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MX2012013021A - Formulaciones resistentes a alcohol. - Google Patents

Formulaciones resistentes a alcohol.

Info

Publication number
MX2012013021A
MX2012013021A MX2012013021A MX2012013021A MX2012013021A MX 2012013021 A MX2012013021 A MX 2012013021A MX 2012013021 A MX2012013021 A MX 2012013021A MX 2012013021 A MX2012013021 A MX 2012013021A MX 2012013021 A MX2012013021 A MX 2012013021A
Authority
MX
Mexico
Prior art keywords
alcohol
dosage form
resistant formulations
resistance
lipid
Prior art date
Application number
MX2012013021A
Other languages
English (en)
Inventor
Ehab Hamed
Original Assignee
Cima Labs Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cima Labs Inc filed Critical Cima Labs Inc
Publication of MX2012013021A publication Critical patent/MX2012013021A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A61K9/2081Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5036Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • A61K9/5042Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
    • A61K9/5047Cellulose ethers containing no ester groups, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Preparation (AREA)

Abstract

La presente descripción se refiere a una forma de dosis oral de liberación prolongada que comprende una matriz que contiene un modificador de viscosidad (pero sin lípidos) y gránulos revestidos que contienen un fármaco en alta dosis, altamente soluble en agua. La forma de dosis tiene resistencia al alcohol y también puede tener resistencia a trituración.
MX2012013021A 2010-05-11 2011-05-09 Formulaciones resistentes a alcohol. MX2012013021A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US33352110P 2010-05-11 2010-05-11
PCT/US2011/035767 WO2011143118A2 (en) 2010-05-11 2011-05-09 Alcohol-resistant formulations

Publications (1)

Publication Number Publication Date
MX2012013021A true MX2012013021A (es) 2012-12-17

Family

ID=44344024

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2012013021A MX2012013021A (es) 2010-05-11 2011-05-09 Formulaciones resistentes a alcohol.

Country Status (10)

Country Link
US (2) US20130202705A1 (es)
EP (1) EP2568969A2 (es)
JP (1) JP5894720B2 (es)
CN (1) CN102883713B (es)
AU (1) AU2011253216B2 (es)
CA (1) CA2798700C (es)
IL (1) IL222637A (es)
MX (1) MX2012013021A (es)
NZ (1) NZ603531A (es)
WO (1) WO2011143118A2 (es)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20130143867A1 (en) 2011-12-02 2013-06-06 Sychroneuron Inc. Acamprosate formulations, methods of using the same, and combinations comprising the same
CN103893146A (zh) * 2012-12-25 2014-07-02 天津药物研究院 含福多司坦缓释剂型
CA2914365C (en) * 2013-06-05 2022-03-15 Synchroneuron, Inc. Acamprosate formulations, methods of using the same, and combinations comprising the same
US9561187B1 (en) * 2014-02-03 2017-02-07 CMAX Technologies, Inc. Sustained release metoprolol formulations
HUE065006T2 (hu) 2014-07-03 2024-04-28 SpecGx LLC Nem-cellulóz poliszacharidokat tartalmazó, visszaélés-gátló, azonnali felszabadulású készítmények
US20180344649A1 (en) 2015-09-29 2018-12-06 Acorda Therapeutics, Inc. Sustained release compositions of 4-aminopyridine
US10736855B2 (en) 2016-02-25 2020-08-11 Dexcel Pharma Technologies Ltd. Compositions comprising proton pump inhibitors
AR113993A1 (es) 2017-12-21 2020-07-08 Faes Farma Sa Formulación una vez al día de hidrosmina
CN110812337B (zh) * 2018-08-08 2022-04-12 上海宣泰医药科技股份有限公司 一种通过流化床制粒法制备氨基己酸片剂的方法
CN110812332B (zh) * 2018-08-10 2022-09-02 北京普德康利医药科技发展有限公司 一种双氯芬酸钠咽部滞留颗粒
WO2020068510A1 (en) 2018-09-25 2020-04-02 SpecGx LLC Abuse deterrent immediate release capsule dosage forms
US12303604B1 (en) 2024-10-16 2025-05-20 Currax Pharmaceuticals Llc Pharmaceutical formulations comprising naltrexone and/or bupropion

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE8703881D0 (sv) * 1987-10-08 1987-10-08 Haessle Ab New pharmaceutical preparation
US5223264A (en) 1989-10-02 1993-06-29 Cima Labs, Inc. Pediatric effervescent dosage form
US5178878A (en) 1989-10-02 1993-01-12 Cima Labs, Inc. Effervescent dosage form with microparticles
US6024981A (en) 1997-04-16 2000-02-15 Cima Labs Inc. Rapidly dissolving robust dosage form
WO2005034923A1 (en) * 2003-10-10 2005-04-21 Ethypharm Sustained-release microgranules containing gingko biloba extract and the process for manufacturing these
US20070092573A1 (en) * 2005-10-24 2007-04-26 Laxminarayan Joshi Stabilized extended release pharmaceutical compositions comprising a beta-adrenoreceptor antagonist
WO2007048223A2 (en) * 2005-10-25 2007-05-03 Pharmascience Inc. A gastric retention drug delivery system
US20080069891A1 (en) * 2006-09-15 2008-03-20 Cima Labs, Inc. Abuse resistant drug formulation
JP2008007293A (ja) * 2006-06-30 2008-01-17 Komori Corp 搬送装置
US8445018B2 (en) 2006-09-15 2013-05-21 Cima Labs Inc. Abuse resistant drug formulation
HUE032012T2 (en) * 2007-09-13 2017-08-28 Cima Labs Inc Anti-Abuse Drug Products

Also Published As

Publication number Publication date
WO2011143118A2 (en) 2011-11-17
EP2568969A2 (en) 2013-03-20
WO2011143118A3 (en) 2012-07-05
CA2798700C (en) 2018-08-21
JP2013526521A (ja) 2013-06-24
US20190133924A1 (en) 2019-05-09
AU2011253216B2 (en) 2016-10-20
NZ603531A (en) 2014-08-29
IL222637A0 (en) 2012-12-31
CN102883713A (zh) 2013-01-16
CA2798700A1 (en) 2011-11-17
AU2011253216A1 (en) 2012-11-29
IL222637A (en) 2017-04-30
CN102883713B (zh) 2016-08-03
US20130202705A1 (en) 2013-08-08
JP5894720B2 (ja) 2016-03-30

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