NO20026167L - Condensed cyclic compounds as modulators of nuclear hormone receptor function - Google Patents
Condensed cyclic compounds as modulators of nuclear hormone receptor functionInfo
- Publication number
- NO20026167L NO20026167L NO20026167A NO20026167A NO20026167L NO 20026167 L NO20026167 L NO 20026167L NO 20026167 A NO20026167 A NO 20026167A NO 20026167 A NO20026167 A NO 20026167A NO 20026167 L NO20026167 L NO 20026167L
- Authority
- NO
- Norway
- Prior art keywords
- modulators
- hormone receptor
- cyclic compounds
- receptor function
- nuclear hormone
- Prior art date
Links
- 102000007399 Nuclear hormone receptor Human genes 0.000 title 1
- 108020005497 Nuclear hormone receptor Proteins 0.000 title 1
- 150000001923 cyclic compounds Chemical class 0.000 title 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/08—Bridged systems
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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- A61K31/655—Azo (—N=N—), diazo (=N2), azoxy (>N—O—N< or N(=O)—N<), azido (—N3) or diazoamino (—N=N—N<) compounds
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/12—Oxygen or sulfur atoms
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Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US21439200P | 2000-06-28 | 2000-06-28 | |
| US28461701P | 2001-04-18 | 2001-04-18 | |
| US28443801P | 2001-04-18 | 2001-04-18 | |
| PCT/US2001/019663 WO2002000653A2 (en) | 2000-06-28 | 2001-06-20 | Fused cyclic compounds as modulators of nuclear hormone receptor function |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO20026167D0 NO20026167D0 (en) | 2002-12-20 |
| NO20026167L true NO20026167L (en) | 2002-12-20 |
Family
ID=27485945
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20026167A NO20026167L (en) | 2000-06-28 | 2002-12-20 | Condensed cyclic compounds as modulators of nuclear hormone receptor function |
Country Status (10)
| Country | Link |
|---|---|
| EP (1) | EP1299385A2 (en) |
| JP (1) | JP2004515462A (en) |
| AU (1) | AU2002215609A1 (en) |
| BR (1) | BR0111869A (en) |
| CA (1) | CA2413683A1 (en) |
| HU (1) | HUP0303165A3 (en) |
| MX (1) | MXPA02012563A (en) |
| NO (1) | NO20026167L (en) |
| NZ (1) | NZ523802A (en) |
| WO (1) | WO2002000653A2 (en) |
Families Citing this family (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2000264876A (en) * | 1998-09-10 | 2000-09-26 | Sumitomo Chem Co Ltd | Fused heterocyclic compound |
| US20040077605A1 (en) | 2001-06-20 | 2004-04-22 | Salvati Mark E. | Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function |
| JP2004509072A (en) | 2000-06-28 | 2004-03-25 | ブリストル−マイヤーズ スクイブ カンパニー | Selective androgen receptor modulators and methods for their identification, design and use |
| US7001911B2 (en) | 2000-06-28 | 2006-02-21 | Bristol-Myers Squibb Company | Fused cyclic modulators of nuclear hormone receptor function |
| US20030114420A1 (en) * | 2000-06-28 | 2003-06-19 | Salvati Mark E. | Fused cyclic modulators of nuclear hormone receptor function |
| EP1317456A2 (en) * | 2000-09-07 | 2003-06-11 | Bayer Corporation | Cyclic and acyclic amidines and pharmaceutical compositions containing them for use as progesterone receptor binding agents |
| US6953679B2 (en) | 2000-09-19 | 2005-10-11 | Bristol-Myers Squibb Company | Method for the preparation of fused heterocyclic succinimide compounds and analogs thereof |
| EP1467979B1 (en) * | 2001-12-19 | 2008-08-13 | Bristol-Myers Squibb Company | Fused heterocyclic compounds and analogs thereof modulators of nuclear hormone receptor function |
| DE10162375A1 (en) * | 2001-12-19 | 2003-07-10 | Bayer Ag | Bicyclic N-aryl amides |
| JP2005523302A (en) * | 2002-03-18 | 2005-08-04 | ファルマシア・コーポレーション | Combination of aldosterone receptor antagonist and fibric acid derivative |
