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MX2018001380A - Agonistas del receptor 5-ht2c y composiciones y metodos de uso. - Google Patents

Agonistas del receptor 5-ht2c y composiciones y metodos de uso.

Info

Publication number
MX2018001380A
MX2018001380A MX2018001380A MX2018001380A MX2018001380A MX 2018001380 A MX2018001380 A MX 2018001380A MX 2018001380 A MX2018001380 A MX 2018001380A MX 2018001380 A MX2018001380 A MX 2018001380A MX 2018001380 A MX2018001380 A MX 2018001380A
Authority
MX
Mexico
Prior art keywords
disorders
sleep
disease
antipsychotic
methods
Prior art date
Application number
MX2018001380A
Other languages
English (en)
Other versions
MX375045B (es
Inventor
S Ren Albert
Semple Graeme
Lehmann Juerg
Feichtinger Konrad
Original Assignee
Arena Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Arena Pharm Inc filed Critical Arena Pharm Inc
Publication of MX2018001380A publication Critical patent/MX2018001380A/es
Publication of MX375045B publication Critical patent/MX375045B/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/32Alcohol-abuse
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D223/00Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/14Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D223/16Benzazepines; Hydrogenated benzazepines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D223/00Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/14Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D223/32Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems containing carbocyclic rings other than six-membered
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • C07D491/044Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
    • C07D491/052Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being six-membered
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/06Peri-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2121/00Preparations for use in therapy

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Diabetes (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Addiction (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)

Abstract

En algunas modalidades se proveen compuestos de la Fórmula A, tal como se define en la presente solicitud, que modulan la actividad del receptor 5-HT2C. En algunas modalidades también se proveen métodos, tales como, para control de peso, inducir saciedad, y disminuir la ingesta de alimentos, y para prevenir y tratar obesidad, aumento de peso inducido por antipsicótico, diabetes tipo 2, síndrome de Prader-Willi, dependencia del tabaco/nicotina, drogadicción, alcoholismo, juego patológico, síndrome de deficiencia de recompensa, y adicción al sexo, trastornos del espectro obsesivo-compulsivo y trastornos del control de los impulsos (incluyendo el hábito de morderse las uñas y onicofagia), trastornos del sueño (incluyendo insomnio, arquitectura del sueño fragmentada, y alteraciones del sueño de onda lenta), incontinencia urinaria, trastornos psiquiátricos (incluyendo esquizofrenia, anorexia nerviosa, y bulimia nerviosa), enfermedad de Alzheimer, disfunción sexual, disfunción eréctil, epilepsia, trastornos del movimiento (incluyendo parkinsonismo y trastorno del movimiento inducido por antipsicótico), hipertensión, dislipidemia, enfermedad de hígado graso no alcohólica, enfermedad renal relacionada con la obesidad, y apnea del sueño.
MX2018001380A 2015-07-31 2016-07-28 Agonistas del receptor 5-ht2c y composiciones y metodos de uso. MX375045B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201562199382P 2015-07-31 2015-07-31
PCT/US2016/044426 WO2017023679A1 (en) 2015-07-31 2016-07-28 5-ht2c receptor agonists and compositions and methods of use

Publications (2)

Publication Number Publication Date
MX2018001380A true MX2018001380A (es) 2018-06-15
MX375045B MX375045B (es) 2025-03-06

Family

ID=56684262

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2018001380A MX375045B (es) 2015-07-31 2016-07-28 Agonistas del receptor 5-ht2c y composiciones y metodos de uso.

Country Status (14)

