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MX2021003681A - Composiciones y metodos para el tratamiento de desordenes inflamatorios. - Google Patents

Composiciones y metodos para el tratamiento de desordenes inflamatorios.

Info

Publication number
MX2021003681A
MX2021003681A MX2021003681A MX2021003681A MX2021003681A MX 2021003681 A MX2021003681 A MX 2021003681A MX 2021003681 A MX2021003681 A MX 2021003681A MX 2021003681 A MX2021003681 A MX 2021003681A MX 2021003681 A MX2021003681 A MX 2021003681A
Authority
MX
Mexico
Prior art keywords
treatment
inflammatory disorders
benzimidazole derivative
patient
compound
Prior art date
Application number
MX2021003681A
Other languages
English (en)
Inventor
Hariharan Venkatesan
Michael Rabinowitz
Mark D Rosen
Original Assignee
Akebia Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akebia Therapeutics Inc filed Critical Akebia Therapeutics Inc
Publication of MX2021003681A publication Critical patent/MX2021003681A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41841,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Se proporcionan aquí métodos de tratamiento y prevención del padecimiento inflamatorio del intestino en un paciente. Los métodos aquí provistos comprenden administrar al paciente que lo necesite una cantidad efectiva de un compuesto de benzoimidazol, Compuesto 1, para tratar o prevenir un padecimiento inflamatorio del intestino en un paciente. También se proporcionan formulaciones y rutas de administración del compuesto.
MX2021003681A 2018-10-03 2019-10-02 Composiciones y metodos para el tratamiento de desordenes inflamatorios. MX2021003681A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201862740748P 2018-10-03 2018-10-03
PCT/US2019/054293 WO2020072645A1 (en) 2018-10-03 2019-10-02 Benzimidazole derivative for use in the treatment of inflammatory disorders

Publications (1)

Publication Number Publication Date
MX2021003681A true MX2021003681A (es) 2021-08-19

Family

ID=68468802

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2021003681A MX2021003681A (es) 2018-10-03 2019-10-02 Composiciones y metodos para el tratamiento de desordenes inflamatorios.

Country Status (11)

Country Link
US (1) US20210369678A1 (es)
EP (1) EP3860593A1 (es)
JP (1) JP2022504293A (es)
KR (1) KR20210100594A (es)
CN (1) CN113382729A (es)
AU (1) AU2019355097A1 (es)
CA (1) CA3114592A1 (es)
MX (1) MX2021003681A (es)
SG (1) SG11202103191QA (es)
TW (1) TW202027745A (es)
WO (1) WO2020072645A1 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY204336A (en) 2013-06-13 2024-08-23 Akebia Therapeutics Inc Compositions and methods for treating anemia
EP4138825A1 (en) 2020-04-20 2023-03-01 Akebia Therapeutics Inc. Treatment of viral infections, of organ injury, and of related conditions using a hif prolyl hydroxylase inhibitor or a hif-alpha stabilizer
WO2022150623A1 (en) 2021-01-08 2022-07-14 Akebia Therapeutics, Inc. Compounds and composition for the treatment of anemia
WO2022251563A1 (en) 2021-05-27 2022-12-01 Keryx Biopharmaceuticals, Inc. Pediatric formulations of ferric citrate
KR102729791B1 (ko) 2022-04-13 2024-11-14 재단법인 대구경북첨단의료산업진흥재단 아릴에텐 유도체를 유효성분으로 포함하는 염증성 장질환 치료용 조성물

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101390144B1 (ko) * 2006-04-13 2014-04-28 다이호야쿠힌고교 가부시키가이샤 염증성 장질환 치료제
PT2294066E (pt) * 2008-04-28 2014-11-21 Janssen Pharmaceutica Nv Benzoimidazoles como inibidores da prolil-hidroxilase
MA40406A (fr) * 2014-07-28 2016-02-04 Nogra Pharma Ltd Procédés et compositions de diagnostic et de traitement des maladies inflammatoires chroniques de l'intestin

Also Published As

Publication number Publication date
US20210369678A1 (en) 2021-12-02
EP3860593A1 (en) 2021-08-11
KR20210100594A (ko) 2021-08-17
AU2019355097A1 (en) 2021-05-27
CN113382729A (zh) 2021-09-10
JP2022504293A (ja) 2022-01-13
SG11202103191QA (en) 2021-04-29
TW202027745A (zh) 2020-08-01
WO2020072645A1 (en) 2020-04-09
CA3114592A1 (en) 2020-04-09

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