| US7405234B2 (en) | 2002-05-17 | 2008-07-29 | Bristol-Myers Squibb Company | Bicyclic modulators of androgen receptor function |
| US7649001B2 (en) | 2002-08-12 | 2010-01-19 | Takeda Pharmaceutical Company Limited | Fused benzene derivative and use |
| EP1567487A4 (en) | 2002-11-15 | 2005-11-16 | Bristol Myers Squibb Co | Open chain prolyl urea-related modulators of androgen receptor function |
| US7199125B2 (en) | 2003-10-02 | 2007-04-03 | Bristol-Myers Squibb Company | Spiro-cyclic compounds useful as anti-inflammatory agents |
| US7820702B2 (en) | 2004-02-04 | 2010-10-26 | Bristol-Myers Squibb Company | Sulfonylpyrrolidine modulators of androgen receptor function and method |
| US7417040B2 (en) | 2004-03-01 | 2008-08-26 | Bristol-Myers Squibb Company | Fused tricyclic compounds as inhibitors of 17β-hydroxysteroid dehydrogenase 3 |
| US7696241B2 (en) | 2004-03-04 | 2010-04-13 | Bristol-Myers Squibb Company | Bicyclic compounds as modulators of androgen receptor function and method |
| US7625923B2 (en) * | 2004-03-04 | 2009-12-01 | Bristol-Myers Squibb Company | Bicyclic modulators of androgen receptor function |
| US9409856B2 (en) | 2005-11-28 | 2016-08-09 | Gtx, Inc. | Estrogen receptor ligands and methods of use thereof |
| US8546451B2 (en) | 2005-11-28 | 2013-10-01 | Gtx, Inc. | Estrogen receptor ligands and methods of use thereof |
| CA2642205C (en) * | 2006-02-10 | 2015-01-27 | Janssen Pharmaceutica N.V. | Bicyclic imidazole or thiadiazole heterocycles useful as selective androgen receptor modulators |
| JPWO2008007664A1 (en) | 2006-07-11 | 2009-12-10 | 武田薬品工業株式会社 | Bicyclic heterocyclic compounds and uses thereof |
| JP5816087B2 (en) | 2008-08-29 | 2015-11-18 | エンメエッセディ・イタリア・エッセ・エッレ・エッレ | Saturated bicyclic heterocyclic derivatives as SMO antagonists |
| US9427418B2 (en) | 2009-02-23 | 2016-08-30 | Gtx, Inc. | Estrogen receptor ligands and methods of use thereof |
| US9624161B2 (en) | 2009-02-23 | 2017-04-18 | Gtx, Inc. | Estrogen receptor ligands and methods of use thereof |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ300739A (en) * | 1994-12-22 | 2000-05-26 | Ligand Pharm Inc | Steroid receptor modulator compounds |
| PT918774E (en) * | 1996-06-27 | 2002-05-31 | Ligand Pharm Inc | ANDROGENE RECEPTOR MODULATORS AND METHODS |
| JP2004509072A (en) * | 2000-06-28 | 2004-03-25 | ブリストル−マイヤーズ スクイブ カンパニー | Selective androgen receptor modulators and methods for their identification, design and use |
-
2001
- 2001-06-20 JP JP2002505777A patent/JP2004515462A/en active Pending
- 2001-06-20 AU AU2002215609A patent/AU2002215609A1/en not_active Abandoned
- 2001-06-20 WO PCT/US2001/019663 patent/WO2002000653A2/en not_active Ceased
- 2001-06-20 HU HU0303165A patent/HUP0303165A3/en unknown
- 2001-06-20 NZ NZ523802A patent/NZ523802A/en unknown
- 2001-06-20 MX MXPA02012563A patent/MXPA02012563A/en unknown
- 2001-06-20 CA CA002413683A patent/CA2413683A1/en not_active Abandoned
- 2001-06-20 BR BR0111869-2A patent/BR0111869A/en not_active IP Right Cessation
- 2001-06-20 EP EP01984054A patent/EP1299385A2/en not_active Withdrawn
-
2002
- 2002-12-20 NO NO20026167A patent/NO20026167L/en not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| WO2002000653A2 (en) | 2002-01-03 |
| AU2002215609A1 (en) | 2002-01-08 |
| NZ523802A (en) | 2005-11-25 |
| EP1299385A2 (en) | 2003-04-09 |
| CA2413683A1 (en) | 2002-01-03 |
| JP2004515462A (en) | 2004-05-27 |
| MXPA02012563A (en) | 2003-05-14 |
| HUP0303165A2 (en) | 2003-12-29 |
| HUP0303165A3 (en) | 2006-05-29 |
| NO20026167D0 (en) | 2002-12-20 |
| WO2002000653A3 (en) | 2002-07-25 |
| BR0111869A (en) | 2003-09-23 |
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| Date | Code | Title | Description |
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| FC2A | Withdrawal, rejection or dismissal of laid open patent application |