NO20082768L - Levodopa prodroge mesylat, sammensetninger og anvendelser derav - Google Patents

Levodopa prodroge mesylat, sammensetninger og anvendelser derav

Info

Publication number: NO20082768L
Authority: NO; Norway
Prior art keywords: compositions; levodopa prodrug; prodrug mesylate; mesylate; methods
Prior art date: 2005-12-05

Application number

NO20082768A

Other languages

English (en)

Norwegian (no)

Inventor

Jia-Ning Xiang

Cindy X Zhou

Mark Nguyen

Xuedong Dai

Jianhua Li

Original Assignee

Xenoport Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2005-12-05

Filing date

2008-06-16

Publication date

2008-06-24

2008-06-16 Application filed by Xenoport Inc filed Critical Xenoport Inc

2008-06-24 Publication of NO20082768L publication Critical patent/NO20082768L/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/34—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
- C07C229/36—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings with at least one amino group and one carboxyl group bound to the same carbon atom of the carbon skeleton
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4458—Non condensed piperidines, e.g. piperocaine only substituted in position 2, e.g. methylphenidate
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/10—Laxatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P25/24—Antidepressants
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/34—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
- C07C309/01—Sulfonic acids
- C07C309/02—Sulfonic acids having sulfo groups bound to acyclic carbon atoms
- C07C309/03—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
- C07C309/04—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton containing only one sulfo group
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Cardiology (AREA)
Psychiatry (AREA)
Heart & Thoracic Surgery (AREA)
Psychology (AREA)
Hospice & Palliative Care (AREA)
Anesthesiology (AREA)
Orthopedic Medicine & Surgery (AREA)
Hematology (AREA)
Obesity (AREA)
Addiction (AREA)
Nutrition Science (AREA)
Pain & Pain Management (AREA)
Dermatology (AREA)
Urology & Nephrology (AREA)
Diabetes (AREA)
Physical Education & Sports Medicine (AREA)
Gynecology & Obstetrics (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Otolaryngology (AREA)
Pulmonology (AREA)
Epidemiology (AREA)

NO20082768A 2005-12-05 2008-06-16 Levodopa prodroge mesylat, sammensetninger og anvendelser derav NO20082768L (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US74187605P	2005-12-05	2005-12-05
PCT/US2006/046273 WO2007067495A2 (en)	2005-12-05	2006-12-04	Levodopa prodrug mesylate, compositions thereof, and uses thereof

Publications (1)

Publication Number	Publication Date
NO20082768L true NO20082768L (no)	2008-06-24

Family

ID=38123406

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20082768A NO20082768L (no)	2005-12-05	2008-06-16	Levodopa prodroge mesylat, sammensetninger og anvendelser derav

Country Status (20)

Country	Link
US (5)	US7563821B2 (ru)
EP (1)	EP1959948B1 (ru)
JP (1)	JP5153641B2 (ru)
KR (1)	KR101396639B1 (ru)
CN (1)	CN101365439B (ru)
AU (1)	AU2006322051B2 (ru)
BR (1)	BRPI0619425A2 (ru)
CA (1)	CA2631643C (ru)
CY (1)	CY1113108T1 (ru)
DK (1)	DK1959948T3 (ru)
ES (1)	ES2391575T3 (ru)
IL (1)	IL191937A (ru)
NO (1)	NO20082768L (ru)
NZ (1)	NZ569485A (ru)
PL (1)	PL1959948T3 (ru)
PT (1)	PT1959948E (ru)
RU (1)	RU2429223C2 (ru)
TW (1)	TWI403493B (ru)
WO (1)	WO2007067495A2 (ru)
ZA (1)	ZA200805511B (ru)

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Also Published As

Publication number	Publication date
RU2008127312A (ru)	2010-01-20
US7563821B2 (en)	2009-07-21
RU2429223C2 (ru)	2011-09-20
HK1121381A1 (en)	2009-04-24
US20120296109A1 (en)	2012-11-22
IL191937A (en)	2014-07-31
US7893105B2 (en)	2011-02-22
WO2007067495A3 (en)	2007-09-27
JP2009520690A (ja)	2009-05-28
ZA200805511B (en)	2010-02-24
ES2391575T3 (es)	2012-11-27
JP5153641B2 (ja)	2013-02-27
US20110111062A1 (en)	2011-05-12
EP1959948B1 (en)	2012-07-18
DK1959948T3 (da)	2012-08-20
CN101365439A (zh)	2009-02-11
US8193242B2 (en)	2012-06-05
TWI403493B (zh)	2013-08-01
EP1959948A2 (en)	2008-08-27
BRPI0619425A2 (pt)	2011-10-04
CY1113108T1 (el)	2016-04-13
AU2006322051B2 (en)	2011-09-29
US20090326067A1 (en)	2009-12-31
AU2006322051A1 (en)	2007-06-14
PL1959948T3 (pl)	2012-12-31
KR20080073365A (ko)	2008-08-08
IL191937A0 (en)	2009-08-03
KR101396639B1 (ko)	2014-05-21
US20090156679A1 (en)	2009-06-18
CA2631643C (en)	2015-07-07
PT1959948E (pt)	2012-09-12
WO2007067495A2 (en)	2007-06-14
CA2631643A1 (en)	2007-06-14
NZ569485A (en)	2011-06-30
US20070225366A1 (en)	2007-09-27
CN101365439B (zh)	2012-12-26
US7968597B2 (en)	2011-06-28
TW200804239A (en)	2008-01-16

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