NO20034003D0 - Fremgangsmåte for fremstilling av imidazol-forbindelser - Google Patents

Fremgangsmåte for fremstilling av imidazol-forbindelser

Info

Publication number: NO20034003D0
Authority: NO; Norway
Prior art keywords: preparation; imidazole compounds; imidazole; compounds
Prior art date: 2001-03-12

Application number

NO20034003A

Other languages

English (en)

Other versions

NO324954B1 (no

NO20034003L (no

Inventor

Walter Ferdinand Mari Filliers

Rudy Laurent Maria Broeckx

Stefan Marcel Herman Leurs

Original Assignee

Janssen Pharmaceutica Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-03-12

Filing date

2003-09-10

Publication date

2003-09-10

2003-09-10 Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv

2003-09-10 Publication of NO20034003D0 publication Critical patent/NO20034003D0/no

2003-10-22 Publication of NO20034003L publication Critical patent/NO20034003L/no

2008-01-14 Publication of NO324954B1 publication Critical patent/NO324954B1/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Epoxy Resins (AREA)

NO20034003A 2001-03-12 2003-09-10 Fremgangsmate for fremstilling av 4-(3-klorfenyl)-6-[(4-klorfenyl)hydroksy(1-metyl-1H-imidazol-5-yl)metyl]-1-metyl-2(1H)-kinolinon og dets farmasoytisk akseptable salter. NO324954B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP01200928		2001-03-12
PCT/EP2002/002459 WO2002072574A1 (en)	2001-03-12	2002-03-05	Process for the preparation of imidazole compounds

Publications (3)

Publication Number	Publication Date
NO20034003D0 true NO20034003D0 (no)	2003-09-10
NO20034003L NO20034003L (no)	2003-10-22
NO324954B1 NO324954B1 (no)	2008-01-14

Family

ID=8180004

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20034003A NO324954B1 (no)	2001-03-12	2003-09-10	Fremgangsmate for fremstilling av 4-(3-klorfenyl)-6-[(4-klorfenyl)hydroksy(1-metyl-1H-imidazol-5-yl)metyl]-1-metyl-2(1H)-kinolinon og dets farmasoytisk akseptable salter.

Country Status (31)

Country	Link
US (1)	US6844439B2 (no)
EP (1)	EP1373255B1 (no)
JP (1)	JP4257698B2 (no)
KR (1)	KR100849042B1 (no)
CN (1)	CN1246318C (no)
AR (1)	AR035944A1 (no)
AT (1)	ATE287882T1 (no)
AU (1)	AU2002253101B2 (no)
BR (1)	BRPI0208075B8 (no)
CA (1)	CA2438421C (no)
CZ (1)	CZ300622B6 (no)
DE (1)	DE60202755T2 (no)
DK (1)	DK1373255T3 (no)
EA (1)	EA006770B1 (no)
EE (1)	EE05247B1 (no)
ES (1)	ES2236505T3 (no)
HR (1)	HRP20030695B1 (no)
HU (1)	HU230282B1 (no)
IL (2)	IL157839A0 (no)
MX (1)	MXPA03008205A (no)
MY (1)	MY124838A (no)
NO (1)	NO324954B1 (no)
NZ (1)	NZ528620A (no)
PL (1)	PL208238B1 (no)
PT (1)	PT1373255E (no)
SI (1)	SI1373255T1 (no)
SK (1)	SK287807B6 (no)
TW (1)	TWI249532B (no)
UA (1)	UA74871C2 (no)
WO (1)	WO2002072574A1 (no)
ZA (1)	ZA200307117B (no)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA2441177A1 (en)	2001-03-12	2002-09-19	Avanir Pharmaceuticals	Benzimidazole compounds for modulating ige and inhibiting cellular proliferation
WO2004024655A2 (en)	2002-09-12	2004-03-25	Avanir Pharmaceuticals	Phenyl-indole compounds for modulating ige and inhibiting cellular proliferation
TWI276631B (en)	2002-09-12	2007-03-21	Avanir Pharmaceuticals	Phenyl-aza-benzimidazole compounds for modulating IgE and inhibiting cellular proliferation
JP2007538004A (ja) *	2004-03-18	2007-12-27	ザブライハムアンドウイメンズホスピタル，インコーポレイテッド	シヌクレイノパチーを治療する方法
DE602005007604D1 (de)	2004-05-03	2008-07-31	Janssen Pharmaceutica Nv	Diastereoselektive addition von lithiiertem n-methylimidazol an sulfinimine
WO2005105784A1 (en) *	2004-05-03	2005-11-10	Janssen Pharmaceutica N.V.	Diastereoselective synthesis process for the preparation of imidazole compounds
US7572916B2 (en)	2004-05-03	2009-08-11	Janssen Pharmaceutica Nv	Diastereoselective synthesis process with 6-bromo-4-(3-chlorophenyl)-2-methoxy-quinoline
US20070213366A1 (en)	2005-12-23	2007-09-13	Justman Craig J	Treatment of Synucleinopathies
WO2009151683A2 (en) *	2008-03-12	2009-12-17	Link Medicine Corporation	Quinolinone farnesyl transferase inhibitors for the treatment of synucleinopathies and other indications
KR101044430B1 (ko) *	2009-09-25	2011-06-27	듀오백코리아 주식회사	요추받이를 포함하는 의자의 등 지지 장치
KR101107900B1 (ko) *	2009-10-21	2012-01-25	성용기업 주식회사	의자용 허리지지장치
HUE049620T2 (hu)	2015-08-17	2020-09-28	Kura Oncology Inc	Módszerek rákos páciensek kezelésére farneziltranszferáz inhibitorokkal
PT3534885T (pt)	2016-11-03	2021-04-13	Kura Oncology Inc	Inibidores de farnesiltransferase para usar em métodos de tratamento do cancro
WO2018103027A1 (zh)	2016-12-08	2018-06-14	杭州领业医药科技有限公司	替吡法尼的晶型及其制备方法及药物组合物
SG11202011378WA (en) *	2018-05-18	2020-12-30	Kura Oncology Inc	Synthesis of tipifarnib

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
TW349948B (en)	1995-10-31	1999-01-11	Janssen Pharmaceutica Nv	Farnesyl transferase inhibiting 2-quinolone derivatives
ATE321757T1 (de) *	1995-12-08	2006-04-15	Janssen Pharmaceutica Nv	(imidazol-5-yl)methyl-2-chinolinonderivate als farnesyl protein transferase inhibitoren
TW591030B (en)	1997-03-10	2004-06-11	Janssen Pharmaceutica Nv	Farnesyl transferase inhibiting 1,8-annelated quinolinone derivatives substituted with N- or C-linked imidazoles
KR100520401B1 (ko)	1997-04-25	2005-10-12	얀센 파마슈티카 엔.브이.	파네실 트랜스퍼라제 억제작용을 갖는 퀴나졸리논
EP1107962B1 (en)	1998-08-27	2005-02-23	Pfizer Products Inc.	Quinolin-2-one derivatives useful as anticancer agents
JP3495706B2 (ja) *	1998-08-27	2004-02-09	ファイザー・プロダクツ・インク	抗癌薬として有用なアルキニル置換キノリン−２−オン誘導体

2002
- 2002-03-05 BR BRPI0208075-3 patent/BRPI0208075B8/pt not_active IP Right Cessation
- 2002-03-05 IL IL15783902A patent/IL157839A0/xx unknown
- 2002-03-05 DE DE60202755T patent/DE60202755T2/de not_active Expired - Lifetime
- 2002-03-05 PT PT02722184T patent/PT1373255E/pt unknown
- 2002-03-05 SI SI200230100T patent/SI1373255T1/xx unknown
- 2002-03-05 SK SK1246-2003A patent/SK287807B6/sk unknown
- 2002-03-05 ES ES02722184T patent/ES2236505T3/es not_active Expired - Lifetime
- 2002-03-05 AT AT02722184T patent/ATE287882T1/de active
- 2002-03-05 PL PL363263A patent/PL208238B1/pl unknown
- 2002-03-05 CA CA2438421A patent/CA2438421C/en not_active Expired - Lifetime
- 2002-03-05 JP JP2002571490A patent/JP4257698B2/ja not_active Expired - Lifetime
- 2002-03-05 CZ CZ20032704A patent/CZ300622B6/cs not_active IP Right Cessation
- 2002-03-05 HU HU0303443A patent/HU230282B1/hu unknown
- 2002-03-05 DK DK02722184T patent/DK1373255T3/da active
- 2002-03-05 AU AU2002253101A patent/AU2002253101B2/en not_active Expired
- 2002-03-05 EE EEP200300442A patent/EE05247B1/xx unknown
- 2002-03-05 KR KR1020037010091A patent/KR100849042B1/ko not_active Expired - Lifetime
- 2002-03-05 EP EP02722184A patent/EP1373255B1/en not_active Expired - Lifetime
- 2002-03-05 MX MXPA03008205A patent/MXPA03008205A/es active IP Right Grant
- 2002-03-05 HR HR20030695A patent/HRP20030695B1/xx not_active IP Right Cessation
- 2002-03-05 EA EA200300998A patent/EA006770B1/ru not_active IP Right Cessation
- 2002-03-05 WO PCT/EP2002/002459 patent/WO2002072574A1/en not_active Ceased
- 2002-03-05 US US10/471,215 patent/US6844439B2/en not_active Expired - Lifetime
- 2002-03-05 NZ NZ528620A patent/NZ528620A/en not_active IP Right Cessation
- 2002-03-05 CN CNB02806335XA patent/CN1246318C/zh not_active Expired - Lifetime
- 2002-03-11 MY MYPI20020866A patent/MY124838A/en unknown
- 2002-03-11 TW TW091104444A patent/TWI249532B/zh not_active IP Right Cessation
- 2002-03-11 AR ARP020100873A patent/AR035944A1/es active IP Right Grant
- 2002-05-03 UA UA2003087776A patent/UA74871C2/uk unknown
2003
- 2003-09-10 IL IL157839A patent/IL157839A/en unknown
- 2003-09-10 NO NO20034003A patent/NO324954B1/no not_active IP Right Cessation
- 2003-09-11 ZA ZA200307117A patent/ZA200307117B/en unknown

Also Published As

Publication number	Publication date
CA2438421A1 (en)	2002-09-19
CA2438421C (en)	2010-05-18
AR035944A1 (es)	2004-07-28
KR20030079971A (ko)	2003-10-10
NO324954B1 (no)	2008-01-14
SI1373255T1 (no)	2005-08-31
PL208238B1 (pl)	2011-04-29
BR0208075A (pt)	2004-03-02
MXPA03008205A (es)	2004-01-29
WO2002072574A1 (en)	2002-09-19
US20040138256A1 (en)	2004-07-15
EA200300998A1 (ru)	2004-02-26
PT1373255E (pt)	2005-05-31
SK287807B6 (sk)	2011-10-04
AU2002253101B2 (en)	2007-08-09
US6844439B2 (en)	2005-01-18
IL157839A0 (en)	2004-03-28
ES2236505T3 (es)	2005-07-16
BRPI0208075B1 (pt)	2018-02-14
EE05247B1 (et)	2009-12-15
CZ300622B6 (cs)	2009-07-01
UA74871C2 (en)	2006-02-15
ATE287882T1 (de)	2005-02-15
EP1373255B1 (en)	2005-01-26
MY124838A (en)	2006-07-31
IL157839A (en)	2008-07-08
PL363263A1 (en)	2004-11-15
HRP20030695B1 (hr)	2011-07-31
BRPI0208075B8 (pt)	2021-05-25
JP4257698B2 (ja)	2009-04-22
KR100849042B1 (ko)	2008-07-29
CZ20032704A3 (en)	2004-03-17
CN1246318C (zh)	2006-03-22
HUP0303443A3 (en)	2012-09-28
EA006770B1 (ru)	2006-04-28
JP2004523575A (ja)	2004-08-05
CN1496363A (zh)	2004-05-12
NO20034003L (no)	2003-10-22
EE200300442A (et)	2003-12-15
DK1373255T3 (da)	2005-05-23
HRP20030695A2 (en)	2005-02-28
HK1063315A1 (zh)	2004-12-24
SK12462003A3 (sk)	2004-06-08
HUP0303443A2 (hu)	2004-01-28
NZ528620A (en)	2005-01-28
EP1373255A1 (en)	2004-01-02
ZA200307117B (en)	2004-09-13
TWI249532B (en)	2006-02-21
HU230282B1 (hu)	2015-12-28
DE60202755D1 (de)	2005-03-03
DE60202755T2 (de)	2006-03-30

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Legal Events

Date	Code	Title	Description
2022-04-11	MK1K	Patent expired