NO20082365L - Ny metode for fremstilling av 5-amino-3H-tiazolo[4,5-D]pyrimidin-2-on - Google Patents
Ny metode for fremstilling av 5-amino-3H-tiazolo[4,5-D]pyrimidin-2-onInfo
- Publication number
- NO20082365L NO20082365L NO20082365A NO20082365A NO20082365L NO 20082365 L NO20082365 L NO 20082365L NO 20082365 A NO20082365 A NO 20082365A NO 20082365 A NO20082365 A NO 20082365A NO 20082365 L NO20082365 L NO 20082365L
- Authority
- NO
- Norway
- Prior art keywords
- preparation
- thiazolo
- pyrimidin
- amino
- new method
- Prior art date
Links
- CGLJYFPRPQWKTN-UHFFFAOYSA-N 5-amino-3h-[1,3]thiazolo[4,5-d]pyrimidin-2-one Chemical compound NC1=NC=C2SC(=O)NC2=N1 CGLJYFPRPQWKTN-UHFFFAOYSA-N 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- YWBULOYFCXZCGF-UHFFFAOYSA-N [1,3]thiazolo[4,5-d]pyrimidine Chemical compound C1=NC=C2SC=NC2=N1 YWBULOYFCXZCGF-UHFFFAOYSA-N 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 230000002519 immonomodulatory effect Effects 0.000 abstract 1
- 239000002718 pyrimidine nucleoside Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US73805505P | 2005-11-21 | 2005-11-21 | |
| PCT/US2006/061111 WO2007062355A2 (fr) | 2005-11-21 | 2006-11-20 | Nouveau procede de preparation de la 5-amino-3h-thiazolo[4,5-d]pyrimidin-2-one |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO20082365L true NO20082365L (no) | 2008-08-18 |
Family
ID=37908057
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20082365A NO20082365L (no) | 2005-11-21 | 2008-05-26 | Ny metode for fremstilling av 5-amino-3H-tiazolo[4,5-D]pyrimidin-2-on |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US7781581B2 (fr) |
| EP (1) | EP1973920B1 (fr) |
| JP (1) | JP5117391B2 (fr) |
| KR (1) | KR20080090400A (fr) |
| CN (1) | CN101365705A (fr) |
| AR (1) | AR058210A1 (fr) |
| AT (1) | ATE474842T1 (fr) |
| AU (1) | AU2006318260B2 (fr) |
| BR (1) | BRPI0618789A2 (fr) |
| CA (1) | CA2630463C (fr) |
| DE (1) | DE602006015700D1 (fr) |
| EA (1) | EA200801404A1 (fr) |
| ES (1) | ES2345904T3 (fr) |
| IL (1) | IL191568A0 (fr) |
| NO (1) | NO20082365L (fr) |
| SG (1) | SG152296A1 (fr) |
| TW (1) | TWI383987B (fr) |
| WO (1) | WO2007062355A2 (fr) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2007150002A2 (fr) | 2006-06-22 | 2007-12-27 | Anadys Pharmaceuticals, Inc. | PROMÉDICAMENTS DE LA 5-AMINO-3-(3'-DÉSOXY-ß-D-RIBOFURANNOSYL)-THIAZOLO[4,5-D]PYRIMIDIN-2,7-DIONE |
| JPWO2012102366A1 (ja) * | 2011-01-28 | 2014-06-30 | 日本たばこ産業株式会社 | 新規ピペラジン化合物の製造方法 |
| CN103012284A (zh) * | 2012-12-26 | 2013-04-03 | 无锡捷化医药科技有限公司 | 一种2-氨基-5-溴嘧啶类化合物的制备方法 |
| ES2864223T3 (es) | 2014-12-08 | 2021-10-13 | Hoffmann La Roche | Compuestos de 5-amino-6H-tiazolo[4,5-d]pirimidin-2,7-diona 3-sustituida para el tratamiento y profilaxis de infección vírica |
| EP3568400B1 (fr) | 2017-01-06 | 2025-11-19 | F. Hoffmann-La Roche AG | Procédé de préparation de composés 5-amino-6h-thiazolo[4,5-d]pyrimidine-2,7-dione à substitution en position 3 |
| CN111635368B (zh) * | 2020-06-12 | 2021-06-29 | 东莞市东阳光仿制药研发有限公司 | 一种胺化合物的制备方法 |
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| US4539205A (en) | 1982-11-09 | 1985-09-03 | Scripps Clinic And Research Foundation | Modulation of animal cellular responses with compositions containing 8-substituted guanine derivatives |
| US4643992A (en) | 1982-11-09 | 1987-02-17 | Scripps Clinic And Research Foundation | Modulation of animal cellular responses with compositions containing 8-substituted guanine derivatives |
| US4746651A (en) | 1983-11-01 | 1988-05-24 | Scripps Clinic And Research Foundation | Antimicrobial chemotherapeutic potentiation using substituted nucleoside derivatives |
| US5166141A (en) | 1983-11-01 | 1992-11-24 | Scripps Clinic And Research Foundation | Immunostimulating 7-deaza-7-oxa- and 7-deaza-7-oxo-analogs of 8-substituted-guanine-9-(1'-beta-D-aldoglycosidyl) derivatives and methods of treating test animals |
| US5011828A (en) | 1985-11-15 | 1991-04-30 | Michael Goodman | Immunostimulating guanine derivatives, compositions and methods |
| GB8712745D0 (en) | 1987-05-30 | 1987-07-01 | Wellcome Found | Antiviral compounds |
| US5041426A (en) * | 1987-12-21 | 1991-08-20 | Brigham Young University | Immune system enhancing 3-β-d-ribofuranosylthiazolo[4,5-d]pyridimine nucleosides and nucleotides |
| US4880784A (en) | 1987-12-21 | 1989-11-14 | Brigham Young University | Antiviral methods utilizing ribofuranosylthiazolo[4,5-d]pyrimdine derivatives |
| US5041542A (en) | 1988-06-03 | 1991-08-20 | Nucleic Acid Research Institute | Substituted pyrimido[5,4-d]pyrimidine nucleosides |
| GB9015914D0 (en) | 1990-07-19 | 1990-09-05 | Wellcome Found | Heterocyclic compounds |
| US5248672A (en) | 1990-11-01 | 1993-09-28 | The Regents Of The University Of Michigan | Polysubstituted benzimidazole nucleosides as antiviral agents |
| GB9105899D0 (en) | 1991-03-20 | 1991-05-08 | Wellcome Found | Therapeutic nucleosides |
| AU5165793A (en) | 1992-10-01 | 1994-04-26 | Mcneilab, Inc. | Derivatives of 7,8-disubstituted guanosines |
| GB9301000D0 (en) | 1993-01-20 | 1993-03-10 | Glaxo Group Ltd | Chemical compounds |
| US5395937A (en) | 1993-01-29 | 1995-03-07 | Minnesota Mining And Manufacturing Company | Process for preparing quinoline amines |
| US5446045A (en) | 1993-12-20 | 1995-08-29 | Revankar; Ganapathi R. | Antiviral guanine analogs |
| US5994321A (en) | 1993-12-20 | 1999-11-30 | Aronex Pharmaceuticals, Inc. | Antiviral guanine analogs |
| US5496816A (en) | 1994-03-14 | 1996-03-05 | Merck & Co., Inc. | Carbapenem antibacterial compounds, compositions containing such compounds and methods of treatment |
| ATE283855T1 (de) | 1996-07-03 | 2004-12-15 | Sumitomo Pharma | Neue purinderivate |
