NL165178C - PROCESS FOR PREPARING A THERAPEUTIC PREPARATION USING A 6-FLUOR-16-METHYL STERID OF THE PREGNA SERIES AND METHOD FOR PREPARING A STERID AND FORMED USE THEREFOR. - Google Patents
PROCESS FOR PREPARING A THERAPEUTIC PREPARATION USING A 6-FLUOR-16-METHYL STERID OF THE PREGNA SERIES AND METHOD FOR PREPARING A STERID AND FORMED USE THEREFOR.Info
- Publication number
- NL165178C NL165178C NL7303262.A NL7303262A NL165178C NL 165178 C NL165178 C NL 165178C NL 7303262 A NL7303262 A NL 7303262A NL 165178 C NL165178 C NL 165178C
- Authority
- NL
- Netherlands
- Prior art keywords
- sterid
- preparing
- pregna
- fluor
- methyl
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- 230000001225 therapeutic effect Effects 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
- A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Rheumatology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pain & Pain Management (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US23333772A | 1972-03-09 | 1972-03-09 | |
| US31697372A | 1972-12-20 | 1972-12-20 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NL7303262A NL7303262A (en) | 1973-09-11 |
| NL165178B NL165178B (en) | 1980-10-15 |
| NL165178C true NL165178C (en) | 1981-03-16 |
Family
ID=26926821
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NL7303262.A NL165178C (en) | 1972-03-09 | 1973-03-08 | PROCESS FOR PREPARING A THERAPEUTIC PREPARATION USING A 6-FLUOR-16-METHYL STERID OF THE PREGNA SERIES AND METHOD FOR PREPARING A STERID AND FORMED USE THEREFOR. |
Country Status (13)
| Country | Link |
|---|---|
| JP (3) | JPS5331156B2 (en) |
| AR (1) | AR197216A1 (en) |
| AU (1) | AU468257B2 (en) |
| CH (3) | CH580116A5 (en) |
| DE (1) | DE2365992C3 (en) |
| DK (1) | DK133382B (en) |
| ES (1) | ES412235A1 (en) |
| FR (1) | FR2181802B1 (en) |
| GB (1) | GB1403962A (en) |
| HK (1) | HK62680A (en) |
| NL (1) | NL165178C (en) |
| PH (1) | PH14703A (en) |
| SE (1) | SE396756B (en) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1430223A (en) * | 1973-10-25 | 1976-03-31 | Upjohn Co | Anti-inflammatory composition comprising steroids |
| ZA77943B (en) * | 1976-03-19 | 1977-12-28 | Upjohn Co | Topical steroid clindamycin preparations |
| NL187577C (en) * | 1978-04-05 | 1991-11-18 | Sibla Srl | 3-ACETOXY-9BETA, 11BETA-EPOXY-PREGNA-1,3,5-TRIEN, PROCESS FOR THE PREPARATION THEREOF, AND PROCESS FOR THE PREPARATION OF 6-alpha-halogen-1,4-diene-3-ones. |
| DE3068965D1 (en) | 1979-11-16 | 1984-09-20 | Sterosynt Ltd | 6-alpha-fluoro-16-methyl-prednisolone-17,21 diesters and pharmaceutical compositions containing them |
| JPH0240957Y2 (en) * | 1986-08-30 | 1990-10-31 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB933859A (en) * | 1958-09-06 | 1963-08-14 | Syntex S.A. |
-
1973
- 1973-02-22 DE DE2365992A patent/DE2365992C3/en not_active Expired
- 1973-02-22 GB GB877373A patent/GB1403962A/en not_active Expired
- 1973-02-26 AU AU52579/73A patent/AU468257B2/en not_active Expired
- 1973-02-26 CH CH277073A patent/CH580116A5/xx not_active IP Right Cessation
- 1973-02-26 CH CH396076A patent/CH580118A5/xx not_active IP Right Cessation
- 1973-02-26 CH CH395976A patent/CH580117A5/xx not_active IP Right Cessation
- 1973-03-02 ES ES412235A patent/ES412235A1/en not_active Expired
- 1973-03-07 JP JP2625073A patent/JPS5331156B2/ja not_active Expired
- 1973-03-07 AR AR246918A patent/AR197216A1/en active
- 1973-03-08 NL NL7303262.A patent/NL165178C/en not_active IP Right Cessation
- 1973-03-08 SE SE7303287A patent/SE396756B/en unknown
- 1973-03-08 DK DK128173AA patent/DK133382B/en unknown
- 1973-03-08 FR FR7308331A patent/FR2181802B1/fr not_active Expired
-
1976
- 1976-05-06 PH PH18405A patent/PH14703A/en unknown
- 1976-09-09 JP JP51107346A patent/JPS5227760A/en active Granted
- 1976-09-09 JP JP51107347A patent/JPS5227761A/en active Granted
-
1980
- 1980-11-06 HK HK626/80A patent/HK62680A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JPS5331156B2 (en) | 1978-08-31 |
| AR197216A1 (en) | 1974-03-22 |
| CH580118A5 (en) | 1976-09-30 |
| GB1403962A (en) | 1975-08-28 |
| FR2181802B1 (en) | 1976-10-22 |
| CH580117A5 (en) | 1976-09-30 |
| DE2365992B2 (en) | 1981-08-06 |
| JPS5227760A (en) | 1977-03-02 |
| AU468257B2 (en) | 1976-01-08 |
| PH14703A (en) | 1981-11-10 |
| SE396756B (en) | 1977-10-03 |
| FR2181802A1 (en) | 1973-12-07 |
| HK62680A (en) | 1980-11-14 |
| DE2365992C3 (en) | 1982-05-19 |
| ES412235A1 (en) | 1976-01-01 |
| DE2365992A1 (en) | 1977-05-18 |
| CH580116A5 (en) | 1976-09-30 |
| JPS4899157A (en) | 1973-12-15 |
| DK133382B (en) | 1976-05-10 |
| JPS5344465B2 (en) | 1978-11-29 |
| AU5257973A (en) | 1974-08-29 |
| JPS5227761A (en) | 1977-03-02 |
| NL7303262A (en) | 1973-09-11 |
| DK133382C (en) | 1976-10-04 |
| JPS5344464B2 (en) | 1978-11-29 |
| NL165178B (en) | 1980-10-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| V4 | Lapsed because of reaching the maximum lifetime of a patent |