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MX9401080A - Compuestos heteroaromaticos. - Google Patents

Compuestos heteroaromaticos.

Info

Publication number
MX9401080A
MX9401080A MX9401080A MX9401080A MX9401080A MX 9401080 A MX9401080 A MX 9401080A MX 9401080 A MX9401080 A MX 9401080A MX 9401080 A MX9401080 A MX 9401080A MX 9401080 A MX9401080 A MX 9401080A
Authority
MX
Mexico
Prior art keywords
heteroaromatic compounds
piperazine
therapy
processes
preparation
Prior art date
Application number
MX9401080A
Other languages
English (en)
Inventor
Mark Henry Norman
Frank Navas Iii
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of MX9401080A publication Critical patent/MX9401080A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D275/00Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/04Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Psychiatry (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

La presente invención se refiere a un grupo de derivados de piperacina y piperidina, a procedimientos para su preparación, a composiciones farmacéuticas que los contienen, y a su uso en terapia, en particular, en el tratamiento de desórdenes psicóticos.
MX9401080A 1993-02-10 1994-02-10 Compuestos heteroaromaticos. MX9401080A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB939302622A GB9302622D0 (en) 1993-02-10 1993-02-10 Heteroaromatic compounds

Publications (1)

Publication Number Publication Date
MX9401080A true MX9401080A (es) 1994-08-31

Family

ID=10730183

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9401080A MX9401080A (es) 1993-02-10 1994-02-10 Compuestos heteroaromaticos.

Country Status (15)

Country Link
EP (1) EP0683778A1 (es)
JP (1) JPH08506337A (es)
CN (1) CN1117731A (es)
AU (1) AU6005194A (es)
BG (1) BG99839A (es)
CA (1) CA2155758A1 (es)
CZ (1) CZ204495A3 (es)
FI (1) FI953777A0 (es)
GB (1) GB9302622D0 (es)
HU (1) HUT73654A (es)
IL (1) IL108601A0 (es)
MX (1) MX9401080A (es)
SK (1) SK99195A3 (es)
WO (1) WO1994018196A1 (es)
ZA (1) ZA94891B (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5364866A (en) 1989-05-19 1994-11-15 Hoechst-Roussel Pharmaceuticals, Inc. Heteroarylpiperidines, pyrrolidines and piperazines and their use as antipsychotics and analetics
US5776963A (en) 1989-05-19 1998-07-07 Hoechst Marion Roussel, Inc. 3-(heteroaryl)-1- (2,3-dihydro-1h-isoindol-2-yl)alkyl!pyrrolidines and 3-(heteroaryl)-1- (2,3-dihydro-1h-indol-1-yl)alkyl!pyrrolidines and related compounds and their therapeutic untility
GB9420521D0 (en) * 1994-10-12 1994-11-30 Smithkline Beecham Plc Novel compounds
JP3274579B2 (ja) * 1995-01-12 2002-04-15 住友製薬株式会社 脳血管障害に伴う精神症候治療剤
DE69618050T2 (de) * 1995-03-17 2002-07-11 Aventis Pharmaceuticals Inc., Cincinnati Substituierte Benzylthienylpiperazine, ihre Anwendung als Arzneimittel und Verfahren für ihre Herstellung
UA73981C2 (en) 2000-03-10 2005-10-17 Merck Patent Gmbh (r)-(-)-2-[5-(4-fluorophenyl)-3-pyridylmethylaminomethyl]-chromane for treatment of extrapyramidal movement disorders (variants), pharmaceutical composition and kit
US20040014788A1 (en) * 2000-11-14 2004-01-22 Gerd Bartoszyk Novel uses of combined selective dopamine d2 receptor antagonists and 5-ht receptor agonists
WO2002066469A2 (en) * 2001-02-16 2002-08-29 Aventis Pharmaceuticals Inc. Novel heterocyclic amide derivatives and their use as dopamine d3 receptor ligands
ATE352302T1 (de) 2001-07-26 2007-02-15 Merck Patent Gmbh Verwendung von 2- 5-(4-fluorphenyl)-3- pyridylmethylaminomethyl-chroman und seiner physiologisch annehmbaren salze
GB0222912D0 (en) 2002-10-03 2002-11-13 Astrazeneca Ab Novel process and intermediates
GB0222909D0 (en) 2002-10-03 2002-11-13 Astrazeneca Ab Novel process and intermediates
RU2403247C2 (ru) * 2004-07-20 2010-11-10 СЬЕНА БИОТЕК С.п.А. Модуляторы никотиновых ацетилхолиновых рецепторов альфа 7 и их терапевтические применения
CL2008000119A1 (es) 2007-01-16 2008-05-16 Wyeth Corp Compuestos derivados de pirazol, antagonistas del receptor nicotinico de acetilcolina; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como demencia senil, alzheimer y esquizofrenia.
US8981095B2 (en) 2011-07-28 2015-03-17 Mapi Pharma Ltd. Intermediate compounds and process for the preparation of lurasidone and salts thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0625181B2 (ja) * 1985-03-27 1994-04-06 住友製薬株式会社 新規なイミド誘導体
JP2660407B2 (ja) * 1986-09-26 1997-10-08 住友製薬株式会社 新規なイミド誘導体
US5143923B1 (en) * 1991-04-29 1993-11-02 Hoechst-Roussel Pharmaceuticals Incorporated Benzoisothiazole-and benzisoxazole-3-carboxamides
MX9201991A (es) * 1991-05-02 1992-11-01 Jonh Wyeth & Brother Limited Derivados de piperazina y procedimiento para su preparacion.

Also Published As

Publication number Publication date
HU9501881D0 (en) 1995-08-28
BG99839A (bg) 1996-02-28
CA2155758A1 (en) 1994-08-18
FI953777A7 (fi) 1995-08-09
FI953777A0 (fi) 1995-08-09
ZA94891B (en) 1995-08-10
CN1117731A (zh) 1996-02-28
CZ204495A3 (en) 1996-03-13
HUT73654A (en) 1996-09-30
JPH08506337A (ja) 1996-07-09
WO1994018196A1 (en) 1994-08-18
AU6005194A (en) 1994-08-29
IL108601A0 (en) 1994-05-30
GB9302622D0 (en) 1993-03-24
EP0683778A1 (en) 1995-11-29
SK99195A3 (en) 1995-12-06

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