Country Link
US (4) US10272094B2 (es)
EP (1) EP3328835B1 (es)
JP (1) JP6789578B2 (es)
KR (1) KR20180031035A (es)
CN (1) CN108137508B (es)
AU (1) AU2016302755B2 (es)
BR (1) BR112018001707A2 (es)
CA (1) CA3002525A1 (es)
EA (1) EA039412B1 (es)
HK (1) HK1255850A1 (es)
IL (1) IL257107B (es)
MA (1) MA42527A (es)
MX (1) MX375045B (es)
WO (1) WO2017023679A1 (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2017023679A1 (en) * 2015-07-31 2017-02-09 Arena Pharmaceuticals, Inc. 5-ht2c receptor agonists and compositions and methods of use
US12459965B2 (en) 2017-10-09 2025-11-04 Compass Pathfinder Limited Preparation of psilocybin, different polymorphic forms, intermediates, formulations and their use
GB2571696B (en) 2017-10-09 2020-05-27 Compass Pathways Ltd Large scale method for the preparation of Psilocybin and formulations of Psilocybin so produced
EP3733204A4 (en) 2017-12-27 2021-09-15 Takeda Pharmaceutical Company Limited THERAPEUTIC AGENT FOR URINARY INCONTINENCE OF STRESS AND FECAL INCONTINENCE
US20210393621A1 (en) 2018-10-26 2021-12-23 The Research Foundation For The State University Of New York Combination serotonin specific reuptake inhibitor and serotonin 1a receptor partial agonist for reducing l-dopa-induced dyskinesia
CN110642721B (zh) * 2018-12-21 2022-09-30 安徽贝克生物制药有限公司 盐酸司来吉兰的制备方法
CN110668951B (zh) * 2018-12-21 2022-09-30 安徽贝克生物制药有限公司 一种盐酸司来吉兰的合成工艺
CN113993523A (zh) 2019-04-17 2022-01-28 指南针探路者有限公司 用赛洛西宾治疗抑郁症和其他各种病症
WO2023279012A2 (en) * 2021-06-29 2023-01-05 Tusimple, Inc. Systems and methods for operating an autonomous vehicle
EP4416027A1 (en) 2021-10-14 2024-08-21 Tusimple, Inc. Systems and methods for operating an autonomous vehicle

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5180733A (en) * 1990-03-30 1993-01-19 Abbott Laboratories Biogenic amine uptake inhibitors
AU1919592A (en) 1991-04-16 1992-11-17 National Institutes Of Health Method of treating trichotillomania and onychophagia
US6953787B2 (en) * 2002-04-12 2005-10-11 Arena Pharmaceuticals, Inc. 5HT2C receptor modulators
CA2482195A1 (en) 2002-04-12 2003-10-23 The University Of Chicago Farnesoid x-activated receptor agonists
TW200307682A (en) * 2002-04-25 2003-12-16 Wyeth Corp 1,2,3,4,7,8-Hexahydro-6H-[1,4]diazepino[6,7,1-ij]quinoline derivatives as antipsychotic and antiobesity agents
CN1805938B (zh) * 2003-06-17 2010-06-16 艾尼纳制药公司 用于治疗5ht2c受体相关疾病的苯并氮杂卓衍生物
ES2332051T3 (es) * 2003-10-08 2010-01-25 Eli Lilly And Company Compuestos y procedimientos para tratar dislipidemia.
EP2510949A4 (en) * 2009-12-11 2013-11-13 Astellas Pharma Inc THERAPEUTICS FOR FIBROMYALGIA
JP6198715B2 (ja) * 2012-03-06 2017-09-20 武田薬品工業株式会社 三環性化合物
BR112015005743A2 (pt) * 2012-09-14 2017-07-04 Abbvie Deutschland derivados tricíclicos de quinoxalina e quinolina
WO2017023679A1 (en) 2015-07-31 2017-02-09 Arena Pharmaceuticals, Inc. 5-ht2c receptor agonists and compositions and methods of use

Also Published As

Publication number Publication date
JP2018522025A (ja) 2018-08-09
WO2017023679A1 (en) 2017-02-09
NZ739883A (en) 2021-03-26
US20180214455A1 (en) 2018-08-02
JP6789578B2 (ja) 2020-11-25
CN108137508A (zh) 2018-06-08
HK1255850A1 (zh) 2019-08-30
AU2016302755B2 (en) 2020-09-10
EA039412B1 (ru) 2022-01-25
IL257107B (en) 2021-03-25
US10624900B2 (en) 2020-04-21
CA3002525A1 (en) 2017-02-09
US11395824B2 (en) 2022-07-26
US20200078368A1 (en) 2020-03-12
MA42527A (fr) 2021-04-07
IL257107A (en) 2018-03-29
EP3328835A1 (en) 2018-06-06
EA201890402A1 (ru) 2018-09-28
KR20180031035A (ko) 2018-03-27
AU2016302755A1 (en) 2018-03-15
CN108137508B (zh) 2021-08-27
US20200383993A1 (en) 2020-12-10
MX375045B (es) 2025-03-06
EP3328835B1 (en) 2022-10-12
US10272094B2 (en) 2019-04-30
BR112018001707A2 (pt) 2018-09-18
US20230055376A1 (en) 2023-02-23

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