MXPA03008727A - Procedimiento para la preparacion de derivados de imidazol tetrasubstituidos y estructuras cristalinas novedosas de los mismos. - Google Patents
Procedimiento para la preparacion de derivados de imidazol tetrasubstituidos y estructuras cristalinas novedosas de los mismos.Info
- Publication number
- MXPA03008727A MXPA03008727A MXPA03008727A MXPA03008727A MXPA03008727A MX PA03008727 A MXPA03008727 A MX PA03008727A MX PA03008727 A MXPA03008727 A MX PA03008727A MX PA03008727 A MXPA03008727 A MX PA03008727A MX PA03008727 A MXPA03008727 A MX PA03008727A
- Authority
- MX
- Mexico
- Prior art keywords
- imidazole derivatives
- preparation
- crystalline structures
- novel crystalline
- tetrasubstituted imidazole
- Prior art date
Links
- 150000002460 imidazoles Chemical class 0.000 title abstract 2
- 229940079865 intestinal antiinfectives imidazole derivative Drugs 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 238000004519 manufacturing process Methods 0.000 abstract 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/44—Radicals substituted by doubly-bound oxygen, sulfur, or nitrogen atoms, or by two such atoms singly-bound to the same carbon atom
- C07D213/46—Oxygen atoms
- C07D213/51—Acetal radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyridine Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
La presente invencion se refiere a un procedimiento para preparar derivados de imidazol tetrasubstituidos de la formula general (I) en donde R1, R2, R3, y R4 son como se definen en la especificacion posterior; la presente invencion tambien se refiere a un procedimiento para preparar un compuesto de la formula (II) (ver formula) y estructuras cristalinas novedosas del compuesto de la formula (II).
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US27860701P | 2001-03-26 | 2001-03-26 | |
| US10/081,553 US7067671B2 (en) | 2001-03-26 | 2002-02-22 | Process for the preparation of tetrasubstituted imidazole derivatives and novel crystalline structures thereof |
| PCT/US2002/005419 WO2002076974A2 (en) | 2001-03-26 | 2002-02-22 | Process for the preparation of tetrasubstituted imidazole derivatives and novel crystalline structures thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MXPA03008727A true MXPA03008727A (es) | 2004-07-30 |
Family
ID=23065636
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MXPA03008727A MXPA03008727A (es) | 2001-03-26 | 2002-02-22 | Procedimiento para la preparacion de derivados de imidazol tetrasubstituidos y estructuras cristalinas novedosas de los mismos. |
Country Status (15)
| Country | Link |
|---|---|
| US (2) | US7067671B2 (es) |
| EP (1) | EP1392678A2 (es) |
| JP (1) | JP2005504004A (es) |
| KR (1) | KR20040005897A (es) |
| CN (3) | CN1781903A (es) |
| BR (1) | BR0208462A (es) |
| CA (1) | CA2442364A1 (es) |
| CZ (1) | CZ20032871A3 (es) |
| HU (1) | HUP0303618A3 (es) |
| MX (1) | MXPA03008727A (es) |
| NZ (1) | NZ528405A (es) |
| RU (1) | RU2286342C2 (es) |
| SK (1) | SK13132003A3 (es) |
| WO (1) | WO2002076974A2 (es) |
| YU (1) | YU75703A (es) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2461100C (en) * | 2001-10-22 | 2009-12-01 | Tanabe Seiyaku Co., Ltd. | 4-imidazolin-2-one compounds |
| US7473695B2 (en) | 2001-10-22 | 2009-01-06 | Mitsubishi Tanabe Pharma Corporation | 4-imidazolin-2-one compounds |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1010969B (de) | 1953-07-03 | 1957-06-27 | Hoffmann La Roche | Verfahren zur Herstellung von neuen 2-Imidazolonen |
| DE2950478A1 (de) | 1979-12-14 | 1981-06-19 | A. Nattermann & Cie GmbH, 5000 Köln | 4,5-diaryl-4-imidazolin-2-on-derivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate |
| DE3504677A1 (de) * | 1985-02-12 | 1986-08-14 | A. Nattermann & Cie GmbH, 5000 Köln | Neue imidazol-2-yloxyalkansaeuren und ihre derivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate |
| ES2149201T3 (es) * | 1992-02-11 | 2000-11-01 | Smithkline Beecham Corp | Inhibidores de coa-it y paf. |
| US5593992A (en) | 1993-07-16 | 1997-01-14 | Smithkline Beecham Corporation | Compounds |
| US5670527A (en) | 1993-07-16 | 1997-09-23 | Smithkline Beecham Corporation | Pyridyl imidazole compounds and compositions |
| AU7138298A (en) * | 1997-04-24 | 1998-11-13 | Ortho-Mcneil Corporation, Inc. | Substituted imidazoles useful in the treatment of inflammatory diseases |
| FR2772377B1 (fr) | 1997-12-12 | 2000-01-07 | Synthelabo | Derives de 1-(1-h-imidazol-2-yl)pyrrolidines et 1-(1-h-imidazol-2-ylpiperidines), leur preparation et leur application en therapeutique |
-
2002
- 2002-02-22 MX MXPA03008727A patent/MXPA03008727A/es unknown
- 2002-02-22 RU RU2003128875/04A patent/RU2286342C2/ru not_active IP Right Cessation
- 2002-02-22 SK SK1313-2003A patent/SK13132003A3/sk not_active Application Discontinuation
- 2002-02-22 KR KR10-2003-7012494A patent/KR20040005897A/ko not_active Ceased
- 2002-02-22 EP EP02753758A patent/EP1392678A2/en not_active Withdrawn
- 2002-02-22 CN CNA2005101370168A patent/CN1781903A/zh active Pending
- 2002-02-22 JP JP2002576232A patent/JP2005504004A/ja active Pending
- 2002-02-22 HU HU0303618A patent/HUP0303618A3/hu unknown
- 2002-02-22 CN CNA2005101317999A patent/CN1800178A/zh active Pending
- 2002-02-22 YU YU75703A patent/YU75703A/sh unknown
- 2002-02-22 US US10/081,553 patent/US7067671B2/en not_active Expired - Fee Related
- 2002-02-22 CZ CZ20032871A patent/CZ20032871A3/cs unknown
- 2002-02-22 CA CA002442364A patent/CA2442364A1/en not_active Abandoned
- 2002-02-22 CN CNA028105133A patent/CN1511150A/zh active Pending
- 2002-02-22 WO PCT/US2002/005419 patent/WO2002076974A2/en not_active Ceased
- 2002-02-22 BR BR0208462-7A patent/BR0208462A/pt not_active IP Right Cessation
- 2002-02-22 NZ NZ528405A patent/NZ528405A/en unknown
-
2005
- 2005-10-04 US US11/243,277 patent/US7132544B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US20060030712A1 (en) | 2006-02-09 |
| SK13132003A3 (sk) | 2004-07-07 |
| BR0208462A (pt) | 2004-03-02 |
| KR20040005897A (ko) | 2004-01-16 |
| US7067671B2 (en) | 2006-06-27 |
| NZ528405A (en) | 2005-07-29 |
| WO2002076974A3 (en) | 2003-02-13 |
| RU2003128875A (ru) | 2005-04-20 |
| CA2442364A1 (en) | 2002-10-03 |
| JP2005504004A (ja) | 2005-02-10 |
| RU2286342C2 (ru) | 2006-10-27 |
| US7132544B2 (en) | 2006-11-07 |
| CN1800178A (zh) | 2006-07-12 |
| YU75703A (sh) | 2006-05-25 |
| CZ20032871A3 (cs) | 2004-08-18 |
| US20030045723A1 (en) | 2003-03-06 |
| HUP0303618A2 (hu) | 2005-04-28 |
| WO2002076974A2 (en) | 2002-10-03 |
| EP1392678A2 (en) | 2004-03-03 |
| CN1781903A (zh) | 2006-06-07 |
| CN1511150A (zh) | 2004-07-07 |
| HUP0303618A3 (en) | 2005-06-28 |
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