NL2009995C2 - Compositions. - Google Patents
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- Publication number
- NL2009995C2 NL2009995C2 NL2009995A NL2009995A NL2009995C2 NL 2009995 C2 NL2009995 C2 NL 2009995C2 NL 2009995 A NL2009995 A NL 2009995A NL 2009995 A NL2009995 A NL 2009995A NL 2009995 C2 NL2009995 C2 NL 2009995C2
- Authority
- NL
- Netherlands
- Prior art keywords
- composition
- capsule
- cetilistat
- formulation
- weight
- Prior art date
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- DBMJMQXJHONAFJ-UHFFFAOYSA-M Sodium laurylsulphate Chemical compound [Na+].CCCCCCCCCCCCOS([O-])(=O)=O DBMJMQXJHONAFJ-UHFFFAOYSA-M 0.000 claims description 29
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- 239000007787 solid Substances 0.000 description 1
- 210000002784 stomach Anatomy 0.000 description 1
- 239000007940 sugar coated tablet Substances 0.000 description 1
- 229910021653 sulphate ion Inorganic materials 0.000 description 1
- 239000000829 suppository Substances 0.000 description 1
- 239000000375 suspending agent Substances 0.000 description 1
- 239000000725 suspension Substances 0.000 description 1
- 239000003765 sweetening agent Substances 0.000 description 1
- 230000008961 swelling Effects 0.000 description 1
- 208000011580 syndromic disease Diseases 0.000 description 1
- 239000006188 syrup Substances 0.000 description 1
- 235000020357 syrup Nutrition 0.000 description 1
- JOXIMZWYDAKGHI-UHFFFAOYSA-M toluene-4-sulfonate Chemical compound CC1=CC=C(S([O-])(=O)=O)C=C1 JOXIMZWYDAKGHI-UHFFFAOYSA-M 0.000 description 1
- 235000021076 total caloric intake Nutrition 0.000 description 1
- 150000003626 triacylglycerols Chemical class 0.000 description 1
- 125000005270 trialkylamine group Chemical group 0.000 description 1
- LENZDBCJOHFCAS-UHFFFAOYSA-N tris Chemical compound OCC(N)(CO)CO LENZDBCJOHFCAS-UHFFFAOYSA-N 0.000 description 1
- 230000037220 weight regain Effects 0.000 description 1
- 238000003466 welding Methods 0.000 description 1
- 238000005550 wet granulation Methods 0.000 description 1
- 239000011701 zinc Substances 0.000 description 1
- 229910052725 zinc Inorganic materials 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
- C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
- C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D265/24—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in positions 2 and 4
- C07D265/26—Two oxygen atoms, e.g. isatoic anhydride
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/536—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/19—Cosmetics or similar toiletry preparations characterised by the composition containing inorganic ingredients
- A61K8/25—Silicon; Compounds thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/46—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing sulfur
- A61K8/463—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing sulfur containing sulfuric acid derivatives, e.g. sodium lauryl sulfate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/72—Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds
- A61K8/73—Polysaccharides
- A61K8/731—Cellulose; Quaternized cellulose derivatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/72—Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds
- A61K8/73—Polysaccharides
- A61K8/732—Starch; Amylose; Amylopectin; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q19/00—Preparations for care of the skin
- A61Q19/06—Preparations for care of the skin for countering cellulitis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2800/00—Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
- A61K2800/20—Chemical, physico-chemical or functional or structural properties of the composition as a whole
- A61K2800/30—Characterized by the absence of a particular group of ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2800/00—Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
- A61K2800/74—Biological properties of particular ingredients
- A61K2800/78—Enzyme modulators, e.g. Enzyme agonists
- A61K2800/782—Enzyme inhibitors; Enzyme antagonists
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Birds (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Child & Adolescent Psychology (AREA)
- Dermatology (AREA)
- Inorganic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Logic Circuits (AREA)
- Manipulation Of Pulses (AREA)
Claims (20)
1. Een samenstelling omvattende een mengsel van bestanddelen (i)-(v): (i) cetilistat; en 5 (ii) microkristallijn cellulose; en (iii) natriumlaurylsulfaat; en (iv) natriumzetmeelglycolaat; en (v) talk.
2. Samenstelling volgens conclusie 1, welke samenstelling geen polyvinylpyrrolidon bevat.
3. Samenstelling volgens conclusie 1 of conclusie 2 bestaande uit een mengsel van bestanddelen (i)-(v): 15 (i) cetilistat; en (ii) microkristallijn cellulose; en (iii) natriumlaurylsulfaat; en (iv) natriumzetmeelglycolaat; en (v) talk.
4. Een capsule bevattende een samenstelling volgens één der conclusies 1-3.
5. Capsule volgens conclusie 4 bevattende een samenstelling bestaande uit een mengsel van bestanddelen (i)-(v): 25 (i) cetilistat; en (ii) microkristallijn cellulose; en (iii) natriumlaurylsulfaat; en (iv) natriumzetmeelglycolaat; en (v) talk. 30
6. Capsule volgens conclusie 4 of conclusie 5, waarin de capsule 10 mg, 40 mg, 50 mg, 60 mg, 80 mg, 120 mg, of 150 mg cetilistat bevat.
7. Capsule volgens één der conclusies 4-6, waarin de capsule een harde capsule is.
8. Een kit omvattende een verpakking welke een aantal capsules bevat, waarin elke capsule een capsule volgens één der conclusies 4-7 is. 5
9. Kit volgens conclusie 8, waarin de verpakking een blister, blisterverpakking, buis, pot, fles, zak, wikkel of een andere houder is.
