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NO20000702L - cGMP PDE-inhibitorer for behandling av erektil dysfunksjon - Google Patents

cGMP PDE-inhibitorer for behandling av erektil dysfunksjon

Info

Publication number
NO20000702L
NO20000702L NO20000702A NO20000702A NO20000702L NO 20000702 L NO20000702 L NO 20000702L NO 20000702 A NO20000702 A NO 20000702A NO 20000702 A NO20000702 A NO 20000702A NO 20000702 L NO20000702 L NO 20000702L
Authority
NO
Norway
Prior art keywords
alkyl
optionally substituted
cycloalkyl
treatment
erectile dysfunction
Prior art date
Application number
NO20000702A
Other languages
English (en)
Other versions
NO325558B1 (no
NO20000702D0 (no
Inventor
Peter Ellis
Nicholas Kenneth Terrett
Original Assignee
Pfizer Res & Dev
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10736901&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20000702(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Publication of NO20000702L publication Critical patent/NO20000702L/no
Application filed by Pfizer Res & Dev filed Critical Pfizer Res & Dev
Publication of NO20000702D0 publication Critical patent/NO20000702D0/no
Publication of NO325558B1 publication Critical patent/NO325558B1/no

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Reproductive Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Urology & Nephrology (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
  • Paper (AREA)
  • Hydroponics (AREA)
NO20000702A 1993-06-09 2000-02-11 Anvendelse av cGMP PDEv-inhibitorer for fremstilling av medikamenter til behandling av erektil dysfunksjon. NO325558B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB939311920A GB9311920D0 (en) 1993-06-09 1993-06-09 Therapeutic agents
PCT/EP1994/001580 WO1994028902A1 (en) 1993-06-09 1994-05-13 Pyrazolopyrimidinones for the treatment of impotence

Publications (3)

Publication Number Publication Date
NO20000702L true NO20000702L (no) 1995-11-24
NO20000702D0 NO20000702D0 (no) 2000-02-11
NO325558B1 NO325558B1 (no) 2008-06-16

Family

ID=10736901

Family Applications (3)

Application Number Title Priority Date Filing Date
NO19954757A NO309227B3 (no) 1993-06-09 1995-11-24 Anvendelse av 5-[2-etoksy-5-(4-metyl-1-piperazinylsulfonyl)fenyl]-1-metyl-3-n-propyl-1,6-dihydro-7H-pyrazolo[4,3-d]pyrimidin-7-on for fremstilling av et medikament for behandling av erektil dysfunksjon
NO20000703A NO321622B1 (no) 1993-06-09 2000-02-11 Pyrazolopyridmidioner for behandling av kvinnelig seksuell dysfunksjon
NO20000702A NO325558B1 (no) 1993-06-09 2000-02-11 Anvendelse av cGMP PDEv-inhibitorer for fremstilling av medikamenter til behandling av erektil dysfunksjon.

Family Applications Before (2)

Application Number Title Priority Date Filing Date
NO19954757A NO309227B3 (no) 1993-06-09 1995-11-24 Anvendelse av 5-[2-etoksy-5-(4-metyl-1-piperazinylsulfonyl)fenyl]-1-metyl-3-n-propyl-1,6-dihydro-7H-pyrazolo[4,3-d]pyrimidin-7-on for fremstilling av et medikament for behandling av erektil dysfunksjon
NO20000703A NO321622B1 (no) 1993-06-09 2000-02-11 Pyrazolopyridmidioner for behandling av kvinnelig seksuell dysfunksjon

Country Status (28)

Country Link
US (2) US6469012B1 (no)
EP (1) EP0702555B1 (no)
JP (4) JP2925034B2 (no)
KR (2) KR100262926B1 (no)
CN (2) CN1071118C (no)
AT (1) ATE163852T1 (no)
AU (1) AU676571C (no)
CA (1) CA2163446C (no)
CY (1) CY2099B1 (no)
CZ (1) CZ284946B6 (no)
DE (1) DE69408981T2 (no)
DK (1) DK0702555T3 (no)
EC (1) ECSP941102A (no)
ES (1) ES2113656T3 (no)
FI (1) FI955911A0 (no)
GB (2) GB9301192D0 (no)
GR (1) GR3026520T3 (no)
HU (1) HU227877B1 (no)
IL (3) IL109873A (no)
LV (1) LV12269B (no)
MY (1) MY111446A (no)
NO (3) NO309227B3 (no)
NZ (2) NZ314110A (no)
PL (1) PL311948A1 (no)
RU (1) RU2373938C9 (no)
TW (1) TW292971B (no)
WO (1) WO1994028902A1 (no)
ZA (1) ZA944018B (no)

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NO325558B1 (no) 2008-06-16
CZ284946B6 (cs) 1999-04-14
CA2163446C (en) 1998-07-07
GR3026520T3 (en) 1998-07-31
NO954757D0 (no) 1995-11-24
AU676571B2 (en) 1997-03-13
CN1071118C (zh) 2001-09-19
ZA944018B (en) 1995-12-08
NZ314110A (en) 2001-02-23
KR960702751A (ko) 1996-05-23
CN1742731A (zh) 2006-03-08
LV12269A (lv) 1999-05-20
TW292971B (no) 1996-12-11
JP2925034B2 (ja) 1999-07-26
WO1994028902A1 (en) 1994-12-22
CY2099B1 (en) 2002-04-05
ES2113656T3 (es) 1998-05-01
ECSP941102A (es) 1994-12-15
HU9501933D0 (en) 1995-09-28
NO20000703L (no) 1995-11-24
LV12269B (en) 1999-08-20
JPH09503996A (ja) 1997-04-22
RU2130776C1 (ru) 1999-05-27
JPH11263728A (ja) 1999-09-28
GB9301192D0 (en) 1993-06-09
HUT73420A (en) 1996-07-29
DE69408981T2 (de) 1998-07-02
IL109873A0 (en) 1994-10-07
IL109873A (en) 1998-12-27
JP2005097304A (ja) 2005-04-14
CZ324295A3 (en) 1996-07-17
NO321622B1 (no) 2006-06-12
IL121836A0 (en) 1998-02-22
GB9311920D0 (en) 1993-07-28
US6469012B1 (en) 2002-10-22
KR100262926B1 (ko) 2000-09-01
HU227877B1 (en) 2012-05-29
NO309227B3 (no) 2011-02-21
ATE163852T1 (de) 1998-03-15
NO309227B1 (no) 2001-01-02
AU676571C (en) 2004-01-15
RU2373938C2 (ru) 2009-11-27
CN1742731B (zh) 2012-02-01
CN1124926A (zh) 1996-06-19
FI955911A0 (fi) 1995-12-08
RU2373938C9 (ru) 2010-05-27
JPH11286444A (ja) 1999-10-19
NZ266463A (en) 1997-03-24
EP0702555B1 (en) 1998-03-11
IL121836A (en) 1998-12-27
NO954757L (no) 1995-11-24
CA2163446A1 (en) 1994-12-22
AU6797394A (en) 1995-01-03
PL311948A1 (en) 1996-03-18
EP0702555A1 (en) 1996-03-27
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