MXPA02003024A - Antibioticos de acido 7-acilamino-3-heteroaril-3-cefem caboxilico y profarmacos de los mismos. - Google Patents
Antibioticos de acido 7-acilamino-3-heteroaril-3-cefem caboxilico y profarmacos de los mismos.Info
- Publication number
- MXPA02003024A MXPA02003024A MXPA02003024A MXPA02003024A MXPA02003024A MX PA02003024 A MXPA02003024 A MX PA02003024A MX PA02003024 A MXPA02003024 A MX PA02003024A MX PA02003024 A MXPA02003024 A MX PA02003024A MX PA02003024 A MXPA02003024 A MX PA02003024A
- Authority
- MX
- Mexico
- Prior art keywords
- heteroarylthio
- acylamino
- prodrugs
- carboxylic acid
- acid antibiotics
- Prior art date
Links
- 239000002253 acid Substances 0.000 title 1
- 125000004442 acylamino group Chemical group 0.000 title 1
- 239000003242 anti bacterial agent Substances 0.000 title 1
- 229940088710 antibiotic agent Drugs 0.000 title 1
- -1 heteroarylthio 3 cephem Chemical compound 0.000 title 1
- 229940002612 prodrug Drugs 0.000 title 1
- 239000000651 prodrug Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/70—Sulfur atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/08—1,2,4-Thiadiazoles; Hydrogenated 1,2,4-thiadiazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/645—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms
- C07F9/6503—Five-membered rings
- C07F9/6506—Five-membered rings having the nitrogen atoms in positions 1 and 3
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Oncology (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Communicable Diseases (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US15549699P | 1999-09-22 | 1999-09-22 | |
| PCT/US2000/026069 WO2001021623A1 (en) | 1999-09-22 | 2000-09-21 | 7-acylamino-3-heteroarylthio-3-cephem carboxylic acid antibiotics and prodrugs thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MXPA02003024A true MXPA02003024A (es) | 2003-09-25 |
Family
ID=22555673
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MXPA02003024A MXPA02003024A (es) | 1999-09-22 | 2000-09-21 | Antibioticos de acido 7-acilamino-3-heteroaril-3-cefem caboxilico y profarmacos de los mismos. |
Country Status (24)
| Country | Link |
|---|---|
| EP (1) | EP1222194B1 (es) |
| JP (1) | JP2003509512A (es) |
| KR (1) | KR20020068508A (es) |
| CN (1) | CN1206231C (es) |
| AR (1) | AR029004A1 (es) |
| AT (1) | ATE297934T1 (es) |
| AU (1) | AU784077B2 (es) |
| BR (1) | BR0014230A (es) |
| CA (1) | CA2385479A1 (es) |
| CZ (1) | CZ2002993A3 (es) |
| DE (1) | DE60020862D1 (es) |
| HK (1) | HK1048121B (es) |
| HU (1) | HUP0202663A3 (es) |
| IL (2) | IL148669A0 (es) |
| MX (1) | MXPA02003024A (es) |
| MY (1) | MY136038A (es) |
| NO (1) | NO20021416L (es) |
| NZ (1) | NZ517761A (es) |
| PL (1) | PL354919A1 (es) |
| RU (1) | RU2225868C2 (es) |
| SK (1) | SK4122002A3 (es) |
| TW (1) | TWI283682B (es) |
| WO (1) | WO2001021623A1 (es) |
| ZA (1) | ZA200202065B (es) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6534656B2 (en) * | 2001-05-31 | 2003-03-18 | North Carolina State University | Short synthesis of pyridine-based pharmaceutical intermediates |
| WO2004098500A2 (en) * | 2003-04-30 | 2004-11-18 | Trine Pharmaceuticals, Inc. | CARBACEPHEM ss-LACTAM ANTIBIOTICS |
| CN111187281B (zh) * | 2020-02-11 | 2023-03-14 | 广西科技大学 | 含胍基的头孢菌素衍生物及其制备方法 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MA18891A1 (fr) * | 1979-07-05 | 1981-04-01 | Ciba Geigy Ag | Composes d'amino-thiadiazolyle,procede pour leur preparation |
| EP0025017A1 (de) * | 1979-08-28 | 1981-03-11 | Ciba-Geigy Ag | Polyazathiaverbindungen, Verfahren zu ihrer Herstellung, pharmazeutische Präparate enthaltend solche Verbindungen und Verwendung von letzteren |
| WO1992005156A1 (en) * | 1990-09-13 | 1992-04-02 | Smithkline Beecham Corporation | Pyridylthio or pyridyloxy alkanoic acids |
