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MX9300779A - 3- (1H-TETRAZOLE-5-Y1) -4H-PYRIDO [1,2-A] PIRIMIDINA-4-ONAS PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM AND THEIR PREPARATION THEREOF - Google Patents

3- (1H-TETRAZOLE-5-Y1) -4H-PYRIDO [1,2-A] PIRIMIDINA-4-ONAS PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM AND THEIR PREPARATION THEREOF

Info

Publication number
MX9300779A
MX9300779A MX9300779A MX9300779A MX9300779A MX 9300779 A MX9300779 A MX 9300779A MX 9300779 A MX9300779 A MX 9300779A MX 9300779 A MX9300779 A MX 9300779A MX 9300779 A MX9300779 A MX 9300779A
Authority
MX
Mexico
Prior art keywords
pyrido
preparation
pirimidina
onas
tetrazole
Prior art date
Application number
MX9300779A
Other languages
Spanish (es)
Inventor
Istvan Hermecz
Judit Sipos
Lelle Vasvari-Nee-Debreczy
Zoltan Kapui
Agnes Horvath
Maria Balogh
Geza Kereszturi
Kinga Boer
Aniko Pajor
Original Assignee
Chinoin Gyogyszer Es Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer Es Vegyeszet filed Critical Chinoin Gyogyszer Es Vegyeszet
Publication of MX9300779A publication Critical patent/MX9300779A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La invención se relaciona con 3-(1H-tetrazol-5-il)-4H-pirido[1,2-a]pirimidin-4-o nas parcialmente nuevas de la fórmula general (I) y sales/o hidratos farmacéuticamente aceptables y con la preparación de las mismas. Estos compuestos poseen actividad antialérgica o antiulcerante significativa.The invention relates to partially new 3- (1H-tetrazol-5-yl) -4H-pyrido [1,2-a] pyrimidin-4-o nas of the general formula (I) and pharmaceutically acceptable salts / hydrates and with the preparation of the same. These compounds possess significant antiallergic or anti-ulcer activity.

MX9300779A 1992-02-13 1993-02-12 3- (1H-TETRAZOLE-5-Y1) -4H-PYRIDO [1,2-A] PIRIMIDINA-4-ONAS PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM AND THEIR PREPARATION THEREOF MX9300779A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU9200432A HUT64064A (en) 1992-02-13 1992-02-13 Process for producing puyrido/1,2-a/pyrimidine derivatives and pharmaceutical compositions comprising same as active ingredient

Publications (1)

Publication Number Publication Date
MX9300779A true MX9300779A (en) 1993-09-30

Family

ID=10981335

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9300779A MX9300779A (en) 1992-02-13 1993-02-12 3- (1H-TETRAZOLE-5-Y1) -4H-PYRIDO [1,2-A] PIRIMIDINA-4-ONAS PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM AND THEIR PREPARATION THEREOF

Country Status (7)

Country Link
CN (1) CN1080289A (en)
AU (1) AU3573793A (en)
HU (1) HUT64064A (en)
IL (1) IL104706A0 (en)
MX (1) MX9300779A (en)
SI (1) SI9300075A (en)
WO (1) WO1993016076A1 (en)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU209793B (en) * 1990-09-25 1994-11-28 Chinoin Gyogyszer Es Vegyeszet Process for the production of pyrido[1,2-a]pyrimidine-derivatives and pharmaceutical compositions containing the same
ITMI20011764A1 (en) * 2001-08-10 2003-02-10 Dinamite Dipharma Spa HIGH PURITY PEMIROLAST METHOD
JP4690043B2 (en) * 2002-10-04 2011-06-01 プラナ バイオテクノロジー リミティッド Nerve active compounds
WO2007093184A2 (en) * 2006-02-13 2007-08-23 Astion Pharma A/S Treatment of mmp-mediated dermatological diseases with pemirolast
EP1818058A3 (en) * 2006-02-13 2007-11-07 Astion Pharma A/S Treatment of mmp-mediated dermatological diseases with pemirolast
CN104945420A (en) 2009-06-29 2015-09-30 因塞特公司 Pyrimidinones as PI3K inhibitors
US8759359B2 (en) 2009-12-18 2014-06-24 Incyte Corporation Substituted heteroaryl fused derivatives as PI3K inhibitors
JP5816678B2 (en) 2010-04-14 2015-11-18 インサイト・コーポレイションＩｎｃｙｔｅ Ｃｏｒｐｏｒａｔｉｏｎ Condensed derivatives as PI3Kδ inhibitors
US9062055B2 (en) 2010-06-21 2015-06-23 Incyte Corporation Fused pyrrole derivatives as PI3K inhibitors
CA2822070C (en) 2010-12-20 2019-09-17 Incyte Corporation N-(1-(substituted-phenyl)ethyl)-9h-purin-6-amines as pi3k inhibitors
US9108984B2 (en) 2011-03-14 2015-08-18 Incyte Corporation Substituted diamino-pyrimidine and diamino-pyridine derivatives as PI3K inhibitors
WO2012135009A1 (en) 2011-03-25 2012-10-04 Incyte Corporation Pyrimidine-4,6-diamine derivatives as pi3k inhibitors
ES2873001T3 (en) 2011-09-02 2021-11-03 Incyte Holdings Corp Heterocyclamines as PI3K inhibitors
AR090548A1 (en) 2012-04-02 2014-11-19 Incyte Corp BICYCLIC AZAHETEROCICLOBENCILAMINS AS PI3K INHIBITORS
WO2015191677A1 (en) 2014-06-11 2015-12-17 Incyte Corporation Bicyclic heteroarylaminoalkyl phenyl derivatives as pi3k inhibitors
JP6816005B2 (en) 2015-02-27 2021-01-20 インサイト・コーポレイションＩｎｃｙｔｅ Ｃｏｒｐｏｒａｔｉｏｎ Salts of PI3K inhibitors and processes for their preparation
US9988401B2 (en) 2015-05-11 2018-06-05 Incyte Corporation Crystalline forms of a PI3K inhibitor
WO2016183060A1 (en) 2015-05-11 2016-11-17 Incyte Corporation Process for the synthesis of a phosphoinositide 3-kinase inhibitor
MA52761A (en) 2018-06-01 2021-04-14 Incyte Corp DOSAGE REGIMEN FOR THE TREATMENT OF PI3K-RELATED DISORDERS

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2044796C (en) * 1990-06-21 2001-10-16 Atsunori Sano Process for producing pyrido[1,2-a] pyrimidine derivative

Also Published As

Publication number Publication date
HU9200432D0 (en) 1992-04-28
AU3573793A (en) 1993-09-03
HUT64064A (en) 1993-11-29
WO1993016076A1 (en) 1993-08-19
SI9300075A (en) 1993-09-30
CN1080289A (en) 1994-01-05
IL104706A0 (en) 1993-06-10

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