MA28841B1 - Analogues tetrapeptidiques - Google Patents
Analogues tetrapeptidiquesInfo
- Publication number
- MA28841B1 MA28841B1 MA29613A MA29613A MA28841B1 MA 28841 B1 MA28841 B1 MA 28841B1 MA 29613 A MA29613 A MA 29613A MA 29613 A MA29613 A MA 29613A MA 28841 B1 MA28841 B1 MA 28841B1
- Authority
- MA
- Morocco
- Prior art keywords
- tetrapeptitiic
- analogs
- tetrapeptitiic analogs
- Prior art date
Links
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- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/10—Tetrapeptides
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- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
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- C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
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- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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| MA28841B1 true MA28841B1 (fr) | 2007-09-03 |
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| MA29613A MA28841B1 (fr) | 2004-07-12 | 2007-01-10 | Analogues tetrapeptidiques |
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| EP (3) | EP2457896A1 (fr) |
| JP (2) | JP2008505976A (fr) |
| KR (1) | KR20070043831A (fr) |
| AU (1) | AU2005271831A1 (fr) |
| BR (1) | BRPI0513310A (fr) |
| CA (1) | CA2573644A1 (fr) |
| CR (1) | CR8919A (fr) |
| EA (1) | EA200700225A1 (fr) |
| GB (1) | GB2430935A (fr) |
| IL (1) | IL180677A0 (fr) |
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| MX (1) | MX2007000490A (fr) |
| NO (1) | NO20070782L (fr) |
| TN (1) | TNSN07005A1 (fr) |
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| CN101029080A (zh) * | 2001-11-21 | 2007-09-05 | 伯纳姆研究院 | 用于对iap抑制卡斯蛋白酶进行去阻遏的方法及组合物 |
| WO2003065987A2 (fr) * | 2002-02-04 | 2003-08-14 | Merck & Co., Inc. | Inhibiteurs de granzyme b |
| US7838496B2 (en) * | 2003-05-02 | 2010-11-23 | Polyphor Ag/Ltd. | Template-fixed peptidomimetics as medicaments against HIV and cancer |
| CA2553874A1 (fr) * | 2004-01-16 | 2005-08-04 | The Regents Of The University Of Michigan | Mimetiques de smac contraints de maniere conformationnelle et utilisations associees |
| PT1778718E (pt) * | 2004-07-02 | 2014-12-03 | Genentech Inc | Inibidores de iap |
-
2005
- 2005-07-12 EA EA200700225A patent/EA200700225A1/ru unknown
- 2005-07-12 US US11/632,441 patent/US20100190688A1/en not_active Abandoned
- 2005-07-12 WO PCT/US2005/024700 patent/WO2006017295A2/fr not_active Ceased
- 2005-07-12 CA CA002573644A patent/CA2573644A1/fr not_active Abandoned
- 2005-07-12 MX MX2007000490A patent/MX2007000490A/es unknown
- 2005-07-12 BR BRPI0513310-6A patent/BRPI0513310A/pt not_active Application Discontinuation
- 2005-07-12 EP EP11184402A patent/EP2457896A1/fr not_active Withdrawn
- 2005-07-12 AU AU2005271831A patent/AU2005271831A1/en not_active Abandoned
- 2005-07-12 JP JP2007521572A patent/JP2008505976A/ja active Pending
- 2005-07-12 EP EP05771672A patent/EP1773348A4/fr not_active Withdrawn
- 2005-07-12 EP EP11184396A patent/EP2457895A1/fr not_active Withdrawn
- 2005-07-12 KR KR1020077003279A patent/KR20070043831A/ko not_active Ceased
-
2007
- 2007-01-10 MA MA29613A patent/MA28841B1/fr unknown
- 2007-01-11 IL IL180677A patent/IL180677A0/en unknown
- 2007-01-11 TN TNP2007000005A patent/TNSN07005A1/fr unknown
- 2007-01-12 ZA ZA2007/00357A patent/ZA200700357B/en unknown
- 2007-01-12 GB GB0700629A patent/GB2430935A/en not_active Withdrawn
- 2007-02-09 NO NO20070782A patent/NO20070782L/no not_active Application Discontinuation
- 2007-02-12 CR CR8919A patent/CR8919A/es not_active Application Discontinuation
-
2011
- 2011-01-06 JP JP2011000916A patent/JP2011102312A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| TNSN07005A1 (fr) | 2008-06-02 |
| BRPI0513310A (pt) | 2008-05-06 |
| GB0700629D0 (en) | 2007-02-21 |
| WO2006017295A2 (fr) | 2006-02-16 |
| US20100190688A1 (en) | 2010-07-29 |
| WO2006017295A3 (fr) | 2007-07-12 |
| GB2430935A (en) | 2007-04-11 |
| MX2007000490A (es) | 2007-06-11 |
| NO20070782L (no) | 2007-04-02 |
| ZA200700357B (en) | 2008-11-26 |
| AU2005271831A1 (en) | 2006-02-16 |
| IL180677A0 (en) | 2008-04-13 |
| EP2457895A1 (fr) | 2012-05-30 |
| EP2457896A1 (fr) | 2012-05-30 |
| JP2008505976A (ja) | 2008-02-28 |
| KR20070043831A (ko) | 2007-04-25 |
| CR8919A (es) | 2007-08-31 |
| CA2573644A1 (fr) | 2006-02-16 |
| JP2011102312A (ja) | 2011-05-26 |
| EA200700225A1 (ru) | 2008-02-28 |
| EP1773348A4 (fr) | 2009-05-20 |
| EP1773348A2 (fr) | 2007-04-18 |
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