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MX2013002261A - N-fenetiltriazolonacetamidas sustituidas y su uso. - Google Patents

N-fenetiltriazolonacetamidas sustituidas y su uso.

Info

Publication number
MX2013002261A
MX2013002261A MX2013002261A MX2013002261A MX2013002261A MX 2013002261 A MX2013002261 A MX 2013002261A MX 2013002261 A MX2013002261 A MX 2013002261A MX 2013002261 A MX2013002261 A MX 2013002261A MX 2013002261 A MX2013002261 A MX 2013002261A
Authority
MX
Mexico
Prior art keywords
phenethyltriazoloneacetamides
prevention
treatment
substituted
diseases
Prior art date
Application number
MX2013002261A
Other languages
English (en)
Inventor
Joerg Keldenich
Peter Kolkhof
Carsten Schmeck
Martina Delbeck
Chantal Fuerstner
Axel Kretschmer
Elisabeth Pook
Hubert Truebel
Original Assignee
Bayer Ip Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ip Gmbh filed Critical Bayer Ip Gmbh
Publication of MX2013002261A publication Critical patent/MX2013002261A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4196—1,2,4-Triazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D249/12—Oxygen or sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Hospice & Palliative Care (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

La presente solicitud se refiere a N-fenetiltriazolonacetamidas sustituidas novedosas, a procedimientos para prepararlas, a su uso solas o en combinaciones para el tratamiento y/o la prevención de enfermedades y también a su uso para la producción de medicamentos para el tratamiento y/o la prevención de enfermedades, más en particular para el tratamiento y/o la prevención de trastornos cardiovasculares.
MX2013002261A 2010-09-02 2011-08-31 N-fenetiltriazolonacetamidas sustituidas y su uso. MX2013002261A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102010040187A DE102010040187A1 (de) 2010-09-02 2010-09-02 Substituierte N-Phenethyl-triazolonacetamide und ihre Verwendung
PCT/EP2011/065000 WO2012028644A1 (de) 2010-09-02 2011-08-31 Substituierte n-phenethyl-triazolonacetamide und ihre verwendung

Publications (1)

Publication Number Publication Date
MX2013002261A true MX2013002261A (es) 2013-05-22

Family

ID=44653279

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2013002261A MX2013002261A (es) 2010-09-02 2011-08-31 N-fenetiltriazolonacetamidas sustituidas y su uso.

Country Status (14)

Country Link
US (1) US9180120B2 (es)
EP (1) EP2619188B1 (es)
JP (1) JP5816284B2 (es)
KR (1) KR20130138216A (es)
CN (1) CN103370309A (es)
AU (1) AU2011298391A1 (es)
BR (1) BR112013005226A2 (es)
CA (1) CA2809716A1 (es)
DE (1) DE102010040187A1 (es)
ES (1) ES2543750T3 (es)
MX (1) MX2013002261A (es)
RU (1) RU2013114413A (es)
WO (1) WO2012028644A1 (es)
ZA (1) ZA201302335B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102010040924A1 (de) 2010-09-16 2012-03-22 Bayer Schering Pharma Aktiengesellschaft Substituierte Phenylacet- und Phenylpropanamide und ihre Verwendung
CN107074783B (zh) 2014-11-03 2020-06-05 拜耳制药股份公司 羟烷基取代的苯基三唑衍生物及其用途
WO2017191117A1 (en) 2016-05-03 2017-11-09 Bayer Pharma Aktiengesellschaft V1a receptor antagonists for use in the treatment of renal diseases
US9988367B2 (en) 2016-05-03 2018-06-05 Bayer Pharma Aktiengesellschaft Amide-substituted pyridinyltriazole derivatives and uses thereof
KR102390194B1 (ko) * 2020-08-03 2022-04-25 셀라이온바이오메드 주식회사 페닐알킬 카바메이트 화합물을 포함하는 Kca3.1채널 매개질환 치료용 조성물

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Also Published As

Publication number Publication date
ES2543750T3 (es) 2015-08-21
AU2011298391A8 (en) 2013-06-13
BR112013005226A2 (pt) 2016-05-03
JP2013538806A (ja) 2013-10-17
US9180120B2 (en) 2015-11-10
JP5816284B2 (ja) 2015-11-18
ZA201302335B (en) 2015-11-25
WO2012028644A1 (de) 2012-03-08
EP2619188A1 (de) 2013-07-31
US20130225646A1 (en) 2013-08-29
AU2011298391A1 (en) 2013-03-14
RU2013114413A (ru) 2014-10-10
CN103370309A (zh) 2013-10-23
KR20130138216A (ko) 2013-12-18
DE102010040187A1 (de) 2012-03-08
CA2809716A1 (en) 2012-03-08
EP2619188B1 (de) 2015-05-06

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal