L NO 20083562 L NO20083562 L NO 20083562L NO 20083562 A NO20083562 A NO 20083562A NO 20083562 A NO20083562 A NO 20083562A NO 20083562 L NO20083562 L NO 20083562L
- Authority
- NO
- Norway
- Prior art keywords
- disorders
- cannabinoidreseptormodulatorer
- addictions
- solvate
- obesity
- Prior art date
Links
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 208000024172 Cardiovascular disease Diseases 0.000 abstract 1
- 206010012335 Dependence Diseases 0.000 abstract 1
- 208000018522 Gastrointestinal disease Diseases 0.000 abstract 1
- 208000008589 Obesity Diseases 0.000 abstract 1
- 208000015114 central nervous system disease Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000035475 disorder Diseases 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 208000030159 metabolic disease Diseases 0.000 abstract 1
- 235000020824 obesity Nutrition 0.000 abstract 1
- 230000000241 respiratory effect Effects 0.000 abstract 1
- 208000023504 respiratory system disease Diseases 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
- C07D209/46—Iso-indoles; Hydrogenated iso-indoles with an oxygen atom in position 1
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/4035—Isoindoles, e.g. phthalimide
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- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
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- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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Abstract
Forbindelse som har den generelle struktur med formel (I): eller farmasøytisk akseptabelt salt, solvat eller ester derav, er anvendbar ved behandling av sykdommer, forstyrrelser eller tilstander, slik som overvekt, metabolske forstyrrelser, avhengighet, sykdommer i sentralnervesystemet, hjerte- og karforstyrrelser, åndedrettsforstyrrelser og mage- og tarmforstyrrelser.
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| US20040167185A1 (en) | 2003-01-16 | 2004-08-26 | Geetha Shankar | Methods of treating conditions associated with an Edg-3 receptor |
| US7183445B2 (en) * | 2003-05-31 | 2007-02-27 | Janssen Pharmaceutica N.V | Cyclohexyl derivatives as selective estrogen receptor modulators |
| EP1718293A1 (en) | 2004-02-20 | 2006-11-08 | Aventis Pharmaceuticals Inc. | Oxydecahydronaphthalene modulators of hm74 |
| CN1921845A (zh) | 2004-02-20 | 2007-02-28 | 安万特药物公司 | 作为hm74调节剂的呋塞米衍生物以及它们用于治疗炎症的用途 |
| WO2006060461A1 (en) | 2004-12-03 | 2006-06-08 | Schering Corporation | Substituted piperazines as cb1 antagonists |
| JP4364175B2 (ja) | 2005-08-01 | 2009-11-11 | 株式会社東芝 | 乗算器及びこれを用いる無線通信装置 |
| CA2637057A1 (en) | 2006-01-13 | 2007-07-26 | Schering Corporation | Diaryl piperidines as cb1 modulators |
| AR059021A1 (es) | 2006-01-18 | 2008-03-05 | Schering Corp | Moduladores de receptores cannabinoides |
| CA2692268A1 (en) | 2007-06-28 | 2009-01-08 | Intervet International B.V. | Substituted piperazines as cb1 antagonists |
-
2007
- 2007-01-16 AR ARP070100181A patent/AR059021A1/es unknown
- 2007-01-16 AU AU2007207706A patent/AU2007207706A1/en not_active Abandoned
- 2007-01-16 BR BRPI0706623-6A patent/BRPI0706623A2/pt not_active IP Right Cessation
- 2007-01-16 EP EP07716633A patent/EP1973877A2/en not_active Withdrawn
- 2007-01-16 KR KR1020087020165A patent/KR20080097426A/ko not_active Ceased
- 2007-01-16 RU RU2008133381/04A patent/RU2008133381A/ru not_active Application Discontinuation
- 2007-01-16 US US11/653,558 patent/US7897601B2/en not_active Expired - Fee Related
- 2007-01-16 PE PE2007000047A patent/PE20071320A1/es not_active Application Discontinuation
- 2007-01-16 JP JP2008551309A patent/JP2009528266A/ja active Pending
- 2007-01-16 MX MX2008009354A patent/MX2008009354A/es unknown
- 2007-01-16 CA CA002637565A patent/CA2637565A1/en not_active Abandoned
- 2007-01-16 WO PCT/US2007/001024 patent/WO2007084450A2/en not_active Ceased
- 2007-01-16 NZ NZ569814A patent/NZ569814A/en not_active IP Right Cessation
- 2007-01-17 TW TW096101681A patent/TW200738632A/zh unknown
-
2008
- 2008-08-15 NO NO20083562A patent/NO20083562L/no not_active Application Discontinuation
- 2008-08-16 EC EC2008008628A patent/ECSP088628A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US7897601B2 (en) | 2011-03-01 |
| RU2008133381A (ru) | 2010-02-27 |
| US20070197628A1 (en) | 2007-08-23 |
| TW200738632A (en) | 2007-10-16 |
| KR20080097426A (ko) | 2008-11-05 |
| PE20071320A1 (es) | 2007-12-29 |
| BRPI0706623A2 (pt) | 2011-04-12 |
| MX2008009354A (es) | 2008-09-30 |
| JP2009528266A (ja) | 2009-08-06 |
| AU2007207706A1 (en) | 2007-07-26 |
| CA2637565A1 (en) | 2007-07-26 |
| EP1973877A2 (en) | 2008-10-01 |
| AR059021A1 (es) | 2008-03-05 |
| WO2007084450A2 (en) | 2007-07-26 |
| NZ569814A (en) | 2011-10-28 |
| WO2007084450A3 (en) | 2007-11-08 |
| ECSP088628A (es) | 2008-08-29 |
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