NO20015897L - Indolylpiperidinderivater som antihistaminiske og antiallergiske midler - Google Patents

Indolylpiperidinderivater som antihistaminiske og antiallergiske midler

Info

Publication number: NO20015897L
Authority: NO; Norway
Prior art keywords: antihistaminic; antiallergic agents; indolylpiperidine derivatives; indolylpiperidine; derivatives
Prior art date: 1999-06-04

Application number

NO20015897A

Other languages

English (en)

Other versions

NO20015897D0 (no

Inventor

Lluis Pages Santacana

Silvia Fonquerna Pou

Carles Puig Duran

Dolors Fernandez Forner

Original Assignee

Almirall Prodesfarma Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-06-04

Filing date

2001-12-03

Publication date

2001-12-03

2001-12-03 Application filed by Almirall Prodesfarma Sa filed Critical Almirall Prodesfarma Sa

2001-12-03 Publication of NO20015897D0 publication Critical patent/NO20015897D0/no

2001-12-03 Publication of NO20015897L publication Critical patent/NO20015897L/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/04—Drugs for disorders of the respiratory system for throat disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pulmonology (AREA)
Engineering & Computer Science (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Otolaryngology (AREA)
Immunology (AREA)
Ophthalmology & Optometry (AREA)
Dermatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

NO20015897A 1999-06-04 2001-12-03 Indolylpiperidinderivater som antihistaminiske og antiallergiske midler NO20015897L (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
ES009901232A ES2165274B1 (es)	1999-06-04	1999-06-04	Nuevos derivados de indolilpiperidina como agentes antihistaminicos y antialergicos.
PCT/EP2000/005010 WO2000075130A1 (en)	1999-06-04	2000-05-31	Indolylpiperidine derivatives as antihistaminic and antiallergic agents

Publications (2)

Publication Number	Publication Date
NO20015897D0 NO20015897D0 (no)	2001-12-03
NO20015897L true NO20015897L (no)	2001-12-03

Family

ID=8308707

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20015897A NO20015897L (no)	1999-06-04	2001-12-03	Indolylpiperidinderivater som antihistaminiske og antiallergiske midler

Country Status (35)