10. Een samenstelling volgens één der conclusies 1-3 of een capsule volgens één der 10 conclusies 4-7, voor gebruik in gewichtsbeheersing.
11. Samenstelling of capsule volgens conclusie 10, voor het helpen van een patiënt bij het beheersen van het gewicht van de patiënt.
12. Samenstelling of capsule volgens conclusie 10 of conclusie 11, voor gebruik in mensen welke een BMI hoger dan 18.5 kg/m2 hebben.
13. Een samenstelling volgens één der conclusies 1-3 of capsule volgens één der conclusies 4-7, voor gebruik bij gewichtsverlies. 20
14. Samenstelling of capsule volgens conclusie 13, voor het bevorderen van gewichtsverlies.
15. Samenstelling of capsule volgens conclusie 14, voor het helpen van een te zware 25 of zwaarlijvige patiënt met het verliezen van gewicht.
16. Samenstelling of capsule volgens één der conclusies 13 to 15, voor gebruik in mensen met een BMI hoger dan 18.5 kg/m2.
17. Een capsule voor gebruik in gewichtsbeheersing, waarin de capsule een samenstelling bevat welke bestaat uit een mengsel van bestanddelen (i)-(v): (i) cetilistat; en (ii) microkristallijn cellulose; en (iii) natriumlaurylsulfaat; en (iv) natriumzetmeelglycolaat; en (v) talk.
18. Een capsule voor gebruik bij gewichtsverlies, waarin de capsule een samenstelling bevat welke bestaat uit een mengsel van bestanddelen (i)-(v): (i) cetilistat; en (ii) microkristallijn cellulose; en (iii) natriumlaurylsulfaat; en 10 (iv) natriumzetmeelglycolaat; en (v) talk.
19. Een samenstelling in hoofdzaak zoals hierin beschreven onder verwijzing naar voorbeeld 1. 15
20. Een capsule in hoofdzaak zoals hierin beschreven onder verwijzing naar voorbeeld 1. 20 25 30
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB201122213 | 2011-12-23 | ||
| GBGB1122213.0A GB201122213D0 (en) | 2011-12-23 | 2011-12-23 | Compositions |
| GBGB1203082.1A GB201203082D0 (en) | 2012-02-22 | 2012-02-22 | Compositions |
| GB201203082 | 2012-02-22 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NL2009995A NL2009995A (en) | 2013-06-26 |
| NL2009995C2 true NL2009995C2 (en) | 2013-09-18 |
Family
ID=47560448
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NL2009995A NL2009995C2 (en) | 2011-12-23 | 2012-12-17 | Compositions. |
Country Status (8)
| Country | Link |
|---|---|
| AU (1) | AU2012101841A4 (nl) |
| DK (1) | DK201200198Y4 (nl) |
| ES (1) | ES2417408B1 (nl) |
| FI (1) | FI10194U1 (nl) |
| FR (1) | FR2984745B3 (nl) |
| IE (1) | IES20120556A2 (nl) |
| IT (1) | ITTO20121118A1 (nl) |
| NL (1) | NL2009995C2 (nl) |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6004996A (en) * | 1997-02-05 | 1999-12-21 | Hoffman-La Roche Inc. | Tetrahydrolipstatin containing compositions |
| AR022204A1 (es) * | 1999-01-08 | 2002-09-04 | Norgine Bv | Compuesto, proceso para su preparacion, composicion farmaceutica y producto comestible que lo comprende. |
| WO2006132440A1 (ja) * | 2005-06-09 | 2006-12-14 | Takeda Pharmaceutical Company Limited | 固形製剤 |
| JP2010254623A (ja) * | 2009-04-24 | 2010-11-11 | Takeda Chem Ind Ltd | ベンゾオキサジノン化合物の結晶 |
-
2012
- 2012-12-17 NL NL2009995A patent/NL2009995C2/en not_active IP Right Cessation
- 2012-12-17 AU AU2012101841A patent/AU2012101841A4/en not_active Ceased
- 2012-12-20 FR FR1262391A patent/FR2984745B3/fr not_active Expired - Lifetime
- 2012-12-20 DK DKBA201200198U patent/DK201200198Y4/da not_active IP Right Cessation
- 2012-12-20 IE IES20120556A patent/IES20120556A2/en not_active IP Right Cessation
- 2012-12-20 ES ES201231973A patent/ES2417408B1/es not_active Expired - Fee Related
- 2012-12-20 IT IT001118A patent/ITTO20121118A1/it unknown
- 2012-12-20 FI FIU20124262U patent/FI10194U1/fi not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| FR2984745B3 (fr) | 2017-12-22 |
| DK201200198Y4 (da) | 2018-09-17 |
| ES2417408R1 (es) | 2013-10-15 |
| IES86183B2 (en) | 2013-05-08 |
| ES2417408A2 (es) | 2013-08-07 |
| FI10194U1 (fi) | 2013-08-20 |
| AU2012101841A4 (en) | 2013-01-17 |
| FR2984745A3 (fr) | 2013-06-28 |
| DK201200198U1 (en) | 2013-04-12 |
| IES20120556A2 (en) | 2013-05-08 |
| NL2009995A (en) | 2013-06-26 |
| ITTO20121118A1 (it) | 2013-06-24 |
| ES2417408B1 (es) | 2014-11-26 |
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Legal Events
| Date | Code | Title | Description |
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| MM | Lapsed because of non-payment of the annual fee |
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