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MX2017008715A - Derivados de glucagon. - Google Patents

Derivados de glucagon.

Info

Publication number
MX2017008715A
MX2017008715A MX2017008715A MX2017008715A MX2017008715A MX 2017008715 A MX2017008715 A MX 2017008715A MX 2017008715 A MX2017008715 A MX 2017008715A MX 2017008715 A MX2017008715 A MX 2017008715A MX 2017008715 A MX2017008715 A MX 2017008715A
Authority
MX
Mexico
Prior art keywords
glucagon
peptide
present
treating obesity
receptors
Prior art date
Application number
MX2017008715A
Other languages
English (en)
Other versions
MX389593B (es
Inventor
Chang Ki Lim
Se Chang Kwon
Sung Youb Jung
Jae Hyuk Choi
Jin Park Young
Suk Lee Jong
Original Assignee
Hanmi Pharm Ind Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hanmi Pharm Ind Co Ltd filed Critical Hanmi Pharm Ind Co Ltd
Publication of MX2017008715A publication Critical patent/MX2017008715A/es
Publication of MX389593B publication Critical patent/MX389593B/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/605—Glucagons
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/26—Glucagons
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Endocrinology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Zoology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Toxicology (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Immunology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invención se refiere a un nuevo péptido de un derivado de glucagón y una composición para prevenir o tratar la obesidad que comprende el péptido como un ingrediente activo; el derivado de glucagón de acuerdo con la presente invención muestra un efecto de activación más excelente con respecto tanto a receptores del péptido 1 similar a glucagón como receptores de glucagón en comparación con el glucagón nativo, y por lo tanto se puede usar ampliamente como un agente efectivo para el tratamiento de la obesidad.
MX2017008715A 2014-12-30 2015-12-30 Derivados de glucagon. MX389593B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
KR1020140193691A KR102418477B1 (ko) 2014-12-30 2014-12-30 글루카곤 유도체
PCT/KR2015/014481 WO2016108617A1 (en) 2014-12-30 2015-12-30 Glucagon derivatives

Publications (2)

Publication Number Publication Date
MX2017008715A true MX2017008715A (es) 2017-11-17
MX389593B MX389593B (es) 2025-03-20

Family

ID=56284668

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2017008715A MX389593B (es) 2014-12-30 2015-12-30 Derivados de glucagon.

Country Status (18)

Country Link
US (3) US10513550B2 (es)
EP (1) EP3240802B1 (es)
JP (1) JP6758297B2 (es)
KR (1) KR102418477B1 (es)
CN (1) CN107250155B (es)
AR (1) AR103323A1 (es)
AU (1) AU2015372767B2 (es)
BR (1) BR112017013845A2 (es)
CA (1) CA2972001C (es)
EA (1) EA036479B1 (es)
IL (1) IL253001B (es)
MX (1) MX389593B (es)
PH (1) PH12017501205A1 (es)
SG (2) SG11201705130XA (es)
TW (1) TWI696631B (es)
UA (1) UA122967C2 (es)
WO (1) WO2016108617A1 (es)
ZA (1) ZA201704328B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
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JP2025526148A (ja) 2022-08-18 2025-08-07 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 長時間作用型ｇｌｐ－１／グルカゴン受容体アゴニスト及びｎｐｙ２受容体アゴニストを含む組合せ治療

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Also Published As

Publication number Publication date
US20200140515A1 (en) 2020-05-07
IL253001A0 (en) 2017-08-31
MX389593B (es) 2025-03-20
UA122967C2 (uk) 2021-01-27
US10513550B2 (en) 2019-12-24
ZA201704328B (en) 2021-01-27
WO2016108617A1 (en) 2016-07-07
BR112017013845A2 (pt) 2018-01-02
AU2015372767A1 (en) 2017-07-13
EP3240802A4 (en) 2018-10-10
US12018060B2 (en) 2024-06-25
EP3240802A1 (en) 2017-11-08
KR20160082026A (ko) 2016-07-08
US20180002395A1 (en) 2018-01-04
HK1246323A1 (en) 2018-09-07
NZ771617A (en) 2024-09-27
CA2972001A1 (en) 2016-07-07
EP3240802B1 (en) 2021-07-21
KR102418477B1 (ko) 2022-07-08
JP6758297B2 (ja) 2020-09-23
US20220025012A1 (en) 2022-01-27
CN107250155B (zh) 2021-08-10
PH12017501205A1 (en) 2017-10-18
US11254724B2 (en) 2022-02-22
AR103323A1 (es) 2017-05-03
EA036479B1 (ru) 2020-11-16
CA2972001C (en) 2024-07-02
TW201632546A (zh) 2016-09-16
JP2018505153A (ja) 2018-02-22
IL253001B (en) 2022-04-01
SG10201906912VA (en) 2019-09-27
EA201791498A1 (ru) 2017-10-31
NZ733649A (en) 2024-07-26
SG11201705130XA (en) 2017-07-28
CN107250155A (zh) 2017-10-13
TWI696631B (zh) 2020-06-21
AU2015372767B2 (en) 2020-07-16

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