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NO20023614L - Pyrimidin-karboksamider som er anvendelige som inhibitorer for PDE4-isoenzymer - Google Patents

Pyrimidin-karboksamider som er anvendelige som inhibitorer for PDE4-isoenzymer

Info

Publication number
NO20023614L
NO20023614L NO20023614A NO20023614A NO20023614L NO 20023614 L NO20023614 L NO 20023614L NO 20023614 A NO20023614 A NO 20023614A NO 20023614 A NO20023614 A NO 20023614A NO 20023614 L NO20023614 L NO 20023614L
Authority
NO
Norway
Prior art keywords
inhibitors
pde4 isoenzymes
carboxamides useful
pyrimidine carboxamides
pyrimidine
Prior art date
Application number
NO20023614A
Other languages
English (en)
Other versions
NO20023614D0 (no
Inventor
Robert James Chambers
Thomas Victor Magee
Anthony Marfat
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of NO20023614D0 publication Critical patent/NO20023614D0/no
Publication of NO20023614L publication Critical patent/NO20023614L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
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    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

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  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
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  • Engineering & Computer Science (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pulmonology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Oncology (AREA)
  • Rheumatology (AREA)
  • Communicable Diseases (AREA)
  • Immunology (AREA)
  • Neurology (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Molecular Biology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
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  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Vascular Medicine (AREA)
  • Ophthalmology & Optometry (AREA)
  • Dermatology (AREA)
  • Psychiatry (AREA)
  • Biotechnology (AREA)
NO20023614A 2000-01-31 2002-07-30 Pyrimidin-karboksamider som er anvendelige som inhibitorer for PDE4-isoenzymer NO20023614L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17928200P 2000-01-31 2000-01-31
PCT/IB2001/000125 WO2001057025A1 (en) 2000-01-31 2001-01-30 Pyrimidine carboxamides useful as inhibitors of pde4 isozymes

Publications (2)

Publication Number Publication Date
NO20023614D0 NO20023614D0 (no) 2002-07-30
NO20023614L true NO20023614L (no) 2002-09-30

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NO20023614A NO20023614L (no) 2000-01-31 2002-07-30 Pyrimidin-karboksamider som er anvendelige som inhibitorer for PDE4-isoenzymer

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US (1) US6740655B2 (no)
EP (1) EP1252157B1 (no)
JP (1) JP2003522165A (no)
KR (1) KR20020071029A (no)
CN (1) CN1404480A (no)
AP (1) AP2002002590A0 (no)
AR (1) AR027336A1 (no)
AT (1) ATE269860T1 (no)
AU (1) AU2700301A (no)
BG (1) BG106868A (no)
BR (1) BR0107934A (no)
CA (1) CA2396458C (no)
CO (1) CO5271669A1 (no)
CR (1) CR6714A (no)
CZ (1) CZ20022413A3 (no)
DE (1) DE60103976T2 (no)
DK (1) DK1252157T3 (no)
DZ (1) DZ3406A1 (no)
EA (1) EA005028B1 (no)
EE (1) EE200200426A (no)
ES (1) ES2223772T3 (no)
GE (1) GEP20043385B (no)
GT (1) GT200100023A (no)
HK (1) HK1054232A1 (no)
HN (1) HN2001000018A (no)
HU (1) HUP0204271A3 (no)
IL (1) IL150486A0 (no)
IS (1) IS6444A (no)
MA (1) MA26871A1 (no)
MX (1) MXPA02007465A (no)
NO (1) NO20023614L (no)
NZ (1) NZ519726A (no)
OA (1) OA12170A (no)
PA (1) PA8511301A1 (no)
PE (1) PE20011059A1 (no)
PL (1) PL357555A1 (no)
PT (1) PT1252157E (no)
SK (1) SK10342002A3 (no)
SV (1) SV2001000298A (no)
TN (1) TNSN01019A1 (no)
TR (1) TR200402292T4 (no)
UY (1) UY26570A1 (no)
WO (1) WO2001057025A1 (no)
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Families Citing this family (86)

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Publication number Priority date Publication date Assignee Title
ES2165768B1 (es) 1999-07-14 2003-04-01 Almirall Prodesfarma Sa Nuevos derivados de quinuclidina y composiciones farmaceuticas que los contienen.
WO2001047493A1 (en) * 1999-12-24 2001-07-05 Glaxo Group Limited Pharmaceutical aerosol formulation of salmeterol and fluticasone propionate
US7776315B2 (en) 2000-10-31 2010-08-17 Boehringer Ingelheim Pharma Gmbh & Co. Kg Pharmaceutical compositions based on anticholinergics and additional active ingredients
DE10110772A1 (de) * 2001-03-07 2002-09-12 Boehringer Ingelheim Pharma Neue Arzneimittelkompositionen auf der Basis von Anticholinergika und PDE-IV-Inhibitoren
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