| CZ126799A3 (cs) | 1996-10-16 | 1999-07-14 | Icn Pharmaceuticals | Purinové L-nukleosidy a jejich analogy a farmaceutické prostředky, které je obsahují |
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| JP4391592B2 (ja) | 1996-10-25 | 2009-12-24 | スリーエム カンパニー | Th2介在性および関連疾患治療のための免疫応答修飾化合物 |
| KR100613634B1 (ko) | 1997-11-28 | 2006-08-18 | 다이닛본 스미토모 세이야꾸 가부시끼가이샤 | 신규한 복소환 화합물 |
| TW572758B (en) | 1997-12-22 | 2004-01-21 | Sumitomo Pharma | Type 2 helper T cell-selective immune response inhibitors comprising purine derivatives |
| EP1068212A1 (fr) * | 1998-04-03 | 2001-01-17 | Bristol-Myers Squibb Pharma Company | PYRIMIDINES ET PYRIDINES THIAZOLO 4,5-d] UTILISEES COMME ANTAGONISTES DU FACTEUR LIBERATEUR DE CORTICOTROPHINE (CRF) |
| US6444652B1 (en) | 1998-08-10 | 2002-09-03 | Novirio Pharmaceuticals Limited | β-L-2'-deoxy-nucleosides for the treatment of hepatitis B |
| US6664264B2 (en) | 2000-12-08 | 2003-12-16 | 3M Innovative Properties Company | Thioether substituted imidazoquinolines |
| US6545017B1 (en) | 2000-12-08 | 2003-04-08 | 3M Innovative Properties Company | Urea substituted imidazopyridines |
| US6667312B2 (en) | 2000-12-08 | 2003-12-23 | 3M Innovative Properties Company | Thioether substituted imidazoquinolines |
| US6664260B2 (en) | 2000-12-08 | 2003-12-16 | 3M Innovative Properties Company | Heterocyclic ether substituted imidazoquinolines |
| US6545016B1 (en) | 2000-12-08 | 2003-04-08 | 3M Innovative Properties Company | Amide substituted imidazopyridines |
| US20020086871A1 (en) | 2000-12-29 | 2002-07-04 | O'neill Brian Thomas | Pharmaceutical composition for the treatment of CNS and other disorders |
| KR100892614B1 (ko) | 2001-04-17 | 2009-04-09 | 다이닛본 스미토모 세이야꾸 가부시끼가이샤 | 신규 아데닌 유도체 |
| HRP20040541A2 (en) | 2001-11-27 | 2004-10-31 | Anadys Pharmaceuticals | 3- -D-RIBOFURANOSYLTHIAZOLO[4,5-d]PYRIMIDINE NUCLEOSIDES AND USES THEREOF |
| US7321033B2 (en) | 2001-11-27 | 2008-01-22 | Anadys Pharmaceuticals, Inc. | 3-B-D-ribofuranosylthiazolo [4,5-d] pyrimidine nucleosides and uses thereof |
| EP1501850A2 (fr) | 2002-05-06 | 2005-02-02 | Genelabs Technologies, Inc. | Derives nucleosidiques destines au traitement de l'infection par le virus de l'hepatite c |
| US7196090B2 (en) * | 2002-07-25 | 2007-03-27 | Warner-Lambert Company | Kinase inhibitors |
| WO2005016235A2 (fr) | 2003-04-14 | 2005-02-24 | The Regents Of The University Of California | Utilisation combinee d'inhibiteurs de l'inosine monophosphate deshydrogenase (impdh) et d'agonistes du toll-like recepteur |
| KR20060027338A (ko) * | 2003-06-12 | 2006-03-27 | 아스텔라스세이야쿠 가부시키가이샤 | 벤즈 아미드 유도체 또는 그 염 |
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| EP1722789A2 (fr) * | 2004-03-08 | 2006-11-22 | Amgen Inc. | Modulation therapeutique de l'activite de recepteur de ppar-gamma |
| CN101087769A (zh) | 2004-10-15 | 2007-12-12 | 拜尔药品公司 | 用于治疗肥胖的联苯-4-基-羰基氨基酸衍生物的制备及用途 |
