MXPA03002891A - Naftilsalicilaniluros como agentes antiinflamatorios y antimicrobianos. - Google Patents
Naftilsalicilaniluros como agentes antiinflamatorios y antimicrobianos.Info
- Publication number
- MXPA03002891A MXPA03002891A MXPA03002891A MXPA03002891A MXPA03002891A MX PA03002891 A MXPA03002891 A MX PA03002891A MX PA03002891 A MXPA03002891 A MX PA03002891A MX PA03002891 A MXPA03002891 A MX PA03002891A MX PA03002891 A MXPA03002891 A MX PA03002891A
- Authority
- MX
- Mexico
- Prior art keywords
- substituted
- naphthylsalicylanilides
- alkyl
- antiinflammatory agents
- antimicrobial
- Prior art date
Links
- 239000002260 anti-inflammatory agent Substances 0.000 title abstract 2
- 229940121363 anti-inflammatory agent Drugs 0.000 title abstract 2
- 230000000845 anti-microbial effect Effects 0.000 title 1
- 239000004599 antimicrobial Substances 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- -1 methoxy, benzoyl Chemical group 0.000 abstract 2
- 125000001624 naphthyl group Chemical group 0.000 abstract 2
- 238000006467 substitution reaction Methods 0.000 abstract 2
- 241000192125 Firmicutes Species 0.000 abstract 1
- JCXJVPUVTGWSNB-UHFFFAOYSA-N Nitrogen dioxide Chemical compound O=[N]=O JCXJVPUVTGWSNB-UHFFFAOYSA-N 0.000 abstract 1
- 230000000844 anti-bacterial effect Effects 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
- C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C255/58—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton
- C07C255/60—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton at least one of the singly-bound nitrogen atoms being acylated
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
- C07C235/70—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton
- C07C235/84—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton with the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a six-membered aromatic ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US23731900P | 2000-10-02 | 2000-10-02 | |
| PCT/US2001/042436 WO2002028819A1 (en) | 2000-10-02 | 2001-10-02 | Naphthylsalicylanilides as antimicrobial and antiinflammatory agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MXPA03002891A true MXPA03002891A (es) | 2003-10-15 |
Family
ID=22893236
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MXPA03002891A MXPA03002891A (es) | 2000-10-02 | 2001-10-02 | Naftilsalicilaniluros como agentes antiinflamatorios y antimicrobianos. |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US6407288B1 (es) |
| EP (1) | EP1328507B1 (es) |
| JP (1) | JP4086658B2 (es) |
| CN (1) | CN1249019C (es) |
| AT (1) | ATE356798T1 (es) |
| AU (1) | AU2002211842A1 (es) |
| CA (1) | CA2424396C (es) |
| DE (1) | DE60127285T2 (es) |
| DK (1) | DK1328507T3 (es) |
| MX (1) | MXPA03002891A (es) |
| WO (1) | WO2002028819A1 (es) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7319112B2 (en) | 2000-07-14 | 2008-01-15 | The Procter & Gamble Co. | Non-halogenated antibacterial agents and processes for making same |
| US7709026B2 (en) * | 2001-10-29 | 2010-05-04 | Columbia Laboratories, Inc. | Low concentration of peroxide for treating or preventing vaginal infections |
| AU2003242127A1 (en) * | 2002-06-05 | 2003-12-22 | Institute Of Medicinal Molecular Design, Inc. | Inhibitors against the activation of ap-1 and nfat |
| JPWO2003103658A1 (ja) * | 2002-06-05 | 2005-10-06 | 株式会社医薬分子設計研究所 | 免疫関連プロテインキナーゼ阻害剤 |
| US20060122243A1 (en) * | 2002-06-06 | 2006-06-08 | Susumu Muto | Antiallergic |
| JP4743382B2 (ja) | 2002-06-06 | 2011-08-10 | 株式会社医薬分子設計研究所 | Ｏ−置換ヒドロキシアリール誘導体 |
| WO2003103655A1 (ja) * | 2002-06-10 | 2003-12-18 | 株式会社医薬分子設計研究所 | 癌治療剤 |
| EP1535609A4 (en) * | 2002-06-10 | 2009-01-07 | Inst Med Molecular Design Inc | Nf-kb activation inhibitors |
| AU2003251944B2 (en) | 2002-07-15 | 2008-06-26 | Myriad Genetics, Inc. | Compounds, compositions, and methods employing same |
| EP1539681A2 (en) * | 2002-09-18 | 2005-06-15 | The Procter & Gamble Company | Non-halogenated antibacterial agents and processes for making same |
| CN104546857B (zh) * | 2013-10-18 | 2017-01-04 | 北京北科德源生物医药科技有限公司 | 化合物naphthoylenequinazolone的抗菌用途 |
| US20190328687A1 (en) * | 2014-11-17 | 2019-10-31 | Victoria Link Limited | Antibacterial Compounds |
| EP4061351A4 (en) * | 2019-11-18 | 2023-12-20 | The Regents of the University of California | Dual androgen receptor/akr1c3 inhibitors |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4287191A (en) * | 1980-04-14 | 1981-09-01 | The Research Foundation Of State University Of New York | Novel salicylanilides and microbiocidal compositions and uses thereof |
| US4358443A (en) * | 1980-04-14 | 1982-11-09 | The Research Foundation Of State University Of New York | Method and composition for controlling the growth of microorganisms |
| US4742083A (en) * | 1983-08-24 | 1988-05-03 | Lever Brothers Company | Method of relieving pain and inflammatory conditions employing substituted salicylamides |
| US4939132A (en) * | 1985-04-15 | 1990-07-03 | The Research Foundation Of State University Of New York | Novel 5-alkylsulfonylsalicylanilides and microbiocidal compositions for controlling the growth of microorganisms |
| US5958911A (en) * | 1996-11-05 | 1999-09-28 | The Research Foundation Of State University Of New York | Method of relieving inflammation by using 5-alkylsulfonylsalicylanilides |
-
2001
- 2001-10-02 MX MXPA03002891A patent/MXPA03002891A/es active IP Right Grant
- 2001-10-02 AU AU2002211842A patent/AU2002211842A1/en not_active Abandoned
- 2001-10-02 JP JP2002532406A patent/JP4086658B2/ja not_active Expired - Lifetime
- 2001-10-02 CA CA002424396A patent/CA2424396C/en not_active Expired - Fee Related
- 2001-10-02 EP EP01979927A patent/EP1328507B1/en not_active Expired - Lifetime
- 2001-10-02 DK DK01979927T patent/DK1328507T3/da active
- 2001-10-02 DE DE60127285T patent/DE60127285T2/de not_active Expired - Fee Related
- 2001-10-02 CN CNB018167055A patent/CN1249019C/zh not_active Expired - Fee Related
- 2001-10-02 AT AT01979927T patent/ATE356798T1/de not_active IP Right Cessation
- 2001-10-02 US US09/969,071 patent/US6407288B1/en not_active Expired - Lifetime
- 2001-10-02 WO PCT/US2001/042436 patent/WO2002028819A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| EP1328507B1 (en) | 2007-03-14 |
| US6407288B1 (en) | 2002-06-18 |
| EP1328507A1 (en) | 2003-07-23 |
| US20020065322A1 (en) | 2002-05-30 |
| EP1328507A4 (en) | 2005-07-27 |
| CA2424396C (en) | 2009-12-08 |
| WO2002028819A1 (en) | 2002-04-11 |
| CA2424396A1 (en) | 2002-04-11 |
| AU2002211842A1 (en) | 2002-04-15 |
| DE60127285T2 (de) | 2007-12-20 |
| ATE356798T1 (de) | 2007-04-15 |
| DE60127285D1 (de) | 2007-04-26 |
| JP4086658B2 (ja) | 2008-05-14 |
| CN1468210A (zh) | 2004-01-14 |
| DK1328507T3 (da) | 2007-07-02 |
| JP2004510756A (ja) | 2004-04-08 |
| CN1249019C (zh) | 2006-04-05 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant or registration |