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MX2009007255A - Sintesis de estereoisomeros seleccionados de ciertos alcoholes sustituidos. - Google Patents

Sintesis de estereoisomeros seleccionados de ciertos alcoholes sustituidos.

Info

Publication number
MX2009007255A
MX2009007255A MX2009007255A MX2009007255A MX2009007255A MX 2009007255 A MX2009007255 A MX 2009007255A MX 2009007255 A MX2009007255 A MX 2009007255A MX 2009007255 A MX2009007255 A MX 2009007255A MX 2009007255 A MX2009007255 A MX 2009007255A
Authority
MX
Mexico
Prior art keywords
synthesis
stereoisomeric
certain substituted
substituted alcohols
selected stereoisomers
Prior art date
Application number
MX2009007255A
Other languages
English (en)
Inventor
Arthur E Harms
Original Assignee
Baush & Lomb Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Baush & Lomb Inc filed Critical Baush & Lomb Inc
Publication of MX2009007255A publication Critical patent/MX2009007255A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Un proceso para producir un esteroisómero seleccionado de un alcohol sustituido comprende hacer reaccionar una amina estereoisomérica con un compuesto heterocíclico sustituido por halógeno o una cetona o aldehído estereoisomérico con un compuesto heterocíclico sustituido por amino. El proceso evita la producción de una mezcla racémica de estereoisómeros de la técnica anterior. Este alcohol sustituido estereoisomérico se puede utilizar para la terapia anti-inflamatoria.
MX2009007255A 2007-01-12 2008-01-08 Sintesis de estereoisomeros seleccionados de ciertos alcoholes sustituidos. MX2009007255A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11/652,767 US20080171873A1 (en) 2007-01-12 2007-01-12 Synthesis of selected stereoisomers of certain substituted alcohols
PCT/US2008/050470 WO2008088969A2 (en) 2007-01-12 2008-01-08 Synthesis of selected stereoisomers of certain substituted alcohols

Publications (1)

Publication Number Publication Date
MX2009007255A true MX2009007255A (es) 2009-08-12

Family

ID=39522056

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2009007255A MX2009007255A (es) 2007-01-12 2008-01-08 Sintesis de estereoisomeros seleccionados de ciertos alcoholes sustituidos.

Country Status (8)

Country Link
US (1) US20080171873A1 (es)
EP (1) EP2121670A2 (es)
JP (1) JP2010515741A (es)
KR (1) KR20090097928A (es)
CN (1) CN101578281A (es)
BR (1) BRPI0806303A2 (es)
MX (1) MX2009007255A (es)
WO (1) WO2008088969A2 (es)

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6856215B2 (en) * 2001-08-24 2005-02-15 Powerwave Technologies, Inc. System and method for adjusting group delay
US6897224B2 (en) * 2002-04-02 2005-05-24 Schering Ag Quinoline and isoquinoline derivatives, a process for their production and their use as inflammation inhibitors
DE10215316C1 (de) * 2002-04-02 2003-12-18 Schering Ag Chinolin- und Isochinolin-Derivate, ein pharmazeutisches Mittel und ihre Verwendung als Entzündungshemmer
DE10330358A1 (de) * 2003-07-01 2005-02-03 Schering Ag Heterozyklisch substituierte Pentanol-Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Entzündungshemmer
US20050090559A1 (en) * 2003-07-01 2005-04-28 Markus Berger Heterocyclically-substituted pentanol derivatives, process for their production and their use as anti-inflammatory agents
US7256300B2 (en) * 2004-03-30 2007-08-14 Boehringer Ingelheim Pharmaceuticals, Inc. Stereoselective synthesis of certain trifluoromethyl-substituted alcohols
DE102005020331A1 (de) * 2005-04-26 2006-11-02 Schering Ag 5-substituierte Chinolin- und Isochinolin-Derivate, ein Verfahren zu ihrer Herstellung und ihre Verwendung als Entzündungshemmer
US7417056B2 (en) * 2004-11-12 2008-08-26 Schering Ag 5-substituted quinoline and isoquinoline derivatives, a process for their production and their use as anti-inflammatory agents
US8093281B2 (en) * 2005-04-14 2012-01-10 Glaxo Group Limited Indazoles as glucocorticoid receptor ligands
US7071356B1 (en) * 2005-12-01 2006-07-04 Isp Investments Inc. Process for the preparation of 1-(aminomethyl) cyclohexaneacetic acid

Also Published As

Publication number Publication date
WO2008088969A3 (en) 2008-12-11
EP2121670A2 (en) 2009-11-25
US20080171873A1 (en) 2008-07-17
JP2010515741A (ja) 2010-05-13
BRPI0806303A2 (pt) 2011-09-06
CN101578281A (zh) 2009-11-11
KR20090097928A (ko) 2009-09-16
WO2008088969A2 (en) 2008-07-24

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal