NO160370C - ANALOGUE PROCEDURE FOR THE PREPARATION OF PHYSIOLOGICALLY ACTIVE PENAM-1,1-DIOXYD COMPOUNDS. - Google Patents

ANALOGUE PROCEDURE FOR THE PREPARATION OF PHYSIOLOGICALLY ACTIVE PENAM-1,1-DIOXYD COMPOUNDS.

Info

Publication number: NO160370C
Authority: NO; Norway
Prior art keywords: dioxyd; penam; compounds; preparation; physiologically active
Prior art date: 1979-09-26

Application number

NO802836A

Other languages

Norwegian (no)

Other versions

NO160370B (en

NO802836L (en

Inventor

Wayne Ernest Barth

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1979-09-26

Filing date

1980-09-25

Publication date

1989-04-12

1980-09-25 Application filed by Pfizer filed Critical Pfizer

1981-03-27 Publication of NO802836L publication Critical patent/NO802836L/en

1983-03-25 Priority to NO83831082A priority Critical patent/NO160299C/en

1989-01-02 Publication of NO160370B publication Critical patent/NO160370B/en

1989-04-12 Publication of NO160370C publication Critical patent/NO160370C/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
- C07D499/32—Esters

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Cephalosporin Compounds (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Saccharide Compounds (AREA)

NO802836A 1979-09-26 1980-09-25 ANALOGUE PROCEDURE FOR THE PREPARATION OF PHYSIOLOGICALLY ACTIVE PENAM-1,1-DIOXYD COMPOUNDS. NO160370C (en)

Priority Applications (1)

Application Number	Priority Date	Filing Date	Title
NO83831082A NO160299C (en)	1979-09-26	1983-03-25	NEW PENAMINE COMPOUNDS WHICH MAY BE USED AS INTERMEDIATE PRODUCTS FOR THE PREPARATION OF BETA-LACTAMASE INHIBITIVE COMPOUNDS.

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US06/079,127 US4256733A (en)	1979-09-26	1979-09-26	Acetoxymethyl penam compounds as β-lactamase inhibitors

Publications (3)

Publication Number	Publication Date
NO802836L NO802836L (en)	1981-03-27
NO160370B NO160370B (en)	1989-01-02
NO160370C true NO160370C (en)	1989-04-12

Family

ID=22148609

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
NO802836A NO160370C (en)	1979-09-26	1980-09-25	ANALOGUE PROCEDURE FOR THE PREPARATION OF PHYSIOLOGICALLY ACTIVE PENAM-1,1-DIOXYD COMPOUNDS.
NO83831082A NO160299C (en)	1979-09-26	1983-03-25	NEW PENAMINE COMPOUNDS WHICH MAY BE USED AS INTERMEDIATE PRODUCTS FOR THE PREPARATION OF BETA-LACTAMASE INHIBITIVE COMPOUNDS.

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
NO83831082A NO160299C (en)	1979-09-26	1983-03-25	NEW PENAMINE COMPOUNDS WHICH MAY BE USED AS INTERMEDIATE PRODUCTS FOR THE PREPARATION OF BETA-LACTAMASE INHIBITIVE COMPOUNDS.

Country Status (36)

Country	Link
US (1)	US4256733A (en)
JP (1)	JPS6016958B2 (en)
KR (1)	KR840000796B1 (en)
AR (1)	AR224547A1 (en)
AT (1)	AT366384B (en)
AU (1)	AU517074B2 (en)
BE (1)	BE885389A (en)
CA (1)	CA1150242A (en)
CH (1)	CH645646A5 (en)
CS (1)	CS212284B2 (en)
DD (1)	DD153123A5 (en)
DE (1)	DE3035995C2 (en)
DK (1)	DK404980A (en)
EG (1)	EG14888A (en)
ES (1)	ES495354A0 (en)
FI (2)	FI67552C (en)
FR (1)	FR2465736A1 (en)
GB (2)	GB2059420B (en)
GR (1)	GR70065B (en)
HU (1)	HU183212B (en)
IE (2)	IE50506B1 (en)
IL (1)	IL61117A (en)
IN (1)	IN154557B (en)
IT (1)	IT1132754B (en)
LU (1)	LU82795A1 (en)
MX (1)	MX6580E (en)
NL (1)	NL185923C (en)
NO (2)	NO160370C (en)
NZ (1)	NZ195058A (en)
PH (1)	PH15697A (en)
PL (1)	PL126949B1 (en)
PT (1)	PT71837B (en)
SE (2)	SE449865B (en)
SU (1)	SU959628A3 (en)
YU (1)	YU41733B (en)
ZA (1)	ZA805132B (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4364957A (en) *	1979-09-26	1982-12-21	Pfizer Inc.	Bis-esters of alkanediols as antibacterial agents
US4511512A (en) *	1980-05-01	1985-04-16	Leo Pharmaceutical Products Ltd. A/S (Lovens Kemiske Produktionsaktiensel skab)	Substantially pure dicyclohexyl ammonium 6-β-bromo-penicillanate
US4361513A (en) *	1980-12-11	1982-11-30	Pfizer Inc.	Esters of penicillanic acid sulfone
US4474698A (en) *	1980-12-11	1984-10-02	Pfizer Inc.	Process for preparing esters of penicillanic acid sulfone
US4558042A (en) *	1981-05-06	1985-12-10	Farmitalia Carlo Erba S.P.A.	β-Lactam-containing antibacterial agents and β-lactamase inhibitors
ZA826687B (en) *	1981-09-14	1983-07-27	Pfizer	Beta-lactamase inhibiting 2-beta-substituted-2-alpha-methyl 5(r)penam-3-alpha-carboxylic acid 1,1-dioxides and intermediates therefor
JPS58185589A (en) *	1982-04-23	1983-10-29	Taiho Yakuhin Kogyo Kk	Penicillin derivative and preparation thereof
US4861768A (en) *	1986-02-27	1989-08-29	Taiho Pharmaceutical Company, Limited	2 β-substituted thiomethylpenicillin derivatives and their preparation and use
JPS62198687A (en) *	1986-02-27	1987-09-02	Taiho Yakuhin Kogyo Kk	2β-substituted thiomethylpenicillin derivatives
WO1993012250A1 (en) *	1991-12-19	1993-06-24	Novo Nordisk A/S	AN IMPROVED METHOD FOR THE PREPARATION OF CERTAIN β-LACTAM ANTIBIOTICS
CN115385934A (en) *	2022-10-26	2022-11-25	北京纳百生物科技有限公司	Sulbactam hapten as well as synthesis method and application thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
BE648188A (en)	1963-05-29	1964-09-16
IN149747B (en)	1977-06-07	1982-04-03	Pfizer

1979
- 1979-09-26 US US06/079,127 patent/US4256733A/en not_active Expired - Lifetime
1980
- 1980-08-13 SE SE8005714A patent/SE449865B/en not_active IP Right Cessation
- 1980-08-20 ZA ZA00805132A patent/ZA805132B/en unknown
- 1980-08-20 IN IN607/DEL/80A patent/IN154557B/en unknown
- 1980-09-19 SU SU802983144A patent/SU959628A3/en active
- 1980-09-19 HU HU802310A patent/HU183212B/en unknown
- 1980-09-22 PL PL1980226868A patent/PL126949B1/en unknown
- 1980-09-22 CS CS806403A patent/CS212284B2/en unknown
- 1980-09-23 GB GB8030639A patent/GB2059420B/en not_active Expired
- 1980-09-23 GR GR62939A patent/GR70065B/el unknown
- 1980-09-23 IL IL61117A patent/IL61117A/en unknown
- 1980-09-23 EG EG584/80A patent/EG14888A/en active
- 1980-09-23 CA CA000360886A patent/CA1150242A/en not_active Expired
- 1980-09-23 AT AT0474680A patent/AT366384B/en not_active IP Right Cessation
- 1980-09-24 DE DE3035995A patent/DE3035995C2/en not_active Expired
- 1980-09-24 AR AR282629A patent/AR224547A1/en active
- 1980-09-24 MX MX809044U patent/MX6580E/en unknown
- 1980-09-24 LU LU82795A patent/LU82795A1/en unknown
- 1980-09-24 PH PH24617A patent/PH15697A/en unknown
- 1980-09-24 KR KR1019800003721A patent/KR840000796B1/en not_active Expired
- 1980-09-25 ES ES495354A patent/ES495354A0/en active Granted
- 1980-09-25 FI FI803028A patent/FI67552C/en not_active IP Right Cessation
- 1980-09-25 AU AU62713/80A patent/AU517074B2/en not_active Ceased
- 1980-09-25 NL NLAANVRAGE8005344,A patent/NL185923C/en not_active IP Right Cessation
- 1980-09-25 JP JP55133639A patent/JPS6016958B2/en not_active Expired
- 1980-09-25 DK DK404980A patent/DK404980A/en not_active Application Discontinuation
- 1980-09-25 NZ NZ195058A patent/NZ195058A/en unknown
- 1980-09-25 YU YU2449/80A patent/YU41733B/en unknown
- 1980-09-25 IT IT24920/80A patent/IT1132754B/en active
- 1980-09-25 PT PT71837A patent/PT71837B/en unknown
- 1980-09-25 DD DD80224128A patent/DD153123A5/en unknown
- 1980-09-25 IE IE1998/80A patent/IE50506B1/en not_active IP Right Cessation
- 1980-09-25 IE IE1095/85A patent/IE50507B1/en unknown
- 1980-09-25 FR FR8020618A patent/FR2465736A1/en active Granted
- 1980-09-25 CH CH719980A patent/CH645646A5/en not_active IP Right Cessation
- 1980-09-25 NO NO802836A patent/NO160370C/en unknown
- 1980-09-25 BE BE0/202222A patent/BE885389A/en not_active IP Right Cessation
1983
- 1983-03-25 NO NO83831082A patent/NO160299C/en unknown
- 1983-07-22 GB GB08319784A patent/GB2125037B/en not_active Expired
1984
- 1984-01-30 FI FI840367A patent/FI67854C/en not_active IP Right Cessation
1985
- 1985-02-27 SE SE8500965A patent/SE461528B/en not_active IP Right Cessation

Also Published As

Publication number	Publication date
FI803028A7 (en)	1981-03-27
HU183212B (en)	1984-04-28
YU41733B (en)	1987-12-31
SE8005714L (en)	1981-03-27
CA1150242A (en)	1983-07-19
JPS6016958B2 (en)	1985-04-30
GR70065B (en)	1982-07-26
SE8500965D0 (en)	1985-02-27
IL61117A (en)	1983-10-31
IE801095L (en)	1981-01-09
DE3035995A1 (en)	1981-04-02
YU244980A (en)	1983-02-28
DD153123A5 (en)	1981-12-23
PH15697A (en)	1983-03-14
FI840367L (en)	1984-01-30
FI67552C (en)	1985-04-10
GB2059420B (en)	1984-03-14
PT71837A (en)	1980-10-01
FI67552B (en)	1984-12-31
PL126949B1 (en)	1983-09-30
PT71837B (en)	1981-07-09
GB2059420A (en)	1981-04-23
SE461528B (en)	1990-02-26
ES8106528A1 (en)	1981-08-16
GB2125037B (en)	1984-08-01
DK404980A (en)	1981-03-27
ZA805132B (en)	1981-12-30
PL226868A1 (en)	1981-10-16
AU517074B2 (en)	1981-07-09
SE449865B (en)	1987-05-25
CH645646A5 (en)	1984-10-15
CS212284B2 (en)	1982-03-26
IE801998L (en)	1981-03-26
JPS5657788A (en)	1981-05-20
NO160370B (en)	1989-01-02
BE885389A (en)	1981-03-25
AT366384B (en)	1982-04-13
DE3035995C2 (en)	1985-01-10
FR2465736A1 (en)	1981-03-27
IT1132754B (en)	1986-07-02
EG14888A (en)	1985-06-30
ES495354A0 (en)	1981-08-16
NO160299B (en)	1988-12-27
FI67854B (en)	1985-02-28
NL185923C (en)	1990-08-16
NZ195058A (en)	1982-12-07
GB2125037A (en)	1984-02-29
SU959628A3 (en)	1982-09-15
ATA474680A (en)	1981-08-15
LU82795A1 (en)	1981-04-17
FI840367A0 (en)	1984-01-30
KR830003494A (en)	1983-06-20
IT8024920A0 (en)	1980-09-25
MX6580E (en)	1985-07-24
NO160299C (en)	1989-04-05
AR224547A1 (en)	1981-12-15
AU6271380A (en)	1981-04-09
KR840000796B1 (en)	1984-06-12
FI67854C (en)	1985-06-10
IE50506B1 (en)	1986-04-30
NL185923B (en)	1990-03-16
FR2465736B1 (en)	1982-04-30
NO831082L (en)	1981-03-27
GB8319784D0 (en)	1983-08-24
NL8005344A (en)	1981-03-30
US4256733A (en)	1981-03-17
IE50507B1 (en)	1986-04-30
IN154557B (en)	1984-11-10
IL61117A0 (en)	1980-11-30
NO802836L (en)	1981-03-27

