MX9709690A - Microdispersiones continuas de fluoroquimicos para el suministro de agentes farmaceuticos. - Google Patents
Microdispersiones continuas de fluoroquimicos para el suministro de agentes farmaceuticos.Info
- Publication number
- MX9709690A MX9709690A MX9709690A MX9709690A MX9709690A MX 9709690 A MX9709690 A MX 9709690A MX 9709690 A MX9709690 A MX 9709690A MX 9709690 A MX9709690 A MX 9709690A MX 9709690 A MX9709690 A MX 9709690A
- Authority
- MX
- Mexico
- Prior art keywords
- pharmaceutical
- pharmaceutical composition
- delivery
- pharmaceutical agents
- microdispersion
- Prior art date
Links
- 239000008177 pharmaceutical agent Substances 0.000 title abstract 3
- 239000008194 pharmaceutical composition Substances 0.000 abstract 5
- 239000007788 liquid Substances 0.000 abstract 2
- 239000006184 cosolvent Substances 0.000 abstract 1
- 239000003085 diluting agent Substances 0.000 abstract 1
- 230000001747 exhibiting effect Effects 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 238000005191 phase separation Methods 0.000 abstract 1
- 239000002904 solvent Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
- A61K9/0026—Blood substitute; Oxygen transporting formulations; Plasma extender
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Dermatology (AREA)
- Hematology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Plant Substances (AREA)
Abstract
Un método para preparar una microdispersion farmacéutica que exhiba biodisponibilidad mejorada, que incluye las siguientes etapas: proporcionar una composicion farmacéutica termodinámicamente estable que comprende al menos un agente farmacéutico incorporado en un portador líquido fisiologicamente aceptable, el portador líquido comprende uno o más solventes lipofílicos, tales como fluoroquímicos, y de preferencia al menos un co-solvente no fluorado, y combinar una composicion farmacéutica estable con una cantidad de al menos un diluyente miscible suficiente para iniciar la separacion de fase del agente farmacéutico a partir de la composicion farmacéutica, en donde se forma una microdispersion de la composicion farmacéutica. También se revelan composiciones farmacéuticas microdispersas, y herramientas para formar dichas composiciones.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US08482176 | 1995-06-07 | ||
| US08/482,176 US5667809A (en) | 1995-06-07 | 1995-06-07 | Continuous fluorochemical microdispersions for the delivery of lipophilic pharmaceutical agents |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| MX9709690A true MX9709690A (es) | 1998-03-29 |
| MXPA97009690A MXPA97009690A (es) | 1998-10-15 |
Family
ID=
Also Published As
| Publication number | Publication date |
|---|---|
| EP0831770B1 (en) | 2000-08-16 |
| DK0831770T3 (da) | 2000-12-18 |
| NO975320D0 (no) | 1997-11-19 |
| AU721759B2 (en) | 2000-07-13 |
| DE69609834T2 (de) | 2000-12-21 |
| GR3034657T3 (en) | 2001-01-31 |
| ATE195415T1 (de) | 2000-09-15 |
| CN1192135A (zh) | 1998-09-02 |
| DE69609834D1 (de) | 2000-09-21 |
| WO1996040053A1 (en) | 1996-12-19 |
| PL323829A1 (en) | 1998-04-27 |
| EP0831770A1 (en) | 1998-04-01 |
| US5667809A (en) | 1997-09-16 |
| ES2150674T3 (es) | 2000-12-01 |
| AU6049496A (en) | 1996-12-30 |
| CA2222081A1 (en) | 1996-12-19 |
| IL122241A0 (en) | 1998-04-05 |
| KR100454377B1 (ko) | 2005-08-04 |
| HUP9900872A2 (hu) | 1999-08-30 |
| NO975320L (no) | 1998-01-27 |
| PT831770E (pt) | 2000-11-30 |
| KR19990022587A (ko) | 1999-03-25 |
| JPH11506783A (ja) | 1999-06-15 |
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