| WO2006066080A1 (fr) * | 2004-12-17 | 2006-06-22 | Anadys Pharmaceuticals, Inc. | Composes de 3h-oxazolo et 3h-thiazolo [4,5-d]pyrimidine-2-one disubstitues en 3, 5 et trisubstitues en 3, 5, 7 et promedicaments associes |
| JP2008540549A (ja) | 2005-05-09 | 2008-11-20 | ハイドラ バイオサイエンシズ インコーポレイテッド | Trpv3機能調節用化合物 |
| WO2007150002A2 (fr) | 2006-06-22 | 2007-12-27 | Anadys Pharmaceuticals, Inc. | PROMÉDICAMENTS DE LA 5-AMINO-3-(3'-DÉSOXY-ß-D-RIBOFURANNOSYL)-THIAZOLO[4,5-D]PYRIMIDIN-2,7-DIONE |
| US7528115B2 (en) | 2006-07-18 | 2009-05-05 | Anadys Pharmaceuticals, Inc. | Carbonate and carbamate prodrugs of thiazolo[4,5-d]pyrimidines |
-
2006
- 2006-11-20 AT AT06846356T patent/ATE474842T1/de not_active IP Right Cessation
- 2006-11-20 BR BRPI0618789A patent/BRPI0618789A2/pt not_active IP Right Cessation
- 2006-11-20 CN CNA200680050892XA patent/CN101365705A/zh active Pending
- 2006-11-20 JP JP2008541505A patent/JP5117391B2/ja not_active Expired - Fee Related
- 2006-11-20 EA EA200801404A patent/EA200801404A1/xx unknown
- 2006-11-20 CA CA2630463A patent/CA2630463C/fr not_active Expired - Fee Related
- 2006-11-20 WO PCT/US2006/061111 patent/WO2007062355A2/fr not_active Ceased
- 2006-11-20 SG SG200903039-6A patent/SG152296A1/en unknown
- 2006-11-20 KR KR1020087014973A patent/KR20080090400A/ko not_active Withdrawn
- 2006-11-20 ES ES06846356T patent/ES2345904T3/es active Active
- 2006-11-20 DE DE602006015700T patent/DE602006015700D1/de active Active
- 2006-11-20 TW TW095142739A patent/TWI383987B/zh not_active IP Right Cessation
- 2006-11-20 EP EP06846356A patent/EP1973920B1/fr not_active Not-in-force
- 2006-11-20 US US11/601,719 patent/US7781581B2/en not_active Expired - Fee Related
- 2006-11-20 AU AU2006318260A patent/AU2006318260B2/en not_active Ceased
- 2006-11-21 AR ARP060105089A patent/AR058210A1/es not_active Application Discontinuation
-
2008
- 2008-05-20 IL IL191568A patent/IL191568A0/en unknown
- 2008-05-26 NO NO20082365A patent/NO20082365L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| CN101365705A (zh) | 2009-02-11 |
| ATE474842T1 (de) | 2010-08-15 |
| KR20080090400A (ko) | 2008-10-08 |
| TWI383987B (zh) | 2013-02-01 |
| BRPI0618789A2 (pt) | 2016-08-30 |
| CA2630463C (fr) | 2015-01-06 |
| TW200736265A (en) | 2007-10-01 |
| DE602006015700D1 (de) | 2010-09-02 |
| CA2630463A1 (fr) | 2007-05-31 |
| EP1973920B1 (fr) | 2010-07-21 |
| ES2345904T3 (es) | 2010-10-05 |
| AU2006318260B2 (en) | 2012-05-17 |
| WO2007062355A2 (fr) | 2007-05-31 |
| AU2006318260A1 (en) | 2007-05-31 |
| AR058210A1 (es) | 2008-01-23 |
| US7781581B2 (en) | 2010-08-24 |
| WO2007062355A3 (fr) | 2007-07-26 |
| JP2009516709A (ja) | 2009-04-23 |
| IL191568A0 (en) | 2008-12-29 |
| EA200801404A1 (ru) | 2008-10-30 |
| JP5117391B2 (ja) | 2013-01-16 |
| US20070117979A1 (en) | 2007-05-24 |
| SG152296A1 (en) | 2009-05-29 |
| EP1973920A2 (fr) | 2008-10-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |