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MX2017002670A - Inhibidores de glucosidasa. - Google Patents

Inhibidores de glucosidasa.

Info

Publication number
MX2017002670A
MX2017002670A MX2017002670A MX2017002670A MX2017002670A MX 2017002670 A MX2017002670 A MX 2017002670A MX 2017002670 A MX2017002670 A MX 2017002670A MX 2017002670 A MX2017002670 A MX 2017002670A MX 2017002670 A MX2017002670 A MX 2017002670A
Authority
MX
Mexico
Prior art keywords
glycosidase inhibitors
formula
glycosidase
inhibitors
tautopathies
Prior art date
Application number
MX2017002670A
Other languages
English (en)
Other versions
MX381417B (es
Inventor
S Kulkarni Santosh
Gajendra Giri Awadut
Quattropani Anna
Original Assignee
Asceneuron Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=54065334&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2017002670(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Asceneuron Sa filed Critical Asceneuron Sa
Publication of MX2017002670A publication Critical patent/MX2017002670A/es
Publication of MX381417B publication Critical patent/MX381417B/es

Links

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Compuestos de la fórmula (I) en donde A, R, W, Q, n y m tienen el significado de acuerdo con las reivindicaciones se pueden emplear, entre otros para el tratamiento de tautopatías y enfermedad de Alzheimer (ver Fórmula).
MX2017002670A 2014-08-28 2015-08-27 Inhibidores de glucosidasa. MX381417B (es)

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PCT/EP2015/069598 WO2016030443A1 (en) 2014-08-28 2015-08-27 Glycosidase inhibitors

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IL250642B (en) 2020-07-30
IL250642A0 (en) 2017-04-30
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AU2015308437A1 (en) 2017-03-16
CA2958966A1 (en) 2016-03-03
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CN107108601B (zh) 2021-08-20
US20190367533A1 (en) 2019-12-05
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JP6563017B2 (ja) 2019-08-21
BR112017003658B1 (pt) 2022-12-06
EP3186243A1 (en) 2017-07-05
WO2016030443A1 (en) 2016-03-03
AU2019200339B2 (en) 2019-12-19
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EP3868752A1 (en) 2021-08-25
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AU2019200339A1 (en) 2019-02-07
US10336775B2 (en) 2019-07-02
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EA201790271A1 (ru) 2017-08-31
MA40532A (fr) 2021-04-28
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US12187741B2 (en) 2025-01-07
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ES2893289T3 (es) 2022-02-08
MA53944A (fr) 2021-08-25
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