Country	Link
US (1)	US6683096B2 (no)
EP (1)	EP1183251B1 (no)
JP (1)	JP2003501424A (no)
KR (1)	KR100683454B1 (no)
CN (1)	CN1191246C (no)
AR (1)	AR029640A1 (no)
AT (1)	ATE259362T1 (no)
AU (1)	AU773164B2 (no)
BG (1)	BG106168A (no)
BR (1)	BR0011340A (no)
CA (1)	CA2375985A1 (no)
CO (1)	CO5180556A1 (no)
CZ (1)	CZ20014334A3 (no)
DE (1)	DE60008239T2 (no)
DK (1)	DK1183251T3 (no)
EE (1)	EE04717B1 (no)
ES (2)	ES2165274B1 (no)
HK (1)	HK1040990A1 (no)
HU (1)	HUP0203320A3 (no)
IL (1)	IL146629A0 (no)
MX (1)	MXPA01012425A (no)
MY (1)	MY127033A (no)
NO (1)	NO20015897L (no)
NZ (1)	NZ515649A (no)
PE (1)	PE20010208A1 (no)
PL (1)	PL196774B1 (no)
PT (1)	PT1183251E (no)
RU (1)	RU2246493C2 (no)
SI (1)	SI1183251T1 (no)
SK (1)	SK17042001A3 (no)
TR (1)	TR200103490T2 (no)
TW (1)	TWI226889B (no)
UA (1)	UA72517C2 (no)
WO (1)	WO2000075130A1 (no)
ZA (1)	ZA200109676B (no)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP1324996A2 (de)	2000-01-17	2003-07-09	Bayer CropScience AG	Substituierte arylketone
ES2172436B1 (es)	2000-10-31	2004-01-16	Almirall Prodesfarma Sa	Derivados de indolilpiperidina como agentes antihistaminicos y antialergicos.
AU2002243394A1 (en) *	2000-11-16	2002-06-24	Wyeth	Aryloxy piperidinyl derivatives for the treatment of depression
ES2201899B1 (es)	2002-04-01	2005-06-01	Almirall Prodesfarma, S.A.	Derivados de la azaindolilpiperidina como agentes antihistaminicos y antialergicos.
ES2201907B1 (es)	2002-05-29	2005-06-01	Almirall Prodesfarma, S.A.	Nuevos derivados de indolilpiperidina como potentes agentes antihistaminicos y antialergicos.
NZ547314A (en) *	2003-11-17	2010-02-26	Boehringer Ingelheim Int	Novel piperidine-substituted indoles- or hetero-derivatives thereof and their use as modulators of chemokine receptor (CCR-3)
US20050245540A1 (en) *	2003-12-09	2005-11-03	Fujisawa Pharmaceutical Co., Ltd.	New methods
ES2431524T3 (es)	2004-04-13	2013-11-26	Incyte Corporation	Derivados de piperazinilpiperidina como antagonistas de los receptores de quimiocinas
JP2008504279A (ja) *	2004-06-24	2008-02-14	インサイト・コーポレイション	アミド化合物およびその医薬としての使用
BRPI0512535A (pt)	2004-06-24	2008-03-25	Incyte Corp	compostos de piperidinas n-substituìdas, suas composições e métodos de modulações
DE602006012650D1 (de) *	2005-04-26	2010-04-15	Hypnion Inc	Benzisoxazolpiperidinverbindungen und verfahren zu deren anwendung
ATE531706T1 (de)	2005-04-30	2011-11-15	Boehringer Ingelheim Int	Neue piperidin-substituierte indole und ihre verwendung als ccr-3-modulatoren
US20060275516A1 (en) *	2005-06-02	2006-12-07	Ram A N S	Compositions and methods for the treatment of allergic rhinitis
WO2008030853A2 (en) *	2006-09-06	2008-03-13	Incyte Corporation	Combination therapy for human immunodeficiency virus infection
WO2008049874A1 (en)	2006-10-27	2008-05-02	Boehringer Ingelheim International Gmbh	Piperidyl-propane-thiol ccr3 modulators
PE20090188A1 (es) *	2007-03-15	2009-03-20	Novartis Ag	Compuestos heterociclicos como moduladores de la senda de hedgehog
US20100041663A1 (en)	2008-07-18	2010-02-18	Novartis Ag	Organic Compounds as Smo Inhibitors
CN101560179B (zh) *	2009-05-25	2012-04-18	浙江大学	具有h3受体亲和能力的含氮吲哚衍生物和用途
CN101747321B (zh) *	2009-12-22	2013-01-02	浙江大学	吲哚-3-苄胺衍生物及制备方法和用途
EP3040334A1 (en) *	2014-12-29	2016-07-06	Faes Farma, S.A.	New benzimidazole derivatives as antihistamine agents
MX2024001155A (es) *	2021-07-30	2024-07-01	Confo Therapeutics N V	Compuestos para el tratamiento del dolor, en particular el dolor neuropatico, y/u otras enfermedades o trastornos que se asocian con at2r y/o se?alizacion mediada por at2r.

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4742057A (en) *	1985-12-05	1988-05-03	Fujisawa Pharmaceutical Co., Ltd.	Antiallergic thiazole compounds
JPS63301881A (ja) *	1987-06-01	1988-12-08	Fujisawa Pharmaceut Co Ltd	インドリルピペリジン誘導体
DK733788A (da) *	1988-01-14	1989-07-15	Fujisawa Pharmaceutical Co	Indolylpiperidinderivater og fremgangsmaade til fremstilling deraf
GB8800795D0 (en) *	1988-01-14	1988-02-17	Fujisawa Pharmaceutical Co	New indolylpiperidine compounds processes for preparations thereof & pharmaceutical composition comprising same
GB8900382D0 (en) *	1989-01-09	1989-03-08	Janssen Pharmaceutica Nv	2-aminopyrimidinone derivatives
PH30434A (en) *	1989-04-07	1997-05-09	Janssen Pharmaceutica Nv	Hydroxyalkylfuranyl derivatives
EP0626968B1 (en) *	1992-02-13	2001-09-26	Merrell Pharmaceuticals Inc.	Piperidinyl thiacyclic derivatives
IT1271417B (it) *	1993-10-15	1997-05-28	Erregierre Ind Chim	Composti ad attivita' antiistaminica procedimento per la loro preperazione e composizioni farmaceutiche che li contengono.
DE19500689A1 (de)	1995-01-12	1996-07-18	Merck Patent Gmbh	Indolpiperidin-Derivate
DE19707628A1 (de)	1997-02-26	1998-08-27	Merck Patent Gmbh	Oxazolidinone
AR013669A1 (es) *	1997-10-07	2001-01-10	Smithkline Beecham Corp	Compuestos y metodos
AR028685A1 (es) *	2000-06-14	2003-05-21	Lundbeck & Co As H	Derivados de indol