| JPH09511738A (ja) * | 1994-04-01 | 1997-11-25 | マイクロサイド・ファーマシューティカルズ・インコーポレーテッド | セファロスポリン抗生物質 |
| US5498777A (en) * | 1994-07-20 | 1996-03-12 | Merck & Co., Inc. | 3-thioheteroaryl cephalosporin compounds, compositions and methods of use |
| AU5985596A (en) * | 1995-05-31 | 1996-12-18 | Microcide Pharmaceuticals, Inc. | Cephalosporin antibiotics |
| MY127641A (en) * | 1995-10-12 | 2006-12-29 | Essential Therapeutics Inc | Cephalosporin antibiotics |
| JP4174093B2 (ja) * | 1998-01-09 | 2008-10-29 | 富士フイルムファインケミカルズ株式会社 | トリアゾール誘導体ハロゲン化合物の製造方法 |
| ATE221889T1 (de) * | 1998-05-13 | 2002-08-15 | Lg Chemical Ltd | Cephalosporin-derivate, verfahren zu ihrer herstellung und diese enthaltende antimikrobielle mittel |
-
2000
- 2000-09-19 AR ARP000104904A patent/AR029004A1/es not_active Application Discontinuation
- 2000-09-21 RU RU2002110444/04A patent/RU2225868C2/ru not_active IP Right Cessation
- 2000-09-21 MX MXPA02003024A patent/MXPA02003024A/es active IP Right Grant
- 2000-09-21 CN CNB008157464A patent/CN1206231C/zh not_active Expired - Fee Related
- 2000-09-21 HU HU0202663A patent/HUP0202663A3/hu unknown
- 2000-09-21 SK SK412-2002A patent/SK4122002A3/sk unknown
- 2000-09-21 HK HK03100320.8A patent/HK1048121B/en not_active IP Right Cessation
- 2000-09-21 PL PL00354919A patent/PL354919A1/xx not_active Application Discontinuation
- 2000-09-21 BR BR0014230-1A patent/BR0014230A/pt not_active IP Right Cessation
- 2000-09-21 EP EP00966807A patent/EP1222194B1/en not_active Expired - Lifetime
- 2000-09-21 DE DE60020862T patent/DE60020862D1/de not_active Expired - Lifetime
- 2000-09-21 IL IL14866900A patent/IL148669A0/xx active IP Right Grant
- 2000-09-21 JP JP2001524998A patent/JP2003509512A/ja active Pending
- 2000-09-21 WO PCT/US2000/026069 patent/WO2001021623A1/en not_active Ceased
- 2000-09-21 CZ CZ2002993A patent/CZ2002993A3/cs unknown
- 2000-09-21 CA CA002385479A patent/CA2385479A1/en not_active Abandoned
- 2000-09-21 AT AT00966807T patent/ATE297934T1/de not_active IP Right Cessation
- 2000-09-21 NZ NZ517761A patent/NZ517761A/en unknown
- 2000-09-21 AU AU77095/00A patent/AU784077B2/en not_active Ceased
- 2000-09-21 MY MYPI20004413A patent/MY136038A/en unknown
- 2000-09-21 KR KR1020027003755A patent/KR20020068508A/ko not_active Ceased
-
2001
- 2001-03-19 TW TW089119608A patent/TWI283682B/zh not_active IP Right Cessation
-
2002
- 2002-03-13 IL IL148669A patent/IL148669A/en not_active IP Right Cessation
- 2002-03-13 ZA ZA200202065A patent/ZA200202065B/en unknown
- 2002-03-21 NO NO20021416A patent/NO20021416L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| NO20021416L (no) | 2002-05-22 |
| JP2003509512A (ja) | 2003-03-11 |
| SK4122002A3 (en) | 2003-03-04 |
| RU2225868C2 (ru) | 2004-03-20 |
| IL148669A0 (en) | 2002-09-12 |
| HK1048121B (en) | 2005-11-04 |
| CZ2002993A3 (cs) | 2002-07-17 |
| PL354919A1 (en) | 2004-03-22 |
| DE60020862D1 (de) | 2005-07-21 |
| IL148669A (en) | 2006-04-10 |
| CA2385479A1 (en) | 2001-03-29 |
| EP1222194B1 (en) | 2005-06-15 |
| CN1206231C (zh) | 2005-06-15 |
| ATE297934T1 (de) | 2005-07-15 |
| WO2001021623A1 (en) | 2001-03-29 |
| CN1451011A (zh) | 2003-10-22 |
| TWI283682B (en) | 2007-07-11 |
| HUP0202663A2 (hu) | 2002-12-28 |
| NO20021416D0 (no) | 2002-03-21 |
| BR0014230A (pt) | 2002-05-21 |
| ZA200202065B (en) | 2007-11-28 |
| EP1222194A1 (en) | 2002-07-17 |
| HUP0202663A3 (en) | 2003-10-28 |
| HK1048121A1 (en) | 2003-03-21 |
| AU7709500A (en) | 2001-04-24 |
| AU784077B2 (en) | 2006-02-02 |
| AR029004A1 (es) | 2003-06-04 |
| MY136038A (en) | 2008-08-29 |
| KR20020068508A (ko) | 2002-08-27 |
| NZ517761A (en) | 2003-10-31 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant or registration |