MX2016002198A - Proceso para la preparación de un compuesto. - Google Patents
Proceso para la preparación de un compuesto.Info
- Publication number
- MX2016002198A MX2016002198A MX2016002198A MX2016002198A MX2016002198A MX 2016002198 A MX2016002198 A MX 2016002198A MX 2016002198 A MX2016002198 A MX 2016002198A MX 2016002198 A MX2016002198 A MX 2016002198A MX 2016002198 A MX2016002198 A MX 2016002198A
- Authority
- MX
- Mexico
- Prior art keywords
- preparing
- compound
- preparation
- compounds
- useful
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 2
- 238000004519 manufacturing process Methods 0.000 title 1
- 101000777293 Homo sapiens Serine/threonine-protein kinase Chk1 Proteins 0.000 abstract 1
- 102100031081 Serine/threonine-protein kinase Chk1 Human genes 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Epidemiology (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
La invención proporciona procesos de preparación de los mismos útiles en la preparación de compuestos que se pueden utilizar como inhibidores de CHK1.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361868933P | 2013-08-22 | 2013-08-22 | |
| PCT/US2014/052146 WO2015027092A1 (en) | 2013-08-22 | 2014-08-21 | Process for preparing a compound |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| MX2016002198A true MX2016002198A (es) | 2016-09-08 |
| MX369174B MX369174B (es) | 2019-10-30 |
Family
ID=52484170
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2016002198A MX369174B (es) | 2013-08-22 | 2014-08-21 | Proceso para la preparación de un compuesto. |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US10329288B2 (es) |
| EP (1) | EP3036227B1 (es) |
| JP (1) | JP6463758B2 (es) |
| KR (1) | KR102325163B1 (es) |
| CN (1) | CN105705499B (es) |
| AR (1) | AR100020A1 (es) |
| CA (1) | CA2921956C (es) |
| MX (1) | MX369174B (es) |
| RU (1) | RU2672725C2 (es) |
| WO (1) | WO2015027092A1 (es) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MA41599A (fr) * | 2015-02-26 | 2018-01-02 | Array Biopharma Inc | Formes cristallines d'un composé pyrrolopyridine |
| CN109796349A (zh) * | 2019-03-01 | 2019-05-24 | 西南石油大学 | 一种还原芳香硝基化合物制备芳胺类化合物的方法 |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE69611443T2 (de) | 1995-05-19 | 2001-07-12 | Novartis Ag, Basel | Verfahren zur katalytischen hydrogenierung von aromatischen nitroverbindungen |
| AU784297C (en) * | 2000-06-26 | 2007-01-11 | Pfizer Products Inc. | Pyrrolo(2,3-d)pyrimidine compounds as immunosuppressive agents |
| WO2003028724A1 (en) | 2001-10-04 | 2003-04-10 | Smithkline Beecham Corporation | Chk1 kinase inhibitors |
| GB0330043D0 (en) * | 2003-12-24 | 2004-01-28 | Pharmacia Italia Spa | Pyrrolo [2,3-b] pyridine derivatives active as kinase inhibitors process for their preparation and pharmaceutical compositions comprising them |
| SE0401001D0 (sv) * | 2004-03-31 | 2004-03-31 | Astrazeneca Ab | Chemical process |
| AR054416A1 (es) * | 2004-12-22 | 2007-06-27 | Incyte Corp | Pirrolo [2,3-b]piridin-4-il-aminas y pirrolo [2,3-b]pirimidin-4-il-aminas como inhibidores de las quinasas janus. composiciones farmaceuticas. |
| CA2598639A1 (en) * | 2005-02-23 | 2006-08-31 | Coley Pharmaceutical Group, Inc. | Hydroxyalkyl substituted imidazonaphthyridines |
| US8163767B2 (en) * | 2005-07-14 | 2012-04-24 | Astellas Pharma Inc. | Heterocyclic Janus Kinase 3 inhibitors |
| EP2242755B1 (en) * | 2008-01-08 | 2012-09-12 | Array Biopharma, Inc. | Pyrrolopyridines as kinase inhibitors |
| ES2392014T3 (es) | 2008-01-09 | 2012-12-03 | Array Biopharma, Inc. | Pirazolopiridinas como inhibidores de la cinasa |
| CL2009001152A1 (es) * | 2008-05-13 | 2009-10-16 | Array Biopharma Inc | Compuestos derivados de n-(4-(cicloalquilo nitrogenado-1-il)-1h-pirrolo[2,3-b]piridin-3-il)amida, inhibidores de cinasa; proceso de preparacion; composicion farmaceutica; y su uso para el tratamiento de una enfermedad proliferativa. |
| HUE026671T2 (en) | 2011-08-18 | 2016-07-28 | Nippon Shinyaku Co Ltd | Heterocyclic derivatives as microsomal prostaglandin E synthetase inhibitors (mPGEs) |
| GB201201566D0 (en) * | 2012-01-30 | 2012-03-14 | Vernalis R&D Ltd | New chemical compounds |
-
2014
- 2014-08-21 MX MX2016002198A patent/MX369174B/es active IP Right Grant
- 2014-08-21 JP JP2016536458A patent/JP6463758B2/ja not_active Expired - Fee Related
- 2014-08-21 KR KR1020167007101A patent/KR102325163B1/ko not_active Expired - Fee Related
- 2014-08-21 RU RU2016110081A patent/RU2672725C2/ru active
- 2014-08-21 CA CA2921956A patent/CA2921956C/en active Active
- 2014-08-21 WO PCT/US2014/052146 patent/WO2015027092A1/en not_active Ceased
- 2014-08-21 CN CN201480054349.1A patent/CN105705499B/zh not_active Expired - Fee Related
- 2014-08-21 EP EP14838336.7A patent/EP3036227B1/en active Active
- 2014-08-21 US US14/913,635 patent/US10329288B2/en active Active
- 2014-08-22 AR ARP140103155A patent/AR100020A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN105705499A (zh) | 2016-06-22 |
| EP3036227B1 (en) | 2020-01-08 |
| KR20160043116A (ko) | 2016-04-20 |
| JP6463758B2 (ja) | 2019-02-06 |
| JP2016528296A (ja) | 2016-09-15 |
| RU2672725C2 (ru) | 2018-11-19 |
| CA2921956A1 (en) | 2015-02-26 |
| KR102325163B1 (ko) | 2021-11-11 |
| AR100020A1 (es) | 2016-09-07 |
| US10329288B2 (en) | 2019-06-25 |
| EP3036227A4 (en) | 2017-01-04 |
| CN105705499B (zh) | 2018-10-12 |
| US20160200723A1 (en) | 2016-07-14 |
| HK1222392A1 (zh) | 2017-06-30 |
| WO2015027092A1 (en) | 2015-02-26 |
| RU2016110081A (ru) | 2017-09-27 |
| MX369174B (es) | 2019-10-30 |
| EP3036227A1 (en) | 2016-06-29 |
| RU2016110081A3 (es) | 2018-05-18 |
| CA2921956C (en) | 2021-10-19 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant or registration |