MX2019006721A - Tratamiento para la colangitis biliar primaria. - Google Patents
Tratamiento para la colangitis biliar primaria.Info
- Publication number
- MX2019006721A MX2019006721A MX2019006721A MX2019006721A MX2019006721A MX 2019006721 A MX2019006721 A MX 2019006721A MX 2019006721 A MX2019006721 A MX 2019006721A MX 2019006721 A MX2019006721 A MX 2019006721A MX 2019006721 A MX2019006721 A MX 2019006721A
- Authority
- MX
- Mexico
- Prior art keywords
- treatment
- primary bile
- cholangitis
- pbc
- bile cholangitis
- Prior art date
Links
- 210000000941 bile Anatomy 0.000 title 1
- 208000003167 cholangitis Diseases 0.000 title 1
- 208000008439 Biliary Liver Cirrhosis Diseases 0.000 abstract 3
- 208000012654 Primary biliary cholangitis Diseases 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/575—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Gastroenterology & Hepatology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
La presente invención proporciona un compuesto terapéutico para la prevención y el tratamiento de la colangitis biliar primaria (PBC). De manera específica, la presente invención proporciona una composición farmacéutica que comprende un compuesto de la Formula (I) o una sal farmacéuticamente aceptable del mismo, para el tratamiento de la PBC. (Ver Fórmula).
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN201621042122 | 2016-12-09 | ||
| PCT/IB2017/057746 WO2018104916A1 (en) | 2016-12-09 | 2017-12-08 | Treatment for primary biliary cholangitis |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| MX2019006721A true MX2019006721A (es) | 2019-10-30 |
| MX382765B MX382765B (es) | 2025-03-13 |
Family
ID=60957351
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2019006721A MX382765B (es) | 2016-12-09 | 2017-12-08 | Tratamiento para la colangitis biliar primaria. |
Country Status (8)
| Country | Link |
|---|---|
| US (7) | US20180243263A1 (es) |
| EP (1) | EP3551180B1 (es) |
| JP (1) | JP6840853B2 (es) |
| BR (1) | BR112019011740A2 (es) |
| ES (1) | ES2894261T3 (es) |
| MX (1) | MX382765B (es) |
| WO (1) | WO2018104916A1 (es) |
| ZA (1) | ZA201903649B (es) |
Families Citing this family (9)
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| CA2606499C (en) | 2005-05-26 | 2017-06-13 | Metabasis Therapeutics, Inc. | Thyromimetics for the treatment of fatty liver diseases |
| WO2018094265A2 (en) | 2016-11-21 | 2018-05-24 | Viking Therapeutics, Inc. | Method of treating glycogen storage disease |
| WO2018104916A1 (en) * | 2016-12-09 | 2018-06-14 | Cadila Healthcare Limited | Treatment for primary biliary cholangitis |
| CN110996966A (zh) | 2017-06-05 | 2020-04-10 | 维京治疗公司 | 用于治疗纤维化的组合物 |
| KR20200138283A (ko) | 2018-03-22 | 2020-12-09 | 바이킹 테라퓨틱스 인코포레이티드 | 결정질 형태, 및 결정질 형태의 화합물을 제조하는 방법 |
| CN110934866B (zh) * | 2018-09-25 | 2023-12-01 | 深圳微芯生物科技股份有限公司 | 西格列羧及其相关化合物的应用 |
| WO2020117962A1 (en) * | 2018-12-05 | 2020-06-11 | Viking Therapeutics, Inc. | Compositions for the treatment of fibrosis and inflammation |
| WO2022040110A2 (en) * | 2020-08-18 | 2022-02-24 | Sheng Liu | Alkylating agent and combinations in the treatment of immune-related and liver diseases, alzheimer's diseases and fibrosis diseases |
| WO2022180612A1 (en) * | 2021-02-26 | 2022-09-01 | Cadila Healthcare Limited | Orodispersible formulation of hypolipidemic agent |
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| WO2018104916A1 (en) * | 2016-12-09 | 2018-06-14 | Cadila Healthcare Limited | Treatment for primary biliary cholangitis |
-
2017
- 2017-12-08 WO PCT/IB2017/057746 patent/WO2018104916A1/en not_active Ceased
- 2017-12-08 MX MX2019006721A patent/MX382765B/es unknown
- 2017-12-08 BR BR112019011740-7A patent/BR112019011740A2/pt not_active Application Discontinuation
- 2017-12-08 ES ES17829016T patent/ES2894261T3/es active Active
- 2017-12-08 EP EP17829016.9A patent/EP3551180B1/en active Active
- 2017-12-08 US US15/835,938 patent/US20180243263A1/en not_active Abandoned
- 2017-12-08 JP JP2019530797A patent/JP6840853B2/ja active Active
-
2019
- 2019-06-07 ZA ZA2019/03649A patent/ZA201903649B/en unknown
-
2020
- 2020-07-02 US US16/919,404 patent/US20210085644A1/en not_active Abandoned
-
2021
- 2021-01-13 US US17/147,829 patent/US20210128525A1/en active Granted
- 2021-10-28 US US17/512,950 patent/US11433050B2/en active Active
-
2022
- 2022-08-04 US US17/880,949 patent/US12178799B2/en active Active
-
2023
- 2023-04-14 US US18/300,668 patent/US11872209B2/en active Active
-
2024
- 2024-10-22 US US18/922,676 patent/US20250041269A1/en active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| US20250041269A1 (en) | 2025-02-06 |
| US11433050B2 (en) | 2022-09-06 |
| US12178799B2 (en) | 2024-12-31 |
| JP6840853B2 (ja) | 2021-03-10 |
| EP3551180B1 (en) | 2021-09-29 |
| WO2018104916A1 (en) | 2018-06-14 |
| US20220062231A1 (en) | 2022-03-03 |
| US20210128525A1 (en) | 2021-05-06 |
| US20180243263A1 (en) | 2018-08-30 |
| ES2894261T3 (es) | 2022-02-14 |
| US11872209B2 (en) | 2024-01-16 |
| US20230255932A1 (en) | 2023-08-17 |
| US20210085644A1 (en) | 2021-03-25 |
| EP3551180A1 (en) | 2019-10-16 |
| ZA201903649B (en) | 2021-01-27 |
| JP2020502095A (ja) | 2020-01-23 |
| BR112019011740A2 (pt) | 2019-10-29 |
| MX382765B (es) | 2025-03-13 |
| US20230201162A1 (en) | 2023-06-29 |
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