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NO20083561L - Forbindelser for behandling av inflammatoriske forstyrrelser - Google Patents

Forbindelser for behandling av inflammatoriske forstyrrelser

Info

Publication number
NO20083561L
NO20083561L NO20083561A NO20083561A NO20083561L NO 20083561 L NO20083561 L NO 20083561L NO 20083561 A NO20083561 A NO 20083561A NO 20083561 A NO20083561 A NO 20083561A NO 20083561 L NO20083561 L NO 20083561L
Authority
NO
Norway
Prior art keywords
compounds
treatment
inflammatory disorders
pharmaceutically acceptable
aggreganase
Prior art date
Application number
NO20083561A
Other languages
English (en)
Inventor
Bandarpalle B Shankar
Vincent Stewart Madison
Joseph A Kozlowski
Ling Tong
Guowel Zhou
Neng-Yang Shih
Wensheng Yu
Lei Chen
Zhuyan Guo
Michael K C Wong
Seong Heon Kim
Brian J Lavey
Peter Orth
De-Yi Yang
M Arshad Siddiqui
Kristin E Rosner
Chaoyang Dai
Janeta Popovici-Muller
Vinay Girijavallabhan
Dansu Li
Original Assignee
Usmicula Aneta S
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Usmicula Aneta S filed Critical Usmicula Aneta S
Publication of NO20083561L publication Critical patent/NO20083561L/no

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4166—1,3-Diazoles having oxo groups directly attached to the heterocyclic ring, e.g. phenytoin
    • A—HUMAN NECESSITIES
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
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    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
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    • C07D495/04—Ortho-condensed systems
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
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  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Dermatology (AREA)
  • Neurosurgery (AREA)
  • Urology & Nephrology (AREA)
  • Pulmonology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Addiction (AREA)
  • Cardiology (AREA)
  • Endocrinology (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Transplantation (AREA)
  • Psychiatry (AREA)
  • Vascular Medicine (AREA)
  • Gastroenterology & Hepatology (AREA)

Abstract

Denne oppfinnelsen vedrører forbindelser med formel (I). eller et farmasøytisk akseptabelt salt, solvat, en farmasøytisk akseptabel ester eller isomer derav, som kan anvendes til behandlingen av sykdommer eller tilstander formidlet av MMP-er, ADAM-er, TACE, aggrekanase, TNF-a eller kombinasjoner derav.
NO20083561A 2006-01-17 2008-08-15 Forbindelser for behandling av inflammatoriske forstyrrelser NO20083561L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11/333,663 US7504424B2 (en) 2004-07-16 2006-01-17 Compounds for the treatment of inflammatory disorders
PCT/US2007/000930 WO2007084415A2 (en) 2006-01-17 2007-01-16 Compounds for the treatment of inflammatory disorders

Publications (1)

Publication Number Publication Date
NO20083561L true NO20083561L (no) 2008-10-16

Family

ID=38169339

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20083561A NO20083561L (no) 2006-01-17 2008-08-15 Forbindelser for behandling av inflammatoriske forstyrrelser

Country Status (17)

Country Link
US (2) US7504424B2 (no)
EP (1) EP1976849B1 (no)
JP (1) JP2009523795A (no)
KR (1) KR20080093048A (no)
CN (1) CN101410388A (no)
AR (1) AR058901A1 (no)
AU (1) AU2007207671A1 (no)
BR (1) BRPI0707152A2 (no)
CA (1) CA2637385A1 (no)
EC (1) ECSP088627A (no)
IL (1) IL192692A0 (no)
NO (1) NO20083561L (no)
PE (1) PE20070852A1 (no)
RU (1) RU2008133388A (no)
TW (1) TW200736248A (no)
WO (1) WO2007084415A2 (no)
ZA (1) ZA200806074B (no)

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US7488745B2 (en) * 2004-07-16 2009-02-10 Schering Corporation Compounds for the treatment of inflammatory disorders
WO2007021803A1 (en) * 2005-08-12 2007-02-22 Schering Corporation Compounds for the treatment of inflammatory disorders
PE20071240A1 (es) * 2006-01-17 2008-01-14 Schering Corp Compuestos derivados de hidantoina para el tratamiento de trastornos inflamatorios
CA2661605A1 (en) 2006-08-31 2008-03-06 Schering Corporation Hydantoin derivatives useful as antibacterial agents
US8859529B2 (en) 2008-09-24 2014-10-14 Merck Sharp & Dohme Corp. Compounds for the treatment of inflammatory disorders
WO2010036640A2 (en) * 2008-09-24 2010-04-01 Schering Corporation Compounds for the treatment of inflammatory disorders
WO2010054279A1 (en) 2008-11-10 2010-05-14 Schering Corporation Compounds for the treatment of inflammatory disorders
WO2010054278A2 (en) * 2008-11-10 2010-05-14 Schering Corporation Compounds for the treatment of inflammatory disorders
EP2597084B1 (en) 2010-07-08 2016-06-29 Kaken Pharmaceutical Co., Ltd. N-hydroxyformamide derivative and pharmaceutical containing same
ES2703498T3 (es) * 2010-11-13 2019-03-11 Innocrin Pharmaceuticals Inc 1-(6,7-Bis(difluorometoxi)naftalen-2-il)-2-metil-1-(1H-1,2,3-triazol-4-il)propan-1-ol como inhibidor de CYP17 para el tratamiento de enfermedades dependientes de andrógenos como el cáncer de próstata
IN2014KN01075A (no) 2011-11-18 2015-10-09 Heptares Therapeutics Ltd
AU2012349288B2 (en) * 2011-12-09 2016-12-01 Kaken Pharmaceutical Co., Ltd. Pyridone derivative and medicine containing same
AU2012352572B2 (en) * 2011-12-12 2017-08-17 Allergan, Inc. Benzisothiazol-3(1H)-one-5-sulfonyl derivatives as chemokine receptor modulators
DK2925757T3 (en) 2012-11-19 2018-01-15 Novartis Ag Compounds and compositions for the treatment of parasitic diseases
US8871754B2 (en) 2012-11-19 2014-10-28 Irm Llc Compounds and compositions for the treatment of parasitic diseases
WO2014122474A1 (en) 2013-02-07 2014-08-14 Takeda Pharmaceutical Company Limited Piperidin-1 -yl and azepin-1 -yl carboxylates as muscarinic m4 receptor agonists
KR102379801B1 (ko) 2013-06-07 2022-03-28 가껭세이야꾸가부시기가이샤 (＋)-5-(3,4-디플루오로페닐)-5-[(3-메틸-2-옥소피리딘-1(2h)-일)메틸]이미다졸리딘-2,4-디온 및 그것을 함유하는 의약
GB201404922D0 (en) 2014-03-19 2014-04-30 Heptares Therapeutics Ltd Pharmaceutical compounds
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