1999
- 1999-06-04 ES ES009901232A patent/ES2165274B1/es not_active Expired - Fee Related
2000
- 2000-05-31 AT AT00940296T patent/ATE259362T1/de not_active IP Right Cessation
- 2000-05-31 HU HU0203320A patent/HUP0203320A3/hu unknown
- 2000-05-31 AU AU55276/00A patent/AU773164B2/en not_active Ceased
- 2000-05-31 EP EP00940296A patent/EP1183251B1/en not_active Expired - Lifetime
- 2000-05-31 IL IL14662900A patent/IL146629A0/xx unknown
- 2000-05-31 JP JP2001502413A patent/JP2003501424A/ja not_active Ceased
- 2000-05-31 SK SK1704-2001A patent/SK17042001A3/sk unknown
- 2000-05-31 RU RU2002100073/04A patent/RU2246493C2/ru not_active IP Right Cessation
- 2000-05-31 DK DK00940296T patent/DK1183251T3/da active
- 2000-05-31 DE DE2000608239 patent/DE60008239T2/de not_active Expired - Lifetime
- 2000-05-31 CN CNB008112819A patent/CN1191246C/zh not_active Expired - Fee Related
- 2000-05-31 WO PCT/EP2000/005010 patent/WO2000075130A1/en not_active Ceased
- 2000-05-31 BR BR0011340-9A patent/BR0011340A/pt not_active Application Discontinuation
- 2000-05-31 CZ CZ20014334A patent/CZ20014334A3/cs unknown
- 2000-05-31 TR TR2001/03490T patent/TR200103490T2/xx unknown
- 2000-05-31 UA UA2001118222A patent/UA72517C2/uk unknown
- 2000-05-31 PT PT00940296T patent/PT1183251E/pt unknown
- 2000-05-31 SI SI200030323T patent/SI1183251T1/xx unknown
- 2000-05-31 CA CA002375985A patent/CA2375985A1/en not_active Abandoned
- 2000-05-31 ES ES00940296T patent/ES2211559T3/es not_active Expired - Lifetime
- 2000-05-31 KR KR1020017015570A patent/KR100683454B1/ko not_active Expired - Fee Related
- 2000-05-31 PE PE2000000524A patent/PE20010208A1/es not_active Application Discontinuation
- 2000-05-31 MY MYPI20002439A patent/MY127033A/en unknown
- 2000-05-31 EE EEP200100653A patent/EE04717B1/xx not_active IP Right Cessation
- 2000-05-31 PL PL353164A patent/PL196774B1/pl not_active IP Right Cessation
- 2000-05-31 NZ NZ515649A patent/NZ515649A/en unknown
- 2000-05-31 HK HK02102119.0A patent/HK1040990A1/zh unknown
- 2000-05-31 MX MXPA01012425A patent/MXPA01012425A/es unknown
- 2000-06-02 TW TW089110816A patent/TWI226889B/zh not_active IP Right Cessation
- 2000-06-02 CO CO00041546A patent/CO5180556A1/es not_active Application Discontinuation
- 2000-06-02 AR ARP000102755A patent/AR029640A1/es not_active Application Discontinuation
2001
- 2001-11-23 ZA ZA200109676A patent/ZA200109676B/en unknown
- 2001-12-03 NO NO20015897A patent/NO20015897L/no not_active Application Discontinuation
- 2001-12-03 BG BG106168A patent/BG106168A/bg unknown
- 2001-12-04 US US10/006,416 patent/US6683096B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
HK1040990A1 (zh)	2002-06-28
BR0011340A (pt)	2002-03-05
CO5180556A1 (es)	2002-07-30
TWI226889B (en)	2005-01-21
IL146629A0 (en)	2002-07-25
CZ20014334A3 (cs)	2002-03-13
PT1183251E (pt)	2004-05-31
ES2165274A1 (es)	2002-03-01
AU5527600A (en)	2000-12-28
DE60008239D1 (de)	2004-03-18
CN1191246C (zh)	2005-03-02
JP2003501424A (ja)	2003-01-14
EE04717B1 (et)	2006-10-16
PL353164A1 (en)	2003-10-20
HUP0203320A2 (hu)	2003-02-28
DK1183251T3 (da)	2004-06-07
ES2211559T3 (es)	2004-07-16
EE200100653A (et)	2003-02-17
MXPA01012425A (es)	2002-06-04
US6683096B2 (en)	2004-01-27
BG106168A (bg)	2002-07-31
KR100683454B1 (ko)	2007-02-20
EP1183251A1 (en)	2002-03-06
ATE259362T1 (de)	2004-02-15
US20020147344A1 (en)	2002-10-10
MY127033A (en)	2006-11-30
EP1183251B1 (en)	2004-02-11
NZ515649A (en)	2003-08-29
NO20015897D0 (no)	2001-12-03
KR20020020721A (ko)	2002-03-15
TR200103490T2 (tr)	2002-04-22
PE20010208A1 (es)	2001-03-19
HUP0203320A3 (en)	2004-01-28
ES2165274B1 (es)	2003-04-01
CA2375985A1 (en)	2000-12-14
CN1368969A (zh)	2002-09-11
SI1183251T1 (en)	2004-06-30
DE60008239T2 (de)	2004-11-18
PL196774B1 (pl)	2008-01-31
AU773164B2 (en)	2004-05-20
AR029640A1 (es)	2003-07-10
RU2002100073A (ru)	2004-01-10
ZA200109676B (en)	2003-02-24
UA72517C2 (uk)	2005-03-15
WO2000075130A1 (en)	2000-12-14
RU2246493C2 (ru)	2005-02-20
SK17042001A3 (sk)	2002-04-04