Publication	Publication Date	Title
NO145657C (en)	1982-05-05	ANALOGUE PROCEDURE FOR THE PREPARATION OF PHYSIOLOGICALLY ACTIVE ALKENDER DERIVATIVES.
NO154918C (en)	1987-01-14	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE DERIVATIVES OF 3,4,5-TRIHYDROXYPIPERIDINE.
NO155774C (en)	1987-05-27	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE IMIDAZO-DIAZEPINE DERIVATIVES.
NO810765L (en)	1981-09-07	PROCEDURE FOR THE PREPARATION OF PHARMASOYYTIC ACTIVE CARBOSTYRIC DERIVATIVES.
NO151362C (en)	1985-03-27	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE URINE DERIVATIVES.
NO803851L (en)	1981-06-22	PROCEDURE FOR THE PREPARATION OF 4,1`, 6`-TRICLOR-4,1`, 6`-TRIDEOXY-GALACTOSUCROSE
NO156785C (en)	1987-11-25	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE CYCLOBUTAN DERIVATIVES.
NO150203C (en)	1984-09-05	ANALOGUE PROCEDURE FOR PREPARATION OF PHYSIOLOGICALLY ACTIVE 4-HYDROXY-2H-1,2-BENZOTIAZINE-3-CARBOXAMIDE-1,1-DIOXYDES
NO150760C (en)	1984-12-12	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE AMINOTIAZOLES.
NO154058C (en)	1986-07-09	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE N-HETEROCYCLYL-4-PIPERIDINAMINES.
NO155055C (en)	1987-02-04	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE BETA-CARBOLIN-3-CARBOXYLIC ACID DERIVATIVES.
NO870240L (en)	1987-07-22	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE TIENO-1,4-DIAZEPINES.
NO150638C (en)	1984-11-21	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE BASIC ETHERS
NO802015L (en)	1981-01-07	PROCEDURE FOR THE PREPARATION OF PHYSIOLOGICALLY ACTIVE INDOLIZIN DERIVATIVES.
NO155665C (en)	1987-05-06	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 5,6,7,7A-TETRAHYDRO-4H-THIENO- (3,2-C) -PYRIDIN-2-ON DERIVATIVES.
NO152649C (en)	1985-10-30	ANALOGUE PROCEDURE FOR THE PREPARATION OF PHARMASOYYTIC ACTIVE PHENYLALKYLAMINES.
NO154268C (en)	1986-08-20	ANALOGUE PROCEDURE FOR THE PREPARATION OF NEW THERAPEUTIC ACTIVE 6ALFA-FLOUR-9A-CHLORINE-PREDNISOLON-17,21-DIESTERS.
NO149428C (en)	1984-04-18	PROCEDURE FOR THE PREPARATION OF PHYSIOLOGICALLY ACTIVE PROSTAGLAND INGREDIATES.
NO160370C (en)	1989-04-12	ANALOGUE PROCEDURE FOR THE PREPARATION OF PHYSIOLOGICALLY ACTIVE PENAM-1,1-DIOXYD COMPOUNDS.
NO148644C (en)	1983-11-16	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE SUGAR DERIVATIVES.
NO159090C (en)	1988-11-30	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE PYRIDOINDOL DERIVATIVES.
NO156167C (en)	1987-08-05	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE INDOLINON DERIVATIVES.
NO158800C (en)	1988-11-02	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE INDENDER DERIVATIVES.
NO147483C (en)	1983-04-20	ANALOGUE PROCEDURE FOR THE PREPARATION OF PHARMACOLOGICALLY ACTIVE BENZYLPYRIMIDINES.
NO164095C (en)	1990-09-05	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE ESTERS OF 3- (3-SUBSTITUTED-AMINO-2-HYDROXYPROPOXY) -4-SUBSTITUTED-1,2,5-THIADIAZOLD DERIVATIVES.