MX2013006332A - Composiciones farmaceuticas orales para uso en dislipidemias. - Google Patents
Composiciones farmaceuticas orales para uso en dislipidemias.Info
- Publication number
- MX2013006332A MX2013006332A MX2013006332A MX2013006332A MX2013006332A MX 2013006332 A MX2013006332 A MX 2013006332A MX 2013006332 A MX2013006332 A MX 2013006332A MX 2013006332 A MX2013006332 A MX 2013006332A MX 2013006332 A MX2013006332 A MX 2013006332A
- Authority
- MX
- Mexico
- Prior art keywords
- oral pharmaceutical
- dyslipidemias
- pharmaceutical compositions
- levels
- producing
- Prior art date
Links
- 239000008203 oral pharmaceutical composition Substances 0.000 title abstract 2
- 208000032928 Dyslipidaemia Diseases 0.000 title 1
- XUKUURHRXDUEBC-KAYWLYCHSA-N Atorvastatin Chemical compound C=1C=CC=CC=1C1=C(C=2C=CC(F)=CC=2)N(CC[C@@H](O)C[C@@H](O)CC(O)=O)C(C(C)C)=C1C(=O)NC1=CC=CC=C1 XUKUURHRXDUEBC-KAYWLYCHSA-N 0.000 abstract 1
- XUKUURHRXDUEBC-UHFFFAOYSA-N Atorvastatin Natural products C=1C=CC=CC=1C1=C(C=2C=CC(F)=CC=2)N(CCC(O)CC(O)CC(O)=O)C(C(C)C)=C1C(=O)NC1=CC=CC=C1 XUKUURHRXDUEBC-UHFFFAOYSA-N 0.000 abstract 1
- 229940121710 HMGCoA reductase inhibitor Drugs 0.000 abstract 1
- 208000001145 Metabolic Syndrome Diseases 0.000 abstract 1
- 201000000690 abdominal obesity-metabolic syndrome Diseases 0.000 abstract 1
- 239000003524 antilipemic agent Substances 0.000 abstract 1
- 229960005370 atorvastatin Drugs 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- YMTINGFKWWXKFG-UHFFFAOYSA-N fenofibrate Chemical compound C1=CC(OC(C)(C)C(=O)OC(C)C)=CC=C1C(=O)C1=CC=C(Cl)C=C1 YMTINGFKWWXKFG-UHFFFAOYSA-N 0.000 abstract 1
- 229960002297 fenofibrate Drugs 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 239000007787 solid Substances 0.000 abstract 1
- 208000001072 type 2 diabetes mellitus Diseases 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/216—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Emergency Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
Abstract
La presente invención comprende una composición farmacéutica oral sólida que contiene una estatina y otro agente antilipidémico, así como un procedimiento para su preparación y el uso de dicha combinación para la elaboración de una formulación farmacéutica útil en el tratamiento de síndrome metabólico, diabetes tipo II, u otras enfermedades. La invención también se refiere al uso de una combinación farmacéutica formada por atorvastatina y fenofibrato, para preparar un medicamento útil para elevar los niveles de HDL2a y HDL2b, y para disminuir los niveles de HDL3a, HDL3b y HDL3c.
Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| MX2013006332A MX2013006332A (es) | 2013-06-05 | 2013-06-05 | Composiciones farmaceuticas orales para uso en dislipidemias. |
| PCT/IB2014/061987 WO2014195900A2 (es) | 2013-06-05 | 2014-06-05 | Composiciones farmacéuticas orales para uso en dislipidemias |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| MX2013006332A MX2013006332A (es) | 2013-06-05 | 2013-06-05 | Composiciones farmaceuticas orales para uso en dislipidemias. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2013006332A true MX2013006332A (es) | 2014-12-19 |
Family
ID=52008666
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2013006332A MX2013006332A (es) | 2013-06-05 | 2013-06-05 | Composiciones farmaceuticas orales para uso en dislipidemias. |
Country Status (2)
| Country | Link |
|---|---|
| MX (1) | MX2013006332A (es) |
| WO (1) | WO2014195900A2 (es) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2022071787A1 (es) | 2020-09-29 | 2022-04-07 | Laboratorios Silanes S.A. De C.V. | Combinaciones farmacéuticas de estatinas y fibratos para el tratamiento y prevención de hiperlipidemias y enfermedades cardiovasculares |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8293277B2 (en) * | 1998-10-01 | 2012-10-23 | Alkermes Pharma Ireland Limited | Controlled-release nanoparticulate compositions |
| GR990100388A (el) * | 1999-11-09 | 2001-07-31 | Φαρμακευτικος συνδυασμος αποτελουμενος απο χωριστες δοσολογικες μορφες σε συσκευασια συμμορφωσης (compliance package) ενος αναστολεα της αναγωγασης του υδροξυ-μεθυλο-γλουταρυλο συνενζυμου α (στατινης, statin) και ενος παραγωγου του φιμπρικου οξεος.... | |
| WO2002024169A1 (en) * | 2000-09-20 | 2002-03-28 | Skyepharma Canada Inc. | Spray drying process and compositions of fenofibrate |
| US20070014846A1 (en) * | 2003-10-10 | 2007-01-18 | Lifecycle Pharma A/S | Pharmaceutical compositions comprising fenofibrate and atorvastatin |
| CA2555316A1 (en) * | 2004-02-09 | 2005-08-18 | Aska Pharmaceutical Co., Ltd. | Combined pharmaceutical composition |
| WO2006134604A1 (en) * | 2005-06-15 | 2006-12-21 | Hetero Drugs Limited | Combination composition of cholesterol absorption inhibitor and 3-hydroxy-3-methylglutaryl-coenzyme a (hmg-coa) reductase inhibitor |
| JP2011521992A (ja) * | 2008-06-06 | 2011-07-28 | ニコックス エス エイ | アトルバスタチン4−(ニトロキシ)ブチルエステルおよび脂質低下剤を含む組成物 |
| WO2011002422A2 (en) * | 2009-07-02 | 2011-01-06 | Bilgic Mahmut | Solubility enhancing pharmaceutical formulation |
-
2013
- 2013-06-05 MX MX2013006332A patent/MX2013006332A/es unknown
-
2014
- 2014-06-05 WO PCT/IB2014/061987 patent/WO2014195900A2/es not_active Ceased
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2022071787A1 (es) | 2020-09-29 | 2022-04-07 | Laboratorios Silanes S.A. De C.V. | Combinaciones farmacéuticas de estatinas y fibratos para el tratamiento y prevención de hiperlipidemias y enfermedades cardiovasculares |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2014195900A3 (es) | 2015-02-05 |
| WO2014195900A2 (es) | 2014-12-11 |
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