Publication	Publication Date	Title
NO20015897L (no)	2001-12-03	Indolylpiperidinderivater som antihistaminiske og antiallergiske midler
DK1204649T3 (da)	2007-12-03	Arylmethylcarbonylaminothiazolderivater og deres anvendelse som antitumormidler
IS6385A (is)	2002-05-15	Ný notkun og nýjar N-asabísýkló-amíð afleiður
IS2116B (is)	2006-06-15	4-fenyl-pyridin afleiður
NO20021077D0 (no)	2002-03-05	Amino-triazolopyridin-derivater
DE60009747D1 (de)	2004-05-13	Admantan-derivate
ATE293104T1 (de)	2005-04-15	Thiazolylamid-derivate
IS6128A (is)	2001-10-26	13-Metýl-erýþrómýsín afleiður
DK1187814T3 (da)	2004-12-20	5-phenyl-pyrimidinderivater
ATE257148T1 (de)	2004-01-15	Propargyletherderivate
DK1154988T3 (da)	2004-11-22	Mevinolinderivater
ATE374747T1 (de)	2007-10-15	Monofluoralkylderivate
DK1187815T3 (da)	2006-06-19	4-phenyl-pyrimidinderivater
DK1218340T3 (da)	2004-03-29	4-hydroxybiphenylhydrazid-derivater
ATE293592T1 (de)	2005-05-15	Resorcinderivate
TR200002831A3 (tr)	2001-04-20	Kinolin-4-Il türevleri I
DE60025348D1 (de)	2006-03-30	Ethansulfonyl-piperidin-derivate
NO20020212L (no)	2002-01-15	3-amino-2-benzyl-1-fenyl-propanderivater
SI1330453T1 (sl)	2006-08-31	Derivati indolilpiperidina kot antihistaminicna in antialergijska sredstva
DK1178984T3 (da)	2003-06-10	1-trifluormethyl-4-hydroxy-7-piperidinylaminomethylchroman-derivater
DE59909774D1 (de)	2004-07-22	1-cycloalkylpyrazolyl-benzoyl-derivate
EG24068A (en)	2008-05-08	Indolylpiperidine derivatives as antihistaminic and antiallergic agents
SI1497292T1 (sl)	2006-10-31	Derivati azaindolilpiperidina kot antihistaminicna in antialergijska sredstva

Legal Events

Date	Code	Title	Description
2005-12-12	FC2A	Withdrawal, rejection or dismissal